Structure-Activity Relationship of Fluorinated Sialic Acid Inhibitors for Bacterial Sialylation.

Haemophilus influenzae / drug effects Halogenation N-Acetylneuraminic Acid / chemistry Structure-Activity Relationship

Journal

Bioconjugate chemistry
ISSN: 1520-4812
Titre abrégé: Bioconjug Chem
Pays: United States
ID NLM: 9010319

Informations de publication

Date de publication:
16 06 2021
Historique:
pubmed: 28 5 2021
medline: 28 8 2021
entrez: 27 5 2021
Statut: ppublish

Résumé

Bacterial pathogens such as Nontypeable

Identifiants

DOI: 10.1021/acs.bioconjchem.1c00194 PMID: 34043338 PMC: PMC8382218
pubmed: 34043338
doi: 10.1021/acs.bioconjchem.1c00194
pmc: PMC8382218
doi:

Substances chimiques

N-Acetylneuraminic Acid GZP2782OP0

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

1047-1051

Références

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Auteurs

Sam J Moons (SJ)

Cluster of Molecular Chemistry, Institute for Molecules and Materials, Radboud University Nijmegen, Nijmegen 6525 AJ, The Netherlands.

Emiel Rossing (E)

Cluster of Molecular Chemistry, Institute for Molecules and Materials, Radboud University Nijmegen, Nijmegen 6525 AJ, The Netherlands.

Jurriaan J A Heming (JJA)

Cluster of Molecular Chemistry, Institute for Molecules and Materials, Radboud University Nijmegen, Nijmegen 6525 AJ, The Netherlands.

Mathilde A C H Janssen (MACH)

Cluster of Molecular Chemistry, Institute for Molecules and Materials, Radboud University Nijmegen, Nijmegen 6525 AJ, The Netherlands.

Monique van Scherpenzeel (M)

Translational Metabolic Laboratory, Department of Neurology, Donders Center for Brain Cognition and Behavior, Radboud University Medical Center, Nijmegen 6525 GA, The Netherlands.

Dirk J Lefeber (DJ)

Translational Metabolic Laboratory, Department of Neurology, Donders Center for Brain Cognition and Behavior, Radboud University Medical Center, Nijmegen 6525 GA, The Netherlands.

Marien I de Jonge (MI)

Laboratory of Medical Immunology, Radboud Center for Infectious Diseases, Radboud Institute for Molecular Sciences, Radboud University Medical Center, Nijmegen 6525 GA, The Netherlands.

Jeroen D Langereis (JD)

Laboratory of Medical Immunology, Radboud Center for Infectious Diseases, Radboud Institute for Molecular Sciences, Radboud University Medical Center, Nijmegen 6525 GA, The Netherlands.

Thomas J Boltje (TJ)

Cluster of Molecular Chemistry, Institute for Molecules and Materials, Radboud University Nijmegen, Nijmegen 6525 AJ, The Netherlands.
ORCID: 0000-0001-9141-8784

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Classifications MeSH

questionsmedicales.fr › Bactéries › Proteobacteria › Gammaproteobacteria › Pasteurellaceae › Haemophilus › Haemophilus influenzae › Structure-Activity Relationship of Fluorinated...
questionsmedicales.fr › Métabolisme › Halogénation › Structure-Activity Relationship of Fluorinated...
questionsmedicales.fr › Glucides › Oses acides › Acides neuraminiques › Acides sialiques › Acide N-acétyl-neuraminique › Structure-Activity Relationship of Fluorinated...
questionsmedicales.fr › Phénomènes physiologiques › Phénomènes pharmacologiques et toxicologiques › Phénomènes pharmacologiques › Relation structure-activité › Structure-Activity Relationship of Fluorinated...