Noscapine Acts as a Protease Inhibitor of In Vitro Elastase-Induced Collagen Deposition in Equine Endometrium.
Animals
Collagen
/ metabolism
Collagen Type I
/ drug effects
Endometriosis
/ drug therapy
Endometrium
/ drug effects
Estrous Cycle
Extracellular Traps
/ metabolism
Female
Fibrosis
Horse Diseases
/ pathology
Horses
Noscapine
/ metabolism
Pancreatic Elastase
/ metabolism
Protease Inhibitors
/ pharmacology
collagen
elastase
endometrosis
equine
fibrosis
inhibition
noscapine
Journal
International journal of molecular sciences
ISSN: 1422-0067
Titre abrégé: Int J Mol Sci
Pays: Switzerland
ID NLM: 101092791
Informations de publication
Date de publication:
19 May 2021
19 May 2021
Historique:
received:
16
04
2021
revised:
07
05
2021
accepted:
17
05
2021
entrez:
2
6
2021
pubmed:
3
6
2021
medline:
3
7
2021
Statut:
epublish
Résumé
Endometrosis is a reproductive pathology that is responsible for mare infertility. Our recent studies have focused on the involvement of neutrophil extracellular traps enzymes, such as elastase (ELA), in the development of equine endometrosis. Noscapine (NOSC) is an alkaloid derived from poppy opium with anticough, antistroke, anticancer, and antifibrotic properties. The present work investigates the putative inhibitory in vitro effect of NOSC on collagen type I alpha 2 chain (
Identifiants
pubmed: 34069423
pii: ijms22105333
doi: 10.3390/ijms22105333
pmc: PMC8159119
pii:
doi:
Substances chimiques
Collagen Type I
0
Protease Inhibitors
0
Noscapine
8V32U4AOQU
Collagen
9007-34-5
Pancreatic Elastase
EC 3.4.21.36
Types de publication
Journal Article
Langues
eng
Sous-ensembles de citation
IM
Subventions
Organisme : Narodowa Agencja Wymiany Akademickiej
ID : PPN/BIL/2018/1/00250/U/0001
Organisme : Fundação para a Ciência e a Tecnologia
ID : UIDB/00276/2020
Organisme : Fundação para a Ciência e a Tecnologia
ID : PTDC/CVT-REP/4202/2014
Organisme : Fundação para a Ciência e a Tecnologia
ID : SFRH/BD/101058/2014
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