Hybrids as NO Donors.


Journal

International journal of molecular sciences
ISSN: 1422-0067
Titre abrégé: Int J Mol Sci
Pays: Switzerland
ID NLM: 101092791

Informations de publication

Date de publication:
10 Sep 2021
Historique:
received: 29 07 2021
revised: 08 09 2021
accepted: 08 09 2021
entrez: 28 9 2021
pubmed: 29 9 2021
medline: 25 2 2023
Statut: epublish

Résumé

Cinnamic acid and its derivatives have been studied for a variety of biological properties, including anti-inflammatory, antioxidant, anticancer, antihypertensive, and antibacterial. Many hybrids of cinnamic derivatives with other bioactive molecules have been synthesized and evaluated as nitric oxide (NO) donors. Since NO plays a significant role in various biological processes, including vasodilation, inflammation, and neurotransmission, NO donor groups are incorporated into the structures of already-known bioactive molecules to enhance their biological properties. In this review, we present cinnamic hybrids with NO-donating ability useful in the treatment of several diseases.

Identifiants

pubmed: 34575950
pii: ijms22189788
doi: 10.3390/ijms22189788
pmc: PMC8469192
pii:
doi:

Substances chimiques

Cinnamates 0
cinnamic acid 140-10-3
Nitric Oxide 31C4KY9ESH

Types de publication

Journal Article Review

Langues

eng

Sous-ensembles de citation

IM

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Auteurs

Ioanna-Chrysoula Tsopka (IC)

Department of Pharmaceutical Chemistry, School of Pharmacy, Faculty of Health Sciences, Aristotle University of Thessaloniki, 54124 Thessaloniki, Greece.

Dimitra Hadjipavlou-Litina (D)

Department of Pharmaceutical Chemistry, School of Pharmacy, Faculty of Health Sciences, Aristotle University of Thessaloniki, 54124 Thessaloniki, Greece.

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Classifications MeSH