Sequential Injection Analysis for Automation and Evaluation of Drug Liberation Profiles: Clotrimazole Liberation Monitoring.


Journal

Molecules (Basel, Switzerland)
ISSN: 1420-3049
Titre abrégé: Molecules
Pays: Switzerland
ID NLM: 100964009

Informations de publication

Date de publication:
12 Sep 2021
Historique:
received: 23 08 2021
revised: 06 09 2021
accepted: 09 09 2021
entrez: 28 9 2021
pubmed: 29 9 2021
medline: 1 12 2021
Statut: epublish

Résumé

A fully automated sequential injection system was tested in terms of its application in liberation testing, and capabilities and limitations were discussed for clotrimazole liberation from three semisolid formulations. An evaluation based on kinetic profiles obtained in short and longer sampling intervals and steady-state flux values were applied as traditional methods. The obtained clotrimazole liberation profile was faster in the case of Delcore and slower for Clotrimazol AL and Canesten cream commercial formulations. The steady-state flux values for the tested formulations were 52 µg cm

Identifiants

pubmed: 34577009
pii: molecules26185538
doi: 10.3390/molecules26185538
pmc: PMC8467677
pii:
doi:

Substances chimiques

Antifungal Agents 0
Clotrimazole G07GZ97H65

Types de publication

Evaluation Study Journal Article

Langues

eng

Sous-ensembles de citation

IM

Subventions

Organisme : Ministerstvo Školství, Mládeže a Tělovýchovy
ID : CZ.02.1.01/0.0/0.0/15_003/0000465
Organisme : Univerzita Karlova v Praze
ID : SVV 260 548
Organisme : International Visegrad Fund
ID : 21930006

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Auteurs

Hana Sklenářová (H)

Department of Analytical Chemistry, Faculty of Pharmacy in Hradec Králové, Charles University, 500 05 Hradec Králové, Czech Republic.

Marek Beran (M)

Department of Analytical Chemistry, Faculty of Pharmacy in Hradec Králové, Charles University, 500 05 Hradec Králové, Czech Republic.

Lucie Novosvětská (L)

Department of Analytical Chemistry, Faculty of Pharmacy in Hradec Králové, Charles University, 500 05 Hradec Králové, Czech Republic.

Daniela Šmejkalová (D)

Contipro a.s., 561 02 Dolní Dobrouč, Czech Republic.

Petr Solich (P)

Department of Analytical Chemistry, Faculty of Pharmacy in Hradec Králové, Charles University, 500 05 Hradec Králové, Czech Republic.

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Classifications MeSH