The Transition of Photoreceptor Guanylate Cyclase Type 1 to the Active State.
GCAP
cGMP
calcium-binding proteins
guanylate cyclase
molecular-dynamics simulation
phototransduction
protein geometry
retina
retinal degeneration
vision
Journal
International journal of molecular sciences
ISSN: 1422-0067
Titre abrégé: Int J Mol Sci
Pays: Switzerland
ID NLM: 101092791
Informations de publication
Date de publication:
05 Apr 2022
05 Apr 2022
Historique:
received:
22
02
2022
accepted:
02
04
2022
entrez:
12
4
2022
pubmed:
13
4
2022
medline:
14
4
2022
Statut:
epublish
Résumé
Membrane-bound guanylate cyclases (GCs), which synthesize the second messenger guanosine-3', 5'-cyclic monophosphate, differ in their activation modes to reach the active state. Hormone peptides bind to the extracellular domain in hormone-receptor-type GCs and trigger a conformational change in the intracellular, cytoplasmic part of the enzyme. Sensory GCs that are present in rod and cone photoreceptor cells have intracellular binding sites for regulatory Ca
Identifiants
pubmed: 35409388
pii: ijms23074030
doi: 10.3390/ijms23074030
pmc: PMC8999790
pii:
doi:
Substances chimiques
Guanylate Cyclase-Activating Proteins
0
Hormones
0
Guanylate Cyclase
EC 4.6.1.2
Alanine
OF5P57N2ZX
Types de publication
Journal Article
Langues
eng
Sous-ensembles de citation
IM
Subventions
Organisme : Deutsche Forschungsgemeinschaft
ID : GRK1885
Organisme : Deutsche Forschungsgemeinschaft
ID : SFB1372
Organisme : Volkswagen Foundation
ID : Lichtenberg Professorship
Organisme : MWK Lower Saxony
ID : SMART
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