Combination of IM-Based Approaches to Unravel the Coexistence of Two Conformers on a Therapeutic Multispecific mAb.


Journal

Analytical chemistry
ISSN: 1520-6882
Titre abrégé: Anal Chem
Pays: United States
ID NLM: 0370536

Informations de publication

Date de publication:
07 06 2022
Historique:
pubmed: 24 5 2022
medline: 9 6 2022
entrez: 23 5 2022
Statut: ppublish

Résumé

Multispecific antibodies, which target multiple antigens at once, are emerging as promising therapeutic entities to offer more effective treatment than conventional monoclonal antibodies (mAbs). However, these highly complex mAb formats pose significant analytical challenges. We report here on the characterization of a trispecific antibody (tsAb), which presents two isomeric forms clearly separated and identified with size exclusion chromatography coupled to native mass spectrometry (SEC-nMS). Previous studies showed that these isomers might originate from a proline

Identifiants

pubmed: 35604400
doi: 10.1021/acs.analchem.2c00928
pmc: PMC9178554
doi:

Substances chimiques

Antibodies, Monoclonal 0
Antineoplastic Agents, Immunological 0

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

7981-7989

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Auteurs

Evolène Deslignière (E)

Laboratoire de Spectrométrie de Masse BioOrganique, Université de Strasbourg, CNRS, IPHC UMR 7178, 67087 Strasbourg, France.
Infrastructure Nationale de Protéomique ProFI - FR2048, 67087 Strasbourg, France.

Simon Ollivier (S)

INRAE, UR BIA, F-44316 Nantes, France.
INRAE, BIBS Facility, F-44316 Nantes, France.

Anthony Ehkirch (A)

Laboratoire de Spectrométrie de Masse BioOrganique, Université de Strasbourg, CNRS, IPHC UMR 7178, 67087 Strasbourg, France.
Infrastructure Nationale de Protéomique ProFI - FR2048, 67087 Strasbourg, France.

Armelle Martelet (A)

CMC Development, BioAnalytics department France, SANOFI R&D, 94400 Vitry-sur-Seine, France.

David Ropartz (D)

INRAE, UR BIA, F-44316 Nantes, France.
INRAE, BIBS Facility, F-44316 Nantes, France.

Nelly Lechat (N)

CMC Development, BioAnalytics department France, SANOFI R&D, 94400 Vitry-sur-Seine, France.

Oscar Hernandez-Alba (O)

Laboratoire de Spectrométrie de Masse BioOrganique, Université de Strasbourg, CNRS, IPHC UMR 7178, 67087 Strasbourg, France.
Infrastructure Nationale de Protéomique ProFI - FR2048, 67087 Strasbourg, France.

Jean-Michel Menet (JM)

CMC Development, BioAnalytics department France, SANOFI R&D, 94400 Vitry-sur-Seine, France.

Séverine Clavier (S)

CMC Development, BioAnalytics department France, SANOFI R&D, 94400 Vitry-sur-Seine, France.

Hélène Rogniaux (H)

INRAE, UR BIA, F-44316 Nantes, France.
INRAE, BIBS Facility, F-44316 Nantes, France.

Bruno Genet (B)

CMC Development, BioAnalytics department France, SANOFI R&D, 94400 Vitry-sur-Seine, France.

Sarah Cianférani (S)

Laboratoire de Spectrométrie de Masse BioOrganique, Université de Strasbourg, CNRS, IPHC UMR 7178, 67087 Strasbourg, France.
Infrastructure Nationale de Protéomique ProFI - FR2048, 67087 Strasbourg, France.

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Classifications MeSH