The Succinate Receptor SUCNR1 Resides at the Endoplasmic Reticulum and Relocates to the Plasma Membrane in Hypoxic Conditions.


Journal

Cells
ISSN: 2073-4409
Titre abrégé: Cells
Pays: Switzerland
ID NLM: 101600052

Informations de publication

Date de publication:
13 07 2022
Historique:
received: 17 05 2022
revised: 08 07 2022
accepted: 09 07 2022
entrez: 27 7 2022
pubmed: 28 7 2022
medline: 29 7 2022
Statut: epublish

Résumé

The GPCR SUCNR1/GPR91 exerts proangiogenesis upon stimulation with the Krebs cycle metabolite succinate. GPCR signaling depends on the surrounding environment and intracellular localization through location bias. Here, we show by microscopy and by cell fractionation that in neurons, SUCNR1 resides at the endoplasmic reticulum (ER), while being fully functional, as shown by calcium release and the induction of the expression of the proangiogenic gene for VEGFA. ER localization was found to depend upon N-glycosylation, particularly at position N8; the nonglycosylated mutant receptor localizes at the plasma membrane shuttled by RAB11. This SUCNR1 glycosylation is physiologically regulated, so that during hypoxic conditions, SUCNR1 is deglycosylated and relocates to the plasma membrane. Downstream signal transduction of SUCNR1 was found to activate the prostaglandin synthesis pathway through direct interaction with COX-2 at the ER; pharmacologic antagonism of the PGE

Identifiants

pubmed: 35883628
pii: cells11142185
doi: 10.3390/cells11142185
pmc: PMC9321536
pii:
doi:

Substances chimiques

Receptors, G-Protein-Coupled 0
Succinates 0
Succinic Acid AB6MNQ6J6L

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Subventions

Organisme : CIHR
Pays : Canada

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Auteurs

Melanie Sanchez (M)

Department of Pharmacology and Therapeutics, McGill University, Montréal, QC H3A 1A3, Canada.

David Hamel (D)

Department of Pharmacology, Université de Montréal, Montréal, QC H3C 3J7, Canada.

Emmanuel Bajon (E)

Department of Pediatrics, Research Center-CHU Ste-Justine, Montréal, QC H3T 1C5, Canada.

François Duhamel (F)

Department of Pharmacology, Université de Montréal, Montréal, QC H3C 3J7, Canada.

Vikrant K Bhosle (VK)

Department of Pharmacology and Therapeutics, McGill University, Montréal, QC H3A 1A3, Canada.
Cell Biology Program, The Hospital for Sick Children Research Institute, Toronto, ON M5G 1X8, Canada.

Tang Zhu (T)

Department of Pediatrics, Research Center-CHU Ste-Justine, Montréal, QC H3T 1C5, Canada.

Jose Carlos Rivera (JC)

Department of Ophthalmology, Research Center of Hôpital Maisonneuve-Rosemont, Université de Montréal, Montréal, QC H1T 2M4, Canada.

Rabah Dabouz (R)

Department of Pharmacology and Therapeutics, McGill University, Montréal, QC H3A 1A3, Canada.

Mathieu Nadeau-Vallée (M)

Department of Pharmacology, Université de Montréal, Montréal, QC H3C 3J7, Canada.

Nicholas Sitaras (N)

Department of Pharmacology, Université de Montréal, Montréal, QC H3C 3J7, Canada.

David-Étienne Tremblay (DÉ)

Department of Pharmacology, Université de Montréal, Montréal, QC H3C 3J7, Canada.

Samy Omri (S)

Department of Ophthalmology, Research Center of Hôpital Maisonneuve-Rosemont, Université de Montréal, Montréal, QC H1T 2M4, Canada.

Tiffany Habelrih (T)

Department of Pharmacology, Université de Montréal, Montréal, QC H3C 3J7, Canada.

Raphael Rouget (R)

Department of Pharmacology and Therapeutics, McGill University, Montréal, QC H3A 1A3, Canada.

Xin Hou (X)

Department of Pediatrics, Research Center-CHU Ste-Justine, Montréal, QC H3T 1C5, Canada.

Fernand Gobeil (F)

Department of Pharmacology, Université de Sherbrooke, Sherbrooke, QC J1H 5N4, Canada.

Jean-Sébastien Joyal (JS)

Department of Pediatrics, Research Center-CHU Ste-Justine, Montréal, QC H3T 1C5, Canada.
Department of Ophthalmology, Research Center of Hôpital Maisonneuve-Rosemont, Université de Montréal, Montréal, QC H1T 2M4, Canada.

Przemyslaw Sapieha (P)

Department of Ophthalmology, Research Center of Hôpital Maisonneuve-Rosemont, Université de Montréal, Montréal, QC H1T 2M4, Canada.

Grant Mitchell (G)

Department of Pediatrics, Research Center-CHU Ste-Justine, Montréal, QC H3T 1C5, Canada.

Alfredo Ribeiro-Da-Silva (A)

Department of Pharmacology and Therapeutics, McGill University, Montréal, QC H3A 1A3, Canada.

Mohammad Ali Mohammad Nezhady (MA)

Department of Pediatrics, Research Center-CHU Ste-Justine, Montréal, QC H3T 1C5, Canada.
Program of Molecular Biology, Faculty of Medicine, Université de Montréal, Montréal, QC H3T 1J4, Canada.
Research Center-CHU Ste-Justine, Departments of Pediatrics, Ophthalmology, and Pharmacology, Faculty of Medicine, Université de Montréal, 3175, Chemin Côte Ste-Catherine, Montréal, QC H3T 1C5, Canada.

Sylvain Chemtob (S)

Department of Pharmacology and Therapeutics, McGill University, Montréal, QC H3A 1A3, Canada.
Department of Pharmacology, Université de Montréal, Montréal, QC H3C 3J7, Canada.
Department of Pediatrics, Research Center-CHU Ste-Justine, Montréal, QC H3T 1C5, Canada.
Department of Ophthalmology, Research Center of Hôpital Maisonneuve-Rosemont, Université de Montréal, Montréal, QC H1T 2M4, Canada.
Research Center-CHU Ste-Justine, Departments of Pediatrics, Ophthalmology, and Pharmacology, Faculty of Medicine, Université de Montréal, 3175, Chemin Côte Ste-Catherine, Montréal, QC H3T 1C5, Canada.

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Classifications MeSH