Preliminary Evidence of the Potent and Selective Adenosine A2B Receptor Antagonist PSB-603 in Reducing Obesity and Some of Its Associated Metabolic Disorders in Mice.
Animals
Mice
Adenosine
/ pharmacology
Adenosine A2 Receptor Antagonists
/ pharmacology
Body Weight
Cholesterol
/ therapeutic use
Glucose
/ metabolism
Metabolic Diseases
Obesity
/ drug therapy
Purine Nucleosides
Purinergic P1 Receptor Antagonists
/ therapeutic use
Receptor, Adenosine A2B
/ metabolism
Theophylline
Triglycerides
/ therapeutic use
PSB-603
Theophylline
adenosine A2B receptor antagonist
glucose tolerance
metabolic disorder
obesity
Journal
International journal of molecular sciences
ISSN: 1422-0067
Titre abrégé: Int J Mol Sci
Pays: Switzerland
ID NLM: 101092791
Informations de publication
Date de publication:
03 Nov 2022
03 Nov 2022
Historique:
received:
21
09
2022
revised:
27
10
2022
accepted:
01
11
2022
entrez:
11
11
2022
pubmed:
12
11
2022
medline:
15
11
2022
Statut:
epublish
Résumé
The adenosine A
Identifiants
pubmed: 36362227
pii: ijms232113439
doi: 10.3390/ijms232113439
pmc: PMC9656786
pii:
doi:
Substances chimiques
Adenosine
K72T3FS567
Adenosine A2 Receptor Antagonists
0
Cholesterol
97C5T2UQ7J
Glucose
IY9XDZ35W2
Purine Nucleosides
0
Purinergic P1 Receptor Antagonists
0
Receptor, Adenosine A2B
0
Theophylline
C137DTR5RG
Triglycerides
0
psb-603
0
Types de publication
Journal Article
Langues
eng
Sous-ensembles de citation
IM
Subventions
Organisme : Faculty of Pharmacy Jagiellonian University Medical College,
ID : N42/DBS/000039
Organisme : qLife Priority Research Area
ID : N/A
Références
Allergol Int. 2007 Dec;56(4):445-56
pubmed: 17965584
Pharmacol Res. 2015 Sep;99:229-36
pubmed: 26142494
Brain Dev. 2004 Oct;26(7):448-52
pubmed: 15351080
Diabetes Metab Res Rev. 2014 Jan;30(1):42-53
pubmed: 23956030
PLoS One. 2015 Oct 27;10(10):e0141327
pubmed: 26506439
Lipids Health Dis. 2019 Jan 5;18(1):1
pubmed: 30611256
Rev Endocr Metab Disord. 2021 Dec;22(4):1073-1090
pubmed: 34165671
J Cell Physiol. 2014 Apr;229(4):414-21
pubmed: 24114647
J Clin Invest. 2009 Mar;119(3):582-94
pubmed: 19221436
Purinergic Signal. 2015 Sep;11(3):389-407
pubmed: 26126429
Cells. 2020 May 18;9(5):
pubmed: 32443525
Gerontology. 2009;55(4):379-86
pubmed: 19365105
Purinergic Signal. 2006 Sep;2(3):559-71
pubmed: 18404493
Front Med. 2013 Mar;7(1):14-24
pubmed: 23471659
Metab Brain Dis. 2016 Oct;31(5):1023-9
pubmed: 27216278
PLoS One. 2012;7(7):e40584
pubmed: 22848385
Int J Obes (Lond). 2012 Mar;36(3):397-406
pubmed: 21730968
Biomed Pharmacother. 2021 Mar;135:111164
pubmed: 33385856
Brain Res Bull. 2006 Feb 15;68(6):464-8
pubmed: 16459204
Diabetes. 2014 Mar;63(3):850-66
pubmed: 24194503
Biochem J. 1987 Nov 15;248(1):35-41
pubmed: 2829826
J Med Chem. 2002 May 23;45(11):2131-8
pubmed: 12014951
Lab Invest. 2013 Jan;93(1):135-44
pubmed: 23069939
Purinergic Signal. 2017 Dec;13(4):497-510
pubmed: 28808842
J Nutr. 2006 Mar;136(3):582-7
pubmed: 16484528
Eur Cytokine Netw. 2006 Mar;17(1):4-12
pubmed: 16613757
Crit Rev Food Sci Nutr. 2019;59(16):2597-2625
pubmed: 29624433
Diabetes. 2011 Feb;60(2):669-79
pubmed: 21270276
Drug Saf. 1990 Jul-Aug;5(4):275-85
pubmed: 2198052
J Med Chem. 2001 Jan 18;44(2):170-9
pubmed: 11170626
J Pharmacol Exp Ther. 2009 Apr;329(1):2-13
pubmed: 19141710
Biochem Pharmacol. 2019 Oct;168:193-203
pubmed: 31295465
Handb Exp Pharmacol. 2011;(200):151-99
pubmed: 20859796
Aging (Albany NY). 2015 Apr;7(4):256-68
pubmed: 25979814
Braz J Med Biol Res. 2020;53(9):e9877
pubmed: 32725081
Naunyn Schmiedebergs Arch Pharmacol. 2018 Aug;391(8):875-881
pubmed: 29802412
Behav Brain Res. 2013 Jun 15;247:217-26
pubmed: 23557694
PLoS One. 2014 Jun 03;9(6):e98775
pubmed: 24892847
PLoS One. 2020 Jun 18;15(6):e0229806
pubmed: 32555600
Front Pharmacol. 2021 Jan 18;11:621955
pubmed: 33536924
Chest. 1991 Jun;99(6):1415-20
pubmed: 2036824
J Pharmacol Exp Ther. 2016 Feb;356(2):333-40
pubmed: 26585572
J Med Chem. 2009 Jul 9;52(13):3994-4006
pubmed: 19569717
Behav Pharmacol. 2012 Sep;23(5-6):567-74
pubmed: 22743606
Biosci Biotechnol Biochem. 2006 May;70(5):1134-9
pubmed: 16717413
Circulation. 2012 Jan 17;125(2):354-63
pubmed: 22144568
Nature. 2014 Dec 18;516(7531):395-9
pubmed: 25317558
Front Physiol. 2015 Aug 07;6:222
pubmed: 26300787
Cell Metab. 2020 Jul 7;32(1):56-70.e7
pubmed: 32589947
Pharmacol Biochem Behav. 2008 May;89(3):345-51
pubmed: 18281083
J Pharm Pharmacol. 2006 Dec;58(12):1639-45
pubmed: 17331328
Front Pharmacol. 2017 Nov 24;8:878
pubmed: 29249968
J Med Primatol. 2011 Oct;40(5):335-41
pubmed: 21812784
Eur J Pharmacol. 2003 Jan 17;459(2-3):159-66
pubmed: 12524141