Multiomics Study of a Novel Naturally Derived Small Molecule, NSC772864, as a Potential Inhibitor of Proto-Oncogenes Regulating Cell Cycle Progression in Colorectal Cancer.
colorectal cancer
drug resistance
molecular docking simulation
protein–ligand interaction
small molecule
Journal
Cells
ISSN: 2073-4409
Titre abrégé: Cells
Pays: Switzerland
ID NLM: 101600052
Informations de publication
Date de publication:
16 01 2023
16 01 2023
Historique:
received:
17
11
2022
revised:
24
12
2022
accepted:
04
01
2023
entrez:
21
1
2023
pubmed:
22
1
2023
medline:
25
1
2023
Statut:
epublish
Résumé
Colorectal cancer (CRC) is one of the most prevalent malignant tumors, and it contributes to high numbers of deaths globally. Although advances in understanding CRC molecular mechanisms have shed significant light on its pathogenicity, current treatment options, including combined chemotherapy and molecular-targeted agents, are still limited due to resistance, with almost 25% of patients developing distant metastasis. Therefore, identifying novel biomarkers for early diagnosis is crucial, as they will also influence strategies for new targeted therapies. The proto-oncogene,
Identifiants
pubmed: 36672275
pii: cells12020340
doi: 10.3390/cells12020340
pmc: PMC9856482
pii:
doi:
Substances chimiques
Glycogen Synthase Kinase 3 beta
EC 2.7.11.1
Types de publication
Journal Article
Research Support, Non-U.S. Gov't
Langues
eng
Sous-ensembles de citation
IM
Références
Crit Rev Clin Lab Sci. 2019 Dec;56(8):533-566
pubmed: 31512514
Clin Cancer Res. 2004 Aug 1;10(15):5168-77
pubmed: 15297421
Gynecol Oncol. 2009 Sep;114(3):472-9
pubmed: 19524285
J Immunother Cancer. 2020 Oct;8(2):
pubmed: 33115942
Asian Pac J Cancer Prev. 2014;15(7):3133-7
pubmed: 24815459
PLoS One. 2015 Feb 06;10(2):e0116570
pubmed: 25659145
Nat Rev Cancer. 2002 Apr;2(4):289-300
pubmed: 12001990
Cancer Res. 2008 Feb 15;68(4):1213-20
pubmed: 18281498
Cancer Cell Int. 2019 Apr 02;19:80
pubmed: 30983885
Pharmacol Rev. 2017 Oct;69(4):479-496
pubmed: 28931623
Oncogenesis. 2019 Feb 26;8(3):19
pubmed: 30808873
J Cell Sci. 2003 Apr 1;116(Pt 7):1175-86
pubmed: 12615961
Proteomics. 2015 Aug;15(15):2597-601
pubmed: 25921073
J Clin Oncol. 2008 Nov 20;26(33):5352-9
pubmed: 18955458
Cancers (Basel). 2022 Jan 05;14(1):
pubmed: 35008426
N Engl J Med. 2004 Jun 3;350(23):2335-42
pubmed: 15175435
Curr Med Chem. 2011;18(10):1488-508
pubmed: 21428893
Eur J Med Chem. 2012 Jan;47(1):323-36
pubmed: 22100139
Eur J Cancer Prev. 2014 Jul;23(4):246-57
pubmed: 24614649
Int J Mol Sci. 2020 Jul 28;21(15):
pubmed: 32731413
J Cell Biol. 1996 Aug;134(3):757-70
pubmed: 8707853
J Comput Aided Mol Des. 2010 May;24(5):417-22
pubmed: 20401516
Oncotarget. 2016 Aug 23;7(34):54627-54631
pubmed: 27421137
Cancer Res. 2015 Jan 15;75(2):245-9
pubmed: 25593032
Mod Pathol. 2013 Feb;26(2):302-13
pubmed: 22936063
Bioorg Med Chem. 2000 Oct;8(10):2461-6
pubmed: 11058041
Onco Targets Ther. 2016 Mar 31;9:1899-920
pubmed: 27099521
Bioorg Med Chem. 2008 Jul 15;16(14):6976-86
pubmed: 18571928
Future Med Chem. 2014;6(17):1869-81
pubmed: 25495981
J Cell Physiol. 2019 Jul;234(7):10336-10344
pubmed: 30480806
CA Cancer J Clin. 2022 Jan;72(1):7-33
pubmed: 35020204
Cancers (Basel). 2021 May 21;13(11):
pubmed: 34063946
Cancer Treat Rev. 2017 Nov;60:1-11
pubmed: 28843992
Nat Commun. 2021 Jan 12;12(1):346
pubmed: 33436641
Eur J Cardiothorac Surg. 2016 Apr;49(4):1103-11; discussion 1111
pubmed: 26503729
Eur J Med Chem. 2015 Jun 15;98:115-26
pubmed: 26005025
Cancer Lett. 2021 Dec 28;523:121-134
pubmed: 34626691
Cell Rep. 2013 Dec 12;5(5):1214-27
pubmed: 24290754
Eur Urol. 2021 Oct;80(4):417-424
pubmed: 34187771
Int J Mol Sci. 2021 Feb 28;22(5):
pubmed: 33671112
Expert Opin Pharmacother. 2007 Oct;8(14):2359-69
pubmed: 17927489
Nucleic Acids Res. 2010 Jul;38(Web Server issue):W609-14
pubmed: 20430828
Nature. 2006 May 25;441(7092):444-50
pubmed: 16724056
Cell Death Dis. 2020 Aug 14;11(8):622
pubmed: 32796813
Int J Mol Sci. 2021 Mar 05;22(5):
pubmed: 33807717
Trends Biochem Sci. 1995 May;20(5):187-90
pubmed: 7610482
Oncology. 1998 Mar-Apr;55(2):145-51
pubmed: 9499189
Tumour Biol. 2015 Dec;36(12):9813-21
pubmed: 26159851
Sci Rep. 2017 Mar 03;7:42717
pubmed: 28256516
Nat Rev Mol Cell Biol. 2010 Dec;11(12):834-48
pubmed: 21102609
Neoplasia. 2017 Aug;19(8):649-658
pubmed: 28732212
Adv Drug Deliv Rev. 2001 Mar 1;46(1-3):3-26
pubmed: 11259830
Hum Pathol. 2013 Aug;44(8):1617-23
pubmed: 23574779
Cold Spring Harb Perspect Biol. 2015 Jan 05;7(1):a020412
pubmed: 25561720
Clin Cancer Res. 1995 Feb;1(2):147-54
pubmed: 9815967
Proteomes. 2016 Sep 12;4(3):
pubmed: 28248238
Neuro Oncol. 2013 Feb;15(2):161-71
pubmed: 23258844
Cancer Discov. 2012 May;2(5):401-4
pubmed: 22588877
Gastroenterology. 2007 Aug;133(2):647-58
pubmed: 17681183
Nat Rev Cancer. 2006 Aug;6(8):637-45
pubmed: 16862193
Biomed Pharmacother. 2014 Oct;68(8):1161-75
pubmed: 25458785
Nat Rev Genet. 2004 Jul;5(7):522-31
pubmed: 15211354
Angew Chem Int Ed Engl. 1999 Oct 4;38(19):2894-2896
pubmed: 10540384
Cancer Lett. 1994 Jun 30;81(2):165-9
pubmed: 8012933
Front Med. 2018 Aug;12(4):412-425
pubmed: 30054853
J Clin Oncol. 2011 May 20;29(15):2011-9
pubmed: 21502544
Nat Rev Cancer. 2006 Oct;6(10):813-23
pubmed: 16990858
Nat Commun. 2019 Sep 27;10(1):4404
pubmed: 31562303
N Engl J Med. 2009 Apr 2;360(14):1408-17
pubmed: 19339720
Lancet. 2014 Apr 26;383(9927):1490-1502
pubmed: 24225001
PLoS One. 2015 Oct 01;10(10):e0139727
pubmed: 26426996
Nucleic Acids Res. 2019 Jan 8;47(D1):D607-D613
pubmed: 30476243
Mol Cancer Ther. 2010 Oct;9(10):2724-36
pubmed: 20876746
Cell Cycle. 2020 Jan;19(2):163-178
pubmed: 31885322
Bioinformatics. 2018 Nov 1;34(21):3771-3772
pubmed: 29790900
Dig Dis Sci. 2015 Mar;60(3):762-72
pubmed: 25492499
Br J Cancer. 2016 Feb 16;114(4):362-7
pubmed: 26742008
J Cheminform. 2012 Aug 13;4(1):17
pubmed: 22889332
J Chem Inf Model. 2016 Feb 22;56(2):300-7
pubmed: 26838127
ChemMedChem. 2016 Jun 6;11(11):1117-21
pubmed: 27218427
Int J Cancer. 2021 Jan 15;148(2):502-511
pubmed: 32875562
Bioorg Med Chem. 2009 Nov 1;17(21):7418-28
pubmed: 19804981
Proc Natl Acad Sci U S A. 2017 Sep 12;114(37):E7697-E7706
pubmed: 28847964
Nature. 2012 Jul 18;487(7407):330-7
pubmed: 22810696
Trends Cell Biol. 2015 Nov;25(11):675-686
pubmed: 26437589
Cancer Lett. 2007 Apr 18;248(2):219-28
pubmed: 16945480
Hum Mol Genet. 2010 Apr 1;19(7):1324-34
pubmed: 20064923
Drug Des Devel Ther. 2015 Apr 08;9:2033-47
pubmed: 25897210
J Natl Cancer Inst. 1989 Jul 19;81(14):1088-92
pubmed: 2738938
Clin Cancer Res. 2013 Dec 15;19(24):6751-65
pubmed: 24122793
Cancer Treat Rev. 2021 Mar;94:102154
pubmed: 33524794
Anticancer Res. 2009 Nov;29(11):4807-11
pubmed: 20032439
Curr Med Chem. 2019;26(6):963-972
pubmed: 28990511
APMIS. 2004 Jan;112(1):49-56
pubmed: 14961975
Ann Oncol. 2016 Aug;27(8):1386-422
pubmed: 27380959
CA Cancer J Clin. 2015 Mar;65(2):87-108
pubmed: 25651787
Expert Opin Drug Discov. 2017 Jun;12(6):583-597
pubmed: 28399679
Nature. 2021 Jul;595(7869):730-734
pubmed: 34290403
Dev Dyn. 2018 Mar;247(3):521-530
pubmed: 28560804
Clin Colorectal Cancer. 2018 Sep;17(3):165-169
pubmed: 29576428
J Mol Med (Berl). 2016 Dec;94(12):1313-1326
pubmed: 27695879
Nat Commun. 2021 Nov 18;12(1):6711
pubmed: 34795238
Nucleic Acids Res. 2019 Jul 2;47(W1):W234-W241
pubmed: 30931480
Genome Biol. 2007;8(9):R183
pubmed: 17784955
Cold Spring Harb Perspect Biol. 2012 May 01;4(5):
pubmed: 22438566
Drug Discov Today. 2011 Jan;16(1-2):65-72
pubmed: 21074634
Bioinformatics. 2019 Jan 1;35(1):156-159
pubmed: 30010797
Hepatology. 2013 Jun;57(6):2299-313
pubmed: 23325601
Cancer Sci. 2016 Dec;107(12):1867-1876
pubmed: 27779808
PLoS One. 2016 Apr 21;11(4):e0154278
pubmed: 27100886
Int J Cancer. 2001 Sep 20;95(5):302-6
pubmed: 11494229
Science. 1998 Sep 4;281(5382):1509-12
pubmed: 9727977
J Med Chem. 2005 May 5;48(9):3164-70
pubmed: 15857122
J Clin Oncol. 2008 Apr 20;26(12):2013-9
pubmed: 18421054
Mol Cancer. 2019 Dec 18;18(1):185
pubmed: 31849331
Cells. 2020 Apr 22;9(4):
pubmed: 32331235
Clin Cancer Res. 2003 May;9(5):1808-14
pubmed: 12738738
N Engl J Med. 2013 Sep 12;369(11):1023-34
pubmed: 24024839
Ann Surg Oncol. 2001 Oct;8(9):729-40
pubmed: 11597015
Cancer Res. 2002 Sep 15;62(18):5126-8
pubmed: 12234972