Discovery of "Molecular Switches" within a Series of mGlu

Journal

ACS bio & med chem Au
ISSN: 2694-2437
Titre abrégé: ACS Bio Med Chem Au
Pays: United States
ID NLM: 9918232604406676

Informations de publication

Date de publication:
15 Dec 2021
Historique:
medline: 20 8 2021
pubmed: 20 8 2021
entrez: 27 4 2023
Statut: epublish

Résumé

In the course of optimizing an M

Identifiants

DOI: 10.1021/acsbiomedchemau.1c00024 PMID: 37101980 PMC: PMC10114714
pubmed: 37101980
doi: 10.1021/acsbiomedchemau.1c00024
pmc: PMC10114714
doi:

Types de publication

Journal Article

Langues

eng

Pagination

21-30

Informations de copyright

© 2021 The Authors. Published by American Chemical Society.

Déclaration de conflit d'intérêts

The authors declare no competing financial interest.

Références

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Auteurs

Lisa Barbaro (L)

Warren Center for Neuroscience Drug Discovery, Department of Pharmacology, Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37232, United States.
Warren Center for Neuroscience Drug Discovery, Department of Pharmacology, Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37232, United States.

Alice L Rodriguez (AL)

Warren Center for Neuroscience Drug Discovery, Department of Pharmacology, Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37232, United States.
Warren Center for Neuroscience Drug Discovery, Department of Pharmacology, Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37232, United States.

Ashlyn N Blevins (AN)

Warren Center for Neuroscience Drug Discovery, Department of Pharmacology, Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37232, United States.
Warren Center for Neuroscience Drug Discovery, Department of Pharmacology, Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37232, United States.
ORCID: 0000-0002-9857-2474

Jonathan W Dickerson (JW)

Warren Center for Neuroscience Drug Discovery, Department of Pharmacology, Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37232, United States.
Warren Center for Neuroscience Drug Discovery, Department of Pharmacology, Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37232, United States.

Natasha Billard (N)

Warren Center for Neuroscience Drug Discovery, Department of Pharmacology, Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37232, United States.
Warren Center for Neuroscience Drug Discovery, Department of Pharmacology, Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37232, United States.

Olivier Boutaud (O)

Warren Center for Neuroscience Drug Discovery, Department of Pharmacology, Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37232, United States.
Warren Center for Neuroscience Drug Discovery, Department of Pharmacology, Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37232, United States.

Jerri L Rook (JL)

Warren Center for Neuroscience Drug Discovery, Department of Pharmacology, Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37232, United States.
Warren Center for Neuroscience Drug Discovery, Department of Pharmacology, Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37232, United States.

Colleen M Niswender (CM)

Warren Center for Neuroscience Drug Discovery, Department of Pharmacology, Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37232, United States.
Warren Center for Neuroscience Drug Discovery, Department of Pharmacology, Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37232, United States.
Vanderbilt Kennedy Center, Vanderbilt University Medical Center, Nashville, Tennessee 37232, United States.
Warren Center for Neuroscience Drug Discovery, Department of Pharmacology, Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37232, United States.
Vanderbilt Brain Institute, Vanderbilt University, Nashville, Tennessee 37232, United States.

P Jeffrey Conn (PJ)

Warren Center for Neuroscience Drug Discovery, Department of Pharmacology, Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37232, United States.
Warren Center for Neuroscience Drug Discovery, Department of Pharmacology, Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37232, United States.
Vanderbilt Kennedy Center, Vanderbilt University Medical Center, Nashville, Tennessee 37232, United States.
Vanderbilt Institute of Chemical Biology, Vanderbilt University, Nashville, Tennessee 37232, United States.

Darren W Engers (DW)

Warren Center for Neuroscience Drug Discovery, Department of Pharmacology, Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37232, United States.
Warren Center for Neuroscience Drug Discovery, Department of Pharmacology, Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37232, United States.

Craig W Lindsley (CW)

Warren Center for Neuroscience Drug Discovery, Department of Pharmacology, Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37232, United States.
Warren Center for Neuroscience Drug Discovery, Department of Pharmacology, Department of Chemistry, Vanderbilt University, Nashville, Tennessee 37232, United States.
Vanderbilt Institute of Chemical Biology, Vanderbilt University, Nashville, Tennessee 37232, United States.
ORCID: 0000-0003-0168-1445

Classifications MeSH