Stabilizing Nitroxide Spin Labels for Structural and Conformational Studies of Biomolecules by Maleimide Treatment.

DEER measurement cell lysates protein spin labelling protein structure stability of NO radical

Journal

Chemistry (Weinheim an der Bergstrasse, Germany)
ISSN: 1521-3765
Titre abrégé: Chemistry
Pays: Germany
ID NLM: 9513783

Informations de publication

Date de publication:
06 Sep 2023
Historique:
received: 28 04 2023
medline: 8 9 2023
pubmed: 24 6 2023
entrez: 24 6 2023
Statut: ppublish

Résumé

Nitroxide (NO) spin radicals are effective in characterizing structures, interactions and dynamics of biomolecules. The EPR applications in cell lysates or intracellular milieu require stable spin labels, but NO radicals are unstable in such conditions. We showed that the destabilization of NO radicals in cell lysates or even in cells is caused by NADPH/NADH related enzymes, but not by the commonly believed reducing reagents such as GSH. Maleimide stabilizes the NO radicals in the cell lysates by consumption of the NADPH/NADH that are essential for the enzymes involved in destabilizing NO radicals, instead of serving as the solo thiol scavenger. The maleimide treatment retains the crowding properties of the intracellular components and allows to perform long-time EPR measurements of NO labeled biomolecules close to the intracellular conditions. The strategy of maleimide treatment on cell lysates for the EPR applications has been demonstrated on double electron-electron resonance (DEER) measurements on a number of NO labeled protein samples. The method opens a broad application range for the NO labeled biomolecules by EPR in conditions that resemble the intracellular milieu.

Identifiants

pubmed: 37354082
doi: 10.1002/chem.202301350
doi:

Substances chimiques

Spin Labels 0
nitroxyl GFQ4MMS07W
NAD 0U46U6E8UK
NADP 53-59-8
Maleimides 0

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

e202301350

Subventions

Organisme : Ministry of Science and Technology of China
ID : 2021YFA1600304
Organisme : National Natural Science Foundation of China
ID : 22161142018, 22174074, and 21991081

Informations de copyright

© 2023 Wiley-VCH GmbH.

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Auteurs

Xi-Wei Wang (XW)

State Key Laboratory of Elemento-organic Chemistry, Tianjin Key Laboratory of Biosensing and Molecular Recognition, College of Chemistry, Nankai University, Tianjin, 300071, China.

Xing Zhang (X)

State Key Laboratory of Elemento-organic Chemistry, Tianjin Key Laboratory of Biosensing and Molecular Recognition, College of Chemistry, Nankai University, Tianjin, 300071, China.

Chao-Yu Cui (CY)

State Key Laboratory of Elemento-organic Chemistry, Tianjin Key Laboratory of Biosensing and Molecular Recognition, College of Chemistry, Nankai University, Tianjin, 300071, China.

Bin Li (B)

State Key Laboratory of Elemento-organic Chemistry, Tianjin Key Laboratory of Biosensing and Molecular Recognition, College of Chemistry, Nankai University, Tianjin, 300071, China.

Daniella Goldfarb (D)

Department of Chemical and Biological Physics, Weizmann Institute of Science, Rehovot, 76100, Israel.

Yin Yang (Y)

State Key Laboratory of Elemento-organic Chemistry, Tianjin Key Laboratory of Biosensing and Molecular Recognition, College of Chemistry, Nankai University, Tianjin, 300071, China.

Xun-Cheng Su (XC)

State Key Laboratory of Elemento-organic Chemistry, Tianjin Key Laboratory of Biosensing and Molecular Recognition, College of Chemistry, Nankai University, Tianjin, 300071, China.

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