Elranatamab in relapsed or refractory multiple myeloma: phase 2 MagnetisMM-3 trial results.


Journal

Nature medicine
ISSN: 1546-170X
Titre abrégé: Nat Med
Pays: United States
ID NLM: 9502015

Informations de publication

Date de publication:
09 2023
Historique:
received: 18 06 2023
accepted: 01 08 2023
medline: 18 9 2023
pubmed: 16 8 2023
entrez: 15 8 2023
Statut: ppublish

Résumé

Elranatamab is a humanized B-cell maturation antigen (BCMA)-CD3 bispecific antibody. In the ongoing phase 2 MagnetisMM-3 trial, patients with relapsed or refractory multiple myeloma received subcutaneous elranatamab once weekly after two step-up priming doses. After six cycles, persistent responders switched to biweekly dosing. Results from cohort A, which enrolled patients without prior BCMA-directed therapy (n = 123) are reported. The primary endpoint of confirmed objective response rate (ORR) by blinded independent central review was met with an ORR of 61.0% (75/123); 35.0% ≥complete response. Fifty responders switched to biweekly dosing, and 40 (80.0%) improved or maintained their response for ≥6 months. With a median follow-up of 14.7 months, median duration of response, progression-free survival and overall survival (secondary endpoints) have not been reached. Fifteen-month rates were 71.5%, 50.9% and 56.7%, respectively. Common adverse events (any grade; grade 3-4) included infections (69.9%, 39.8%), cytokine release syndrome (57.7%, 0%), anemia (48.8%, 37.4%), and neutropenia (48.8%, 48.8%). With biweekly dosing, grade 3-4 adverse events decreased from 58.6% to 46.6%. Elranatamab induced deep and durable responses with a manageable safety profile. Switching to biweekly dosing may improve long-term safety without compromising efficacy. ClinicalTrials.gov identifier: NCT04649359 .

Identifiants

pubmed: 37582952
doi: 10.1038/s41591-023-02528-9
pii: 10.1038/s41591-023-02528-9
pmc: PMC10504075
doi:

Substances chimiques

B-Cell Maturation Antigen 0

Banques de données

ClinicalTrials.gov
['NCT04649359']

Types de publication

Clinical Trial, Phase II Journal Article Research Support, N.I.H., Extramural Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

2259-2267

Subventions

Organisme : NCI NIH HHS
ID : P30 CA008748
Pays : United States
Organisme : NCI NIH HHS
ID : P30 CA086862
Pays : United States

Informations de copyright

© 2023. The Author(s).

Références

Mateos, M. V. et al. LocoMMotion: a prospective, non-interventional, multinational study of real-life current standards of care in patients with relapsed and/or refractory multiple myeloma. Leukemia 36, 1371–1376 (2022).
doi: 10.1038/s41375-022-01531-2 pubmed: 35332278 pmcid: 9061296
Rodriguez-Otero, P. & San-Miguel, J. F. Cellular therapy for multiple myeloma: what’s now and what’s next. Hematol. Am. Soc. Hematol. Educ. Program 2022, 180–189 (2022).
doi: 10.1182/hematology.2022000396
Shah, N., Chari, A., Scott, E., Mezzi, K. & Usmani, S. Z. B-cell maturation antigen (BCMA) in multiple myeloma: rationale for targeting and current therapeutic approaches. Leukemia 34, 985–1005 (2020).
doi: 10.1038/s41375-020-0734-z pubmed: 32055000 pmcid: 7214244
Moreau, P. et al. Teclistamab in relapsed or refractory multiple myeloma. N. Engl. J. Med. 387, 495–505 (2022).
doi: 10.1056/NEJMoa2203478 pubmed: 35661166
Munshi, N. C. et al. Idecabtagene vicleucel in relapsed and refractory multiple myeloma. N. Engl. J. Med. 384, 705–716 (2021).
doi: 10.1056/NEJMoa2024850 pubmed: 33626253
Berdeja, J. G. et al. Ciltacabtagene autoleucel, a B-cell maturation antigen-directed chimeric antigen receptor T-cell therapy in patients with relapsed or refractory multiple myeloma (CARTITUDE-1): a phase 1b/2 open-label study. Lancet 398, 314–324 (2021).
doi: 10.1016/S0140-6736(21)00933-8 pubmed: 34175021
Celgene Corporation, a Bristol-Myers Squibb Company. ABECMA
Janssen Biotech, Inc. CARVYKTI
Janssen Biotech, Inc. TECVAYLI
Panowski, S. H. et al. Preclinical efficacy and safety comparison of CD3 bispecific and ADC modalities targeting BCMA for the treatment of multiple myeloma. Mol. Cancer Ther. 18, 2008–2020 (2019).
doi: 10.1158/1535-7163.MCT-19-0007 pubmed: 31434693
Nizar, J. B. et al. Efficacy and safety of elranatamab (PF-06863135), a B-cell maturation antigen (BCMA)-CD3 bispecific antibody, in patients with relapsed or refractory multiple myeloma (MM). J. Clin. Oncol. 39, 8006 (2021).
doi: 10.1200/JCO.2021.39.15_suppl.8006
Sebag, M. et al. Elranatamab (PF-06863135), a B-cell maturation antigen (BCMA) targeted CD3-engaging bispecific molecule, for patients with relapsed or refractory multiple myeloma: results from MagnetisMM-1. Blood 138, 895 (2021).
doi: 10.1182/blood-2021-150519
Andrzej, J. J. et al. Elranatamab, a BCMA-targeted T-cell redirecting immunotherapy, for patients with relapsed or refractory multiple myeloma: updated results from MagnetisMM-1. J. Clin. Oncol. 40, 8014 (2022).
doi: 10.1200/JCO.2022.40.16_suppl.8014
Raje, N. et al. Elranatamab, a BCMA targeted T-cell engaging bispecific antibody, induces durable clinical and molecular responses for patients with relapsed or refractory multiple myeloma. Blood 140, 388–390 (2022).
doi: 10.1182/blood-2022-166494
Lesokhin, A. M. et al. Initial safety results for MagnetisMM-3: a phase 2 trial of elranatamab, a B-cell maturation antigen (BCMA)-CD3 bispecific antibody, in patients (pts) with relapsed/refractory (R/R) multiple myeloma (MM). J. Clin. Oncol. 40, 8006 (2022).
doi: 10.1200/JCO.2022.40.16_suppl.8006
Lesokhin, A. et al. Magnetismm-3: an open-label, multicenter, non-randomized phase 2 study of elranatamab (PF-06863135) in patients with relapsed or refractory multiple myeloma. Blood 138, 1674 (2021).
doi: 10.1182/blood-2021-152984
Kumar, S. et al. International Myeloma Working Group consensus criteria for response and minimal residual disease assessment in multiple myeloma. Lancet Oncol. 17, e328–e346 (2016).
doi: 10.1016/S1470-2045(16)30206-6 pubmed: 27511158
Lee, D. W. et al. ASTCT consensus grading for cytokine release syndrome and neurologic toxicity associated with immune effector cells. Biol. Blood Marrow Transplant. 25, 625–638 (2019).
doi: 10.1016/j.bbmt.2018.12.758 pubmed: 30592986
Lonial, S. et al. Belantamab mafodotin for relapsed or refractory multiple myeloma (DREAMM-2): a two-arm, randomised, open-label, phase 2 study. Lancet Oncol. 21, 207–221 (2020).
doi: 10.1016/S1470-2045(19)30788-0 pubmed: 31859245
Blade, J. et al. Extramedullary disease in multiple myeloma: a systematic literature review. Blood Cancer J. 12, 45 (2022).
doi: 10.1038/s41408-022-00643-3 pubmed: 35314675 pmcid: 8938478
Palumbo, A. et al. Revised international staging system for multiple myeloma: a report from International Myeloma Working Group. J. Clin. Oncol. 33, 2863–2869 (2015).
doi: 10.1200/JCO.2015.61.2267 pubmed: 26240224 pmcid: 4846284
Gill, S. K. et al. I-OPen: inferior outcomes of penta-refractory compared to penta-exposed multiple myeloma patients. Blood Cancer J. 12, 138 (2022).
doi: 10.1038/s41408-022-00733-2 pubmed: 36151090 pmcid: 9508328
Lonial, S. et al. Longer term outcomes with single-agent belantamab mafodotin in patients with relapsed or refractory multiple myeloma: 13-month follow-up from the pivotal DREAMM-2 study. Cancer 127, 4198–4212 (2021).
doi: 10.1002/cncr.33809 pubmed: 34314018
Donk de van, N. W. C. J. et al. Long-term follow-up from MajesTEC-1 of teclistamab, a B-cell maturation antigen (BCMA) x CD3 bispecific antibody, in patients with relapsed/refractory multiple myeloma (RRMM). J. Clin. Oncol. 41, 8011 (2023).
doi: 10.1200/JCO.2023.41.16_suppl.8011
Martin, T. et al. Ciltacabtagene autoleucel, an anti-B-cell maturation antigen chimeric antigen receptor T-cell therapy, for relapsed/refractory multiple myeloma: CARTITUDE-1 2-year follow-up. J. Clin. Oncol. 41, 1265–1274 (2023).
doi: 10.1200/JCO.22.00842 pubmed: 35658469
Chari, A. et al. Talquetamab, a T-cell-redirecting GPRC5D bispecific antibody for multiple myeloma. N. Engl. J. Med. 387, 2232–2244 (2022).
doi: 10.1056/NEJMoa2204591 pubmed: 36507686
GlaxoSmithKline, Ltd. BLENREP (belantamab mafodotin-blmf) prescribing information. https://www.accessdata.fda.gov/drugsatfda_docs/label/2020/761158s000lbl.pdf (2020).
Richardson, P. G. et al. A phase 2 study of bortezomib in relapsed, refractory myeloma. N. Engl. J. Med. 348, 2609–2617 (2003).
doi: 10.1056/NEJMoa030288 pubmed: 12826635
Rajkumar, S. V. Thalidomide in the treatment of multiple myeloma. Expert Rev. Anticancer Ther. 1, 20–28 (2001).
doi: 10.1586/14737140.1.1.20 pubmed: 12113124
Sim, B. Z. et al. Infectious complications of bispecific antibody therapy in patients with multiple myeloma. Blood Cancer J. 13, 34 (2023).
doi: 10.1038/s41408-023-00808-8 pubmed: 36894539 pmcid: 9998258
Mazahreh, F. et al. Risk of infections associated with the use of bispecific antibodies in multiple myeloma: a pooled analysis. Blood Adv. 7, 3069–3074 (2023).
doi: 10.1182/bloodadvances.2022009435 pubmed: 36857755 pmcid: 10331406
Kambhampati, S. et al. Infectious complications in patients with relapsed refractory multiple myeloma after BCMA CAR T-cell therapy. Blood Adv. 6, 2045–2054 (2022).
doi: 10.1182/bloodadvances.2020004079 pubmed: 34543400 pmcid: 9006279
Mikkilineni, L. et al. Infectious complications of CAR T-cell therapy across novel antigen targets in the first 30 days. Blood Adv. 5, 5312–5322 (2021).
doi: 10.1182/bloodadvances.2021004896 pubmed: 34619768 pmcid: 9153053
Mohan, M. et al. Risk of infections with B-cell maturation antigen-directed immunotherapy in multiple myeloma. Blood Adv. 6, 2466–2470 (2022).
doi: 10.1182/bloodadvances.2021006178 pubmed: 34933344 pmcid: 9043928
D’Souza, A. et al. A phase I first-in-human study of ABBV-383, a B-cell maturation antigen x CD3 bispecific T-cell redirecting antibody, in patients with relapsed/refractory multiple myeloma. J. Clin. Oncol. 40, 3576–3586 (2022).
doi: 10.1200/JCO.22.01504 pubmed: 36029527 pmcid: 9622641
Raje, N. S. et al. Consensus guidelines and recommendations for infection prevention in multiple myeloma: a report from the International Myeloma Working Group. Lancet Haematol. 9, e143–e161 (2022).
doi: 10.1016/S2352-3026(21)00283-0 pubmed: 35114152
Ludwig, H. et al. Prevention and management of adverse events during treatment with bispecific antibodies and CAR T cells in multiple myeloma: a consensus report of the European Myeloma Network. Lancet Oncol. 24, e255–e269 (2023).
doi: 10.1016/S1470-2045(23)00159-6 pubmed: 37269857
Terpos, E. et al. Management of patients with multiple myeloma and COVID-19 in the post pandemic era: a consensus paper from the European Myeloma Network (EMN). Leukemia 37, 1175–1185 (2023).
doi: 10.1038/s41375-023-01920-1 pubmed: 37142661 pmcid: 10157596
Raje, N. A. et al. Monitoring, prophylaxis, and treatment of infections in patients with MM receiving 1 bispecific antibody therapy: consensus recommendations from an expert panel. Blood Cancer J. 13, 116 (2023).
doi: 10.1038/s41408-023-00879-7 pubmed: 37528088 pmcid: 10394080

Auteurs

Alexander M Lesokhin (AM)

Division of Hematology and Oncology, Memorial Sloan Kettering Cancer Center/Weill Cornell Medical College, New York City, NY, USA. lesokhia@mskcc.org.

Michael H Tomasson (MH)

Department of Internal Medicine, University of Iowa, Iowa City, IA, USA.

Bertrand Arnulf (B)

Hôpital Saint-Louis, Paris, France.

Nizar J Bahlis (NJ)

Arnie Charbonneau Cancer Institute, University of Calgary, Calgary, Alberta, Canada.

H Miles Prince (H)

Epworth Healthcare and University of Melbourne, Melbourne, Victoria, Australia.

Ruben Niesvizky (R)

Weill Cornell Medical College/New York Presbyterian Hospital, New York City, NY, USA.

Paula Rodrίguez-Otero (P)

Clinica Universidad de Navarra, Madrid, Spain.

Joaquin Martinez-Lopez (J)

Hospital Universitario 12 de Octubre, Madrid, Spain.

Guenther Koehne (G)

Miami Cancer Institute, Miami, FL, USA.

Cyrille Touzeau (C)

University Hospital of Nantes, Nantes, France.

Yogesh Jethava (Y)

Indiana Blood & Marrow Transplant, Indianapolis, IN, USA.

Hang Quach (H)

University of Melbourne, St. Vincent's Hospital Melbourne, Melbourne, Victoria, Australia.

Julien Depaus (J)

Université Catholique de Louvain, CHU UCL Namur, Yvoir, Belgium.

Hisayuki Yokoyama (H)

Tohoku University Graduate School of Medicine, Sendai, Japan.

Afshin Eli Gabayan (AE)

Beverly Hills Cancer Center, Beverly Hills, CA, USA.

Don A Stevens (DA)

Norton Cancer Center, Louisville, KY, USA.

Ajay K Nooka (AK)

Winship Cancer Institute, Atlanta, GA, USA.

Salomon Manier (S)

Lille University Hospital and INSERM UMR-S1277, Lille, France.

Noopur Raje (N)

Massachusetts General Hospital Cancer Center, Harvard Medical School, Boston, MA, USA.

Shinsuke Iida (S)

Department of Hematology & Oncology, Nagoya City University Graduate School of Medical Sciences, Nagoya, Japan.

Marc-Steffen Raab (MS)

Heidelberg Myeloma Center, Department of Hematology/Oncology, Heidelberg University Hospital, Heidelberg, Germany.

Emma Searle (E)

The Christie Hospital, The University of Manchester, Manchester, UK.

Eric Leip (E)

Pfizer Inc, Cambridge, MA, USA.

Sharon T Sullivan (ST)

Pfizer Inc, Cambridge, MA, USA.

Umberto Conte (U)

Pfizer Inc, New York, NY, USA.

Mohamed Elmeliegy (M)

Pfizer Inc, San Diego, CA, USA.

Akos Czibere (A)

Pfizer Inc, New York, NY, USA.

Andrea Viqueira (A)

Pfizer SLU, Madrid, Spain.

Mohamad Mohty (M)

Sorbonne University, Hôpital Saint-Antoine, and INSERM UMRs938, Paris, France.

Articles similaires

[Redispensing of expensive oral anticancer medicines: a practical application].

Lisanne N van Merendonk, Kübra Akgöl, Bastiaan Nuijen
1.00
Humans Antineoplastic Agents Administration, Oral Drug Costs Counterfeit Drugs

Smoking Cessation and Incident Cardiovascular Disease.

Jun Hwan Cho, Seung Yong Shin, Hoseob Kim et al.
1.00
Humans Male Smoking Cessation Cardiovascular Diseases Female
Humans United States Aged Cross-Sectional Studies Medicare Part C
1.00
Humans Yoga Low Back Pain Female Male

Classifications MeSH