Pharmaceutical stability of methemoglobin-albumin cluster as an antidote for hydrogen sulfide poisoning after one-year storage in freeze-dried form.


Journal

International journal of pharmaceutics
ISSN: 1873-3476
Titre abrégé: Int J Pharm
Pays: Netherlands
ID NLM: 7804127

Informations de publication

Date de publication:
15 Oct 2023
Historique:
received: 17 07 2023
revised: 23 08 2023
accepted: 19 09 2023
medline: 9 10 2023
pubmed: 23 9 2023
entrez: 22 9 2023
Statut: ppublish

Résumé

Long-term stability during storage is an important requirement for pharmaceutical preparations. The methemoglobin (metHb)-albumin cluster, in which bovine metHb is covalently enveloped with an average of three human albumin molecules, is a promising antidote for hydrogen sulfide (H

Identifiants

pubmed: 37739098
pii: S0378-5173(23)00854-2
doi: 10.1016/j.ijpharm.2023.123433
pii:
doi:

Substances chimiques

Methemoglobin 9008-37-1
Antidotes 0
Hydrogen Sulfide YY9FVM7NSN
Powders 0
Albumins 0

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

123433

Informations de copyright

Copyright © 2023 Elsevier B.V. All rights reserved.

Déclaration de conflit d'intérêts

Declaration of Competing Interest The authors declare that they have no known competing financial interests or personal relationships that could have appeared to influence the work reported in this paper.

Auteurs

Yuto Suzuki (Y)

Division of Pharmacodynamics, Faculty of Pharmacy, Keio University, Tokyo 105-8512, Japan.

Kazuaki Taguchi (K)

Division of Pharmacodynamics, Faculty of Pharmacy, Keio University, Tokyo 105-8512, Japan. Electronic address: taguchi-kz@pha.keio.ac.jp.

Wataru Okamoto (W)

Department of Applied Chemistry, Faculty of Science and Engineering, Chuo University, Tokyo 112-8551, Japan.

Yuki Enoki (Y)

Division of Pharmacodynamics, Faculty of Pharmacy, Keio University, Tokyo 105-8512, Japan.

Teruyuki Komatsu (T)

Department of Applied Chemistry, Faculty of Science and Engineering, Chuo University, Tokyo 112-8551, Japan.

Kazuaki Matsumoto (K)

Division of Pharmacodynamics, Faculty of Pharmacy, Keio University, Tokyo 105-8512, Japan.

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Classifications MeSH