Enhancing luciferase activity and stability through generative modeling of natural enzyme sequences.

enzyme catalysis enzyme design generative model mutation effects natural evolution

Journal

Proceedings of the National Academy of Sciences of the United States of America
ISSN: 1091-6490
Titre abrégé: Proc Natl Acad Sci U S A
Pays: United States
ID NLM: 7505876

Informations de publication

Date de publication:
28 Nov 2023
Historique:
pmc-release: 20 05 2024
medline: 22 11 2023
pubmed: 20 11 2023
entrez: 20 11 2023
Statut: ppublish

Résumé

The availability of natural protein sequences synergized with generative AI provides new paradigms to engineer enzymes. Although active enzyme variants with numerous mutations have been designed using generative models, their performance often falls short of their wild type counterparts. Additionally, in practical applications, choosing fewer mutations that can rival the efficacy of extensive sequence alterations is usually more advantageous. Pinpointing beneficial single mutations continues to be a formidable task. In this study, using the generative maximum entropy model to analyze

Identifiants

pubmed: 37983512
doi: 10.1073/pnas.2312848120
pmc: PMC10691223
doi:

Substances chimiques

Luciferases, Renilla EC 1.13.12.5

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

e2312848120

Subventions

Organisme : NIGMS NIH HHS
ID : R35 GM122472
Pays : United States

Commentaires et corrections

Type : UpdateOf

Déclaration de conflit d'intérêts

Competing interests statement:The authors declare no competing interest.

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Auteurs

Wen Jun Xie (WJ)

Department of Chemistry, University of Southern California, Los Angeles, CA 90089.
Department of Medicinal Chemistry, Center for Natural Products, Drug Discovery and Development, Genetics Institute, University of Florida, Gainesville, FL 32610.

Dangliang Liu (D)

State Key Laboratory of Natural and Biomimetic Drugs, Chemical Biology Center, School of Pharmaceutical Sciences, Peking University, Beijing 100191, China.

Xiaoya Wang (X)

State Key Laboratory of Natural and Biomimetic Drugs, Chemical Biology Center, School of Pharmaceutical Sciences, Peking University, Beijing 100191, China.

Aoxuan Zhang (A)

Department of Chemistry, University of Southern California, Los Angeles, CA 90089.

Qijia Wei (Q)

State Key Laboratory of Natural and Biomimetic Drugs, Chemical Biology Center, School of Pharmaceutical Sciences, Peking University, Beijing 100191, China.

Ashim Nandi (A)

Department of Chemistry, University of Southern California, Los Angeles, CA 90089.

Suwei Dong (S)

State Key Laboratory of Natural and Biomimetic Drugs, Chemical Biology Center, School of Pharmaceutical Sciences, Peking University, Beijing 100191, China.

Arieh Warshel (A)

Department of Chemistry, University of Southern California, Los Angeles, CA 90089.

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Classifications MeSH