Accueil
Frederic Feru
Frederic Feru
Affiliations
Department of Cancer Biology, Dana-Farber Cancer Institute, Boston, MA 02115, USA; Department of Biological Chemistry & Molecular Pharmacology, Harvard Medical School, 360 Longwood Ave, Boston, MA 02115, USA.
Publications (5)
Discovery of a series of benzopyrimidodiazepinone TNK2 inhibitors via scaffold morphing.
Bioorganic & medicinal chemistry letters
Avec:
Zhengnian Li
,
Chelsea E Powell
,
Brian J Groendyke
,
Thomas W Gero
,
Frederic Feru
,
John Feutrill
,
Bailing Chen
,
Bin Li
,
Hilary Szabo
,
Nathanael S Gray
,
David A Scott
Benzopyrimidodiazepinone inhibitors of TNK2.
Bioorganic & medicinal chemistry letters
Avec:
Brian J Groendyke
,
Chelsea E Powell
,
Frederic Feru
,
Thomas W Gero
,
Zhengnian Li
,
Hilary Szabo
,
Kevin Pang
,
John Feutrill
,
Bailing Chen
,
Bin Li
,
Nathanael S Gray
,
David A Scott
Exploring Targeted Degradation Strategy for Oncogenic KRAS
Cell chemical biology
Avec:
Mei Zeng
,
Yuan Xiong
,
Nozhat Safaee
,
Radosław P Nowak
,
Katherine A Donovan
,
Christine J Yuan
,
Behnam Nabet
,
Thomas W Gero
,
Frederic Feru
,
Lianbo Li
,
Sudershan Gondi
,
Lincoln J Ombelets
,
Chunshan Quan
,
Pasi A Jänne
,
Milka Kostic
,
David A Scott
,
Kenneth D Westover
,
Eric S Fischer
,
Nathanael S Gray
Quinazolinones as allosteric fourth-generation EGFR inhibitors for the treatment of NSCLC.
Bioorganic & medicinal chemistry letters
Avec:
Thomas W Gero
,
David E Heppner
,
Tyler S Beyett
,
Ciric To
,
Seth C Azevedo
,
Jaebong Jang
,
Thomas Bunnell
,
Frederic Feru
,
Zhengnian Li
,
Bo Hee Shin
,
Kara M Soroko
,
Prafulla C Gokhale
,
Nathanael S Gray
,
Pasi A Jänne
,
Michael J Eck
,
David A Scott
From hit to vial: Precision discovery and development of an imidazopyrimidine TLR7/8 agonist adjuvant formulation.
Science advances
Avec:
Dheeraj Soni
,
Francesco Borriello
,
David A Scott
,
Frederic Feru
,
Maria DeLeon
,
Spencer E Brightman
,
Wing Ki Cheng
,
Gandolina Melhem
,
Jennifer A Smith
,
Juan C Ramirez
,
Soumik Barman
,
Michael Cameron
,
Aisling Kelly
,
Kristina Walker
,
Etsuro Nanishi
,
Simon Daniel van Haren
,
Tony Phan
,
Yizhi Qi
,
Robert Kinsey
,
Michal M Raczy
,
Al Ozonoff
,
Matthew A Pettengill
,
Jeffery A Hubbell
,
Christopher B Fox
,
David J Dowling
,
Ofer Levy
Réseau de co-auteurs
David A Scott
5 collaborations
Thomas W Gero
4 collaborations
Nathanael S Gray
4 collaborations
Zhengnian Li
3 collaborations
Chelsea E Powell
2 collaborations
Brian J Groendyke
2 collaborations
John Feutrill
2 collaborations
Bailing Chen
2 collaborations
Bin Li
2 collaborations
Hilary Szabo
2 collaborations
Pasi A Jänne
2 collaborations
Kevin Pang
1 collaboration
Mei Zeng
1 collaboration
Yuan Xiong
1 collaboration
Nozhat Safaee
1 collaboration
Radosław P Nowak
1 collaboration
Katherine A Donovan
1 collaboration
Christine J Yuan
1 collaboration
Behnam Nabet
1 collaboration
Lianbo Li
1 collaboration
Sudershan Gondi
1 collaboration
Lincoln J Ombelets
1 collaboration
Chunshan Quan
1 collaboration
Milka Kostic
1 collaboration
Kenneth D Westover
1 collaboration
Eric S Fischer
1 collaboration
David E Heppner
1 collaboration
Tyler S Beyett
1 collaboration
Ciric To
1 collaboration
Seth C Azevedo
1 collaboration
Jaebong Jang
1 collaboration
Thomas Bunnell
1 collaboration
Bo Hee Shin
1 collaboration
Kara M Soroko
1 collaboration
Prafulla C Gokhale
1 collaboration
Michael J Eck
1 collaboration
Dheeraj Soni
1 collaboration
Francesco Borriello
1 collaboration
Maria DeLeon
1 collaboration
Spencer E Brightman
1 collaboration
Wing Ki Cheng
1 collaboration
Gandolina Melhem
1 collaboration
Jennifer A Smith
1 collaboration
Juan C Ramirez
1 collaboration
Soumik Barman
1 collaboration
Michael Cameron
1 collaboration
Aisling Kelly
1 collaboration
Kristina Walker
1 collaboration
Etsuro Nanishi
1 collaboration
Simon Daniel van Haren
1 collaboration
Tony Phan
1 collaboration
Yizhi Qi
1 collaboration
Robert Kinsey
1 collaboration
Michal M Raczy
1 collaboration
Al Ozonoff
1 collaboration
Matthew A Pettengill
1 collaboration
Jeffery A Hubbell
1 collaboration
Christopher B Fox
1 collaboration
David J Dowling
1 collaboration
Ofer Levy
1 collaboration