Titre : Inhibiteur tissulaire de métalloprotéinase-1

Inhibiteur tissulaire de métalloprotéinase-1 : Questions médicales fréquentes

Termes MeSH sélectionnés :

Molecular Docking Simulation
{ "@context": "https://schema.org", "@graph": [ { "@type": "MedicalWebPage", "name": "Inhibiteur tissulaire de métalloprotéinase-1 : Questions médicales les plus fréquentes", "headline": "Inhibiteur tissulaire de métalloprotéinase-1 : Comprendre les symptômes, diagnostics et traitements", "description": "Guide complet et accessible sur les Inhibiteur tissulaire de métalloprotéinase-1 : explications, diagnostics, traitements et prévention. Information médicale validée destinée aux patients.", "datePublished": "2024-04-08", "dateModified": "2025-04-03", "inLanguage": "fr", "medicalAudience": [ { "@type": "MedicalAudience", "name": "Grand public", "audienceType": "Patient", "healthCondition": { "@type": "MedicalCondition", "name": "Inhibiteur tissulaire de métalloprotéinase-1" }, "suggestedMinAge": 18, "suggestedGender": "unisex" }, { "@type": "MedicalAudience", "name": "Médecins", "audienceType": "Physician", "geographicArea": { "@type": "AdministrativeArea", "name": "France" } }, { "@type": "MedicalAudience", "name": "Chercheurs", "audienceType": "Researcher", "geographicArea": { "@type": "AdministrativeArea", "name": "International" } } ], "reviewedBy": { "@type": "Person", "name": "Dr Olivier Menir", "jobTitle": "Expert en Médecine", "description": "Expert en Médecine, Optimisation des Parcours de Soins et Révision Médicale", "url": "/static/pages/docteur-olivier-menir.html", "alumniOf": { "@type": "EducationalOrganization", "name": "Université Paris Descartes" } }, "isPartOf": { "@type": "MedicalWebPage", "name": "Inhibiteur tissulaire des métalloprotéinases", "url": "https://questionsmedicales.fr/mesh/D019714", "about": { "@type": "MedicalCondition", "name": "Inhibiteur tissulaire des métalloprotéinases", "code": { "@type": "MedicalCode", "code": "D019714", "codingSystem": "MeSH" }, "identifier": { "@type": "PropertyValue", "propertyID": "MeSH Tree", "value": "D12.776.815.875" } } }, "about": { "@type": "MedicalCondition", "name": "Inhibiteur tissulaire de métalloprotéinase-1", "alternateName": "Tissue Inhibitor of Metalloproteinase-1", "code": { "@type": "MedicalCode", "code": "D019715", "codingSystem": "MeSH" } }, "author": [ { "@type": "Person", "name": "Anna Pryczynicz", "url": "https://questionsmedicales.fr/author/Anna%20Pryczynicz", "affiliation": { "@type": "Organization", "name": "Department of Pathomorphology, Medical University of Bialystok, Bialystok, Poland." } }, { "@type": "Person", "name": "Adina Elena Stanciu", "url": "https://questionsmedicales.fr/author/Adina%20Elena%20Stanciu", "affiliation": { "@type": "Organization", "name": "Department of Carcinogenesis and Molecular Biology, 'Prof. Dr. Alexandru Trestioreanu' Institute of Oncology, 022328 Bucharest, Romania." } }, { "@type": "Person", "name": "Adina Zamfir-Chiru-Anton", "url": "https://questionsmedicales.fr/author/Adina%20Zamfir-Chiru-Anton", "affiliation": { "@type": "Organization", "name": "ENT Department, 'Grigore Alexandrescu' Children's Emergency Hospital, 011743 Bucharest, Romania." } }, { "@type": "Person", "name": "Marcel Marian Stanciu", "url": "https://questionsmedicales.fr/author/Marcel%20Marian%20Stanciu", "affiliation": { "@type": "Organization", "name": "Electrical Engineering Faculty, 'Politehnica' University, 060042 Bucharest, Romania." } }, { "@type": "Person", "name": "Mirela Gherghe", "url": "https://questionsmedicales.fr/author/Mirela%20Gherghe", "affiliation": { "@type": "Organization", "name": "Department of Nuclear Medicine, 'Prof. Dr. Alexandru Trestioreanu' Institute of Oncology, 022328 Bucharest, Romania." } } ], "citation": [ { "@type": "ScholarlyArticle", "name": "Molecular docking, simulation and binding free energy analysis of small molecules as PfHT1 inhibitors.", "datePublished": "2022-08-26", "url": "https://questionsmedicales.fr/article/36026508", "identifier": { "@type": "PropertyValue", "propertyID": "DOI", "value": "10.1371/journal.pone.0268269" } }, { "@type": "ScholarlyArticle", "name": "Py-CoMFA, docking, and molecular dynamics simulations of Leishmania (L.) amazonensis arginase inhibitors.", "datePublished": "2024-05-21", "url": "https://questionsmedicales.fr/article/38773273", "identifier": { "@type": "PropertyValue", "propertyID": "DOI", "value": "10.1038/s41598-024-62520-2" } }, { "@type": "ScholarlyArticle", "name": "Exploring the molecular mechanism of ginseng against anthracycline-induced cardiotoxicity based on network pharmacology, molecular docking and molecular dynamics simulation.", "datePublished": "2024-09-06", "url": "https://questionsmedicales.fr/article/39243097", "identifier": { "@type": "PropertyValue", "propertyID": "DOI", "value": "10.1186/s41065-024-00334-y" } }, { "@type": "ScholarlyArticle", "name": "Study of the antidiabetic mechanism of berberine compound on FOXO1 transcription factor through molecular docking and molecular dynamics simulations.", "datePublished": "2024-07-09", "url": "https://questionsmedicales.fr/article/38981921", "identifier": { "@type": "PropertyValue", "propertyID": "DOI", "value": "10.1007/s00894-024-06060-6" } }, { "@type": "ScholarlyArticle", "name": "Research advances of molecular docking and molecular dynamic simulation in recognizing interaction between muscle proteins and exogenous additives.", "datePublished": "2023-07-08", "url": "https://questionsmedicales.fr/article/37453331", "identifier": { "@type": "PropertyValue", "propertyID": "DOI", "value": "10.1016/j.foodchem.2023.136836" } } ], "breadcrumb": { "@type": "BreadcrumbList", "itemListElement": [ { "@type": "ListItem", "position": 1, "name": "questionsmedicales.fr", "item": "https://questionsmedicales.fr" }, { "@type": "ListItem", "position": 2, "name": "Acides aminés, peptides et protéines", "item": "https://questionsmedicales.fr/mesh/D000602" }, { "@type": "ListItem", "position": 3, "name": "Protéines", "item": "https://questionsmedicales.fr/mesh/D011506" }, { "@type": "ListItem", "position": 4, "name": "Protéines sécrétoires inhibitrices de protéinases", "item": "https://questionsmedicales.fr/mesh/D053491" }, { "@type": "ListItem", "position": 5, "name": "Inhibiteur tissulaire des métalloprotéinases", "item": "https://questionsmedicales.fr/mesh/D019714" }, { "@type": "ListItem", "position": 6, "name": "Inhibiteur tissulaire de métalloprotéinase-1", "item": "https://questionsmedicales.fr/mesh/D019715" } ] } }, { "@type": "MedicalWebPage", "name": "Article complet : Inhibiteur tissulaire de métalloprotéinase-1 - Questions et réponses", "headline": "Questions et réponses médicales fréquentes sur Inhibiteur tissulaire de métalloprotéinase-1", "description": "Une compilation de questions et réponses structurées, validées par des experts médicaux.", "datePublished": "2025-05-10", "inLanguage": "fr", "hasPart": [ { "@type": "MedicalWebPage", "name": "Diagnostic", "headline": "Diagnostic sur Inhibiteur tissulaire de métalloprotéinase-1", "description": "Comment diagnostiquer une anomalie de TIMP-1 ?\nQuels symptômes indiquent un déséquilibre de TIMP-1 ?\nY a-t-il des biomarqueurs associés à TIMP-1 ?\nQuel rôle joue TIMP-1 dans le cancer ?\nComment TIMP-1 est-il mesuré en clinique ?", "url": "https://questionsmedicales.fr/mesh/D019715?mesh_terms=Molecular+Docking+Simulation&page=3#section-diagnostic" }, { "@type": "MedicalWebPage", "name": "Symptômes", "headline": "Symptômes sur Inhibiteur tissulaire de métalloprotéinase-1", "description": "Quels symptômes sont liés à une surproduction de TIMP-1 ?\nTIMP-1 affecte-t-il la cicatrisation des plaies ?\nQuels signes indiquent une carence en TIMP-1 ?\nY a-t-il des symptômes associés à des maladies inflammatoires ?\nComment TIMP-1 influence-t-il l'inflammation ?", "url": "https://questionsmedicales.fr/mesh/D019715?mesh_terms=Molecular+Docking+Simulation&page=3#section-symptômes" }, { "@type": "MedicalWebPage", "name": "Prévention", "headline": "Prévention sur Inhibiteur tissulaire de métalloprotéinase-1", "description": "Peut-on prévenir les déséquilibres de TIMP-1 ?\nQuels facteurs de mode de vie influencent TIMP-1 ?\nY a-t-il des recommandations pour maintenir TIMP-1 ?\nLes suppléments peuvent-ils aider TIMP-1 ?\nComment le suivi médical aide-t-il TIMP-1 ?", "url": "https://questionsmedicales.fr/mesh/D019715?mesh_terms=Molecular+Docking+Simulation&page=3#section-prévention" }, { "@type": "MedicalWebPage", "name": "Traitements", "headline": "Traitements sur Inhibiteur tissulaire de métalloprotéinase-1", "description": "Quels traitements ciblent TIMP-1 ?\nTIMP-1 peut-il être utilisé comme cible thérapeutique ?\nQuels médicaments influencent TIMP-1 ?\nY a-t-il des essais cliniques sur TIMP-1 ?\nComment les traitements affectent-ils TIMP-1 ?", "url": "https://questionsmedicales.fr/mesh/D019715?mesh_terms=Molecular+Docking+Simulation&page=3#section-traitements" }, { "@type": "MedicalWebPage", "name": "Complications", "headline": "Complications sur Inhibiteur tissulaire de métalloprotéinase-1", "description": "Quelles complications peuvent survenir avec un excès de TIMP-1 ?\nTIMP-1 est-il lié à des maladies chroniques ?\nComment TIMP-1 affecte-t-il la santé cardiovasculaire ?\nY a-t-il des risques de cancer liés à TIMP-1 ?\nQuels effets secondaires peuvent résulter d'un traitement de TIMP-1 ?", "url": "https://questionsmedicales.fr/mesh/D019715?mesh_terms=Molecular+Docking+Simulation&page=3#section-complications" }, { "@type": "MedicalWebPage", "name": "Facteurs de risque", "headline": "Facteurs de risque sur Inhibiteur tissulaire de métalloprotéinase-1", "description": "Quels facteurs augmentent le risque de déséquilibre de TIMP-1 ?\nLes maladies auto-immunes influencent-elles TIMP-1 ?\nLe stress a-t-il un impact sur TIMP-1 ?\nL'alimentation joue-t-elle un rôle dans TIMP-1 ?\nY a-t-il un lien entre TIMP-1 et l'inactivité physique ?", "url": "https://questionsmedicales.fr/mesh/D019715?mesh_terms=Molecular+Docking+Simulation&page=3#section-facteurs de risque" } ] }, { "@type": "FAQPage", "mainEntity": [ { "@type": "Question", "name": "Comment diagnostiquer une anomalie de TIMP-1 ?", "position": 1, "acceptedAnswer": { "@type": "Answer", "text": "Des tests sanguins mesurant les niveaux de TIMP-1 peuvent être effectués." } }, { "@type": "Question", "name": "Quels symptômes indiquent un déséquilibre de TIMP-1 ?", "position": 2, "acceptedAnswer": { "@type": "Answer", "text": "Des symptômes comme l'inflammation ou des troubles de cicatrisation peuvent survenir." } }, { "@type": "Question", "name": "Y a-t-il des biomarqueurs associés à TIMP-1 ?", "position": 3, "acceptedAnswer": { "@type": "Answer", "text": "Oui, des biomarqueurs comme le collagène et les métalloprotéinases sont souvent étudiés." } }, { "@type": "Question", "name": "Quel rôle joue TIMP-1 dans le cancer ?", "position": 4, "acceptedAnswer": { "@type": "Answer", "text": "TIMP-1 peut inhiber la progression tumorale en régulant la dégradation de la matrice." } }, { "@type": "Question", "name": "Comment TIMP-1 est-il mesuré en clinique ?", "position": 5, "acceptedAnswer": { "@type": "Answer", "text": "Il est mesuré par des tests immunologiques spécifiques dans des échantillons de sang." } }, { "@type": "Question", "name": "Quels symptômes sont liés à une surproduction de TIMP-1 ?", "position": 6, "acceptedAnswer": { "@type": "Answer", "text": "Une surproduction peut entraîner des douleurs articulaires et une fibrose tissulaire." } }, { "@type": "Question", "name": "TIMP-1 affecte-t-il la cicatrisation des plaies ?", "position": 7, "acceptedAnswer": { "@type": "Answer", "text": "Oui, un excès de TIMP-1 peut ralentir la cicatrisation des plaies." } }, { "@type": "Question", "name": "Quels signes indiquent une carence en TIMP-1 ?", "position": 8, "acceptedAnswer": { "@type": "Answer", "text": "Une carence peut se manifester par une dégradation excessive de la matrice extracellulaire." } }, { "@type": "Question", "name": "Y a-t-il des symptômes associés à des maladies inflammatoires ?", "position": 9, "acceptedAnswer": { "@type": "Answer", "text": "Oui, des maladies comme l'arthrite peuvent être liées à des niveaux anormaux de TIMP-1." } }, { "@type": "Question", "name": "Comment TIMP-1 influence-t-il l'inflammation ?", "position": 10, "acceptedAnswer": { "@type": "Answer", "text": "TIMP-1 peut moduler l'inflammation en régulant les métalloprotéinases impliquées." } }, { "@type": "Question", "name": "Peut-on prévenir les déséquilibres de TIMP-1 ?", "position": 11, "acceptedAnswer": { "@type": "Answer", "text": "Une alimentation équilibrée et un mode de vie sain peuvent aider à maintenir l'équilibre." } }, { "@type": "Question", "name": "Quels facteurs de mode de vie influencent TIMP-1 ?", "position": 12, "acceptedAnswer": { "@type": "Answer", "text": "Le tabagisme et l'obésité peuvent affecter les niveaux de TIMP-1." } }, { "@type": "Question", "name": "Y a-t-il des recommandations pour maintenir TIMP-1 ?", "position": 13, "acceptedAnswer": { "@type": "Answer", "text": "Pratiquer une activité physique régulière et gérer le stress sont recommandés." } }, { "@type": "Question", "name": "Les suppléments peuvent-ils aider TIMP-1 ?", "position": 14, "acceptedAnswer": { "@type": "Answer", "text": "Certains suppléments antioxydants peuvent soutenir la régulation de TIMP-1." } }, { "@type": "Question", "name": "Comment le suivi médical aide-t-il TIMP-1 ?", "position": 15, "acceptedAnswer": { "@type": "Answer", "text": "Un suivi régulier permet de détecter et de corriger les déséquilibres de TIMP-1." } }, { "@type": "Question", "name": "Quels traitements ciblent TIMP-1 ?", "position": 16, "acceptedAnswer": { "@type": "Answer", "text": "Des thérapies géniques et des inhibiteurs spécifiques sont en cours d'étude." } }, { "@type": "Question", "name": "TIMP-1 peut-il être utilisé comme cible thérapeutique ?", "position": 17, "acceptedAnswer": { "@type": "Answer", "text": "Oui, en régulant TIMP-1, on peut potentiellement traiter certaines pathologies." } }, { "@type": "Question", "name": "Quels médicaments influencent TIMP-1 ?", "position": 18, "acceptedAnswer": { "@type": "Answer", "text": "Certains anti-inflammatoires peuvent moduler l'expression de TIMP-1." } }, { "@type": "Question", "name": "Y a-t-il des essais cliniques sur TIMP-1 ?", "position": 19, "acceptedAnswer": { "@type": "Answer", "text": "Oui, plusieurs essais cliniques explorent son rôle dans diverses maladies." } }, { "@type": "Question", "name": "Comment les traitements affectent-ils TIMP-1 ?", "position": 20, "acceptedAnswer": { "@type": "Answer", "text": "Les traitements peuvent soit augmenter, soit diminuer les niveaux de TIMP-1 selon le contexte." } }, { "@type": "Question", "name": "Quelles complications peuvent survenir avec un excès de TIMP-1 ?", "position": 21, "acceptedAnswer": { "@type": "Answer", "text": "Un excès peut entraîner des maladies fibrosantes et des troubles cardiovasculaires." } }, { "@type": "Question", "name": "TIMP-1 est-il lié à des maladies chroniques ?", "position": 22, "acceptedAnswer": { "@type": "Answer", "text": "Oui, des niveaux anormaux de TIMP-1 sont associés à des maladies chroniques comme le diabète." } }, { "@type": "Question", "name": "Comment TIMP-1 affecte-t-il la santé cardiovasculaire ?", "position": 23, "acceptedAnswer": { "@type": "Answer", "text": "Des niveaux élevés de TIMP-1 peuvent contribuer à l'athérosclérose." } }, { "@type": "Question", "name": "Y a-t-il des risques de cancer liés à TIMP-1 ?", "position": 24, "acceptedAnswer": { "@type": "Answer", "text": "Des niveaux élevés de TIMP-1 peuvent être associés à une progression tumorale." } }, { "@type": "Question", "name": "Quels effets secondaires peuvent résulter d'un traitement de TIMP-1 ?", "position": 25, "acceptedAnswer": { "@type": "Answer", "text": "Les traitements peuvent entraîner des effets secondaires comme des réactions allergiques." } }, { "@type": "Question", "name": "Quels facteurs augmentent le risque de déséquilibre de TIMP-1 ?", "position": 26, "acceptedAnswer": { "@type": "Answer", "text": "L'âge avancé, le tabagisme et l'obésité sont des facteurs de risque connus." } }, { "@type": "Question", "name": "Les maladies auto-immunes influencent-elles TIMP-1 ?", "position": 27, "acceptedAnswer": { "@type": "Answer", "text": "Oui, les maladies auto-immunes peuvent perturber l'équilibre de TIMP-1." } }, { "@type": "Question", "name": "Le stress a-t-il un impact sur TIMP-1 ?", "position": 28, "acceptedAnswer": { "@type": "Answer", "text": "Oui, le stress chronique peut affecter les niveaux de TIMP-1 dans l'organisme." } }, { "@type": "Question", "name": "L'alimentation joue-t-elle un rôle dans TIMP-1 ?", "position": 29, "acceptedAnswer": { "@type": "Answer", "text": "Une alimentation riche en graisses saturées peut perturber les niveaux de TIMP-1." } }, { "@type": "Question", "name": "Y a-t-il un lien entre TIMP-1 et l'inactivité physique ?", "position": 30, "acceptedAnswer": { "@type": "Answer", "text": "Oui, l'inactivité physique peut contribuer à des déséquilibres de TIMP-1." } } ] } ] }

Sources (10000 au total)

Exploring the molecular mechanism of ginseng against anthracycline-induced cardiotoxicity based on network pharmacology, molecular docking and molecular dynamics simulation.

Previous clinical and basic studies have revealed that ginseng might have cardioprotective properties against anthracycline-induced cardiotoxicity (AIC). However, the underlying mechanism of ginseng a... Fourteen drug-disease common targets were identified. Enrichment analysis showed that the AGE-RAGE in diabetic complications, fluid shear stress and atherosclerosis, and TNF signaling pathway were pot... This study suggested that ginseng might exert their protective effects against AIC through the derived effector compounds beta-Sitosterol, Kaempferol and Fumarine by targeting CCNA2, STAT1, and ICAM1,...

Study of the antidiabetic mechanism of berberine compound on FOXO1 transcription factor through molecular docking and molecular dynamics simulations.

Diabetes mellitus (DM) is a metabolic disorder disease that causes hyperglycemia conditions and associated with various chronic complications leading to mortality. Due to high toxicity of conventional... Docking between ligand and FOXO1 receptor was carried out with Autodock4.2. For molecular dynamics simulations, the force fields of DNA.OL15, protein.ff14SB, gaff2, and tip3p were used....

Research advances of molecular docking and molecular dynamic simulation in recognizing interaction between muscle proteins and exogenous additives.

During storage and processing, muscle proteins, e.g. myosin and myoglobin, will inevitably undergo degeneration, which is thus accompanied by quality deterioration of muscle foods. Some exogenous addi...

Discovery of Highly Potent CRBN Ligands and Insight into Their Binding Mode through Molecular Docking and Molecular Dynamics Simulations.

Cereblon (CRBN) is a substrate receptor of E3 ubiquitin ligase as well as the target of thalidomide and lenalidomide, plays a vital role in endogenous protein degradation. In this article, two series ...

QSAR Study, Molecular Docking and Molecular Dynamic Simulation of Aurora Kinase Inhibitors Derived from Imidazo[4,5-

Cancer is a serious threat to human life and social development and the use of scientific methods for cancer prevention and control is necessary. In this study, HQSAR, CoMFA, CoMSIA and TopomerCoMFA m...

Molecular modelling on multiepitope-based vaccine against SARS-CoV-2 using immunoinformatics, molecular docking, and molecular dynamics simulation.

The pandemic of COVID-19 caused by SARS-CoV-2 has made a worldwide health emergency. Despite the fact that current vaccines are readily available, several SARSCoV-2 variants affecting the existing vac...

In silico molecular targets, docking, dynamics simulation and physiologically based pharmacokinetics modeling of oritavancin.

Oritavancin is a semi-synthetic lipoglycopeptide antibiotic primarily used to treat serious infections caused by Gram-positive bacteria. The aim of this study was to elucidate possible molecular targe... Computational methods were used in this study which include target prediction, molecular docking, molecular dynamics simulation, pharmacokinetics prediction, and physiological-based pharmacokinetics (... Oritavancin was moderately soluble in water and did not permeate the blood-brain barrier. Seven molecular targets were identified in humans. Molecular docking results showed highest binding affinity o... This comprehensive computational study has provided invaluable insights into the pharmacological profile of Oritavancin, aiding its further development and optimization for clinical use....