The blocking of kappa-opioid receptor reverses the changes in dorsolateral striatum dopamine dynamics during the amphetamine sensitization.


Journal

Journal of neurochemistry
ISSN: 1471-4159
Titre abrégé: J Neurochem
Pays: England
ID NLM: 2985190R

Informations de publication

Date de publication:
02 2019
Historique:
received: 08 08 2018
revised: 25 09 2018
accepted: 05 10 2018
pubmed: 14 10 2018
medline: 28 10 2019
entrez: 14 10 2018
Statut: ppublish

Résumé

Kappa-opioid receptors (KOR) control dopamine (DA) levels in the striatum and contribute significantly to the progression of drug addiction. Repeated exposure to psychostimulants has been associated with up-regulated KOR activity and increased DA levels in dorsal striatum. However, it has not been tested if both processes are linked. In this work, we studied if a mechanism mediated by KOR is contributing to the increase in DA levels in the dorsolateral striatum (DLS) after amphetamine (AMPH) sensitization. The AMPH sensitization was assessed after single or repeated once-a-day AMPH injections (1 mg/kg). Only repeated AMPH exposure produced a significant locomotor sensitization. No-net flux microdialysis was used to assess basal DA dialysate, DA extracellular concentration (C

Identifiants

pubmed: 30315655
doi: 10.1111/jnc.14612
doi:

Substances chimiques

Central Nervous System Stimulants 0
Receptors, Opioid, kappa 0
Amphetamine CK833KGX7E
Dopamine VTD58H1Z2X

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

348-358

Informations de copyright

© 2018 International Society for Neurochemistry.

Auteurs

Victor Hugo Azocar (VH)

Department of Pharmacy and Interdisciplinary Center of Neuroscience, Pontificia Universidad Catolica de Chile, Santiago, Chile.

Gladys Sepúlveda (G)

Department of Pharmacy and Interdisciplinary Center of Neuroscience, Pontificia Universidad Catolica de Chile, Santiago, Chile.

Catalina Ruiz (C)

Department of Pharmacy and Interdisciplinary Center of Neuroscience, Pontificia Universidad Catolica de Chile, Santiago, Chile.

Consuelo Aguilera (C)

Department of Pharmacy and Interdisciplinary Center of Neuroscience, Pontificia Universidad Catolica de Chile, Santiago, Chile.

Maria Estela Andrés (ME)

Department of Cellular and Molecular Biology, Faculty of Biological Science, Pontificia Universidad Católica de Chile, Santiago, Chile.

José Antonio Fuentealba (JA)

Department of Pharmacy and Interdisciplinary Center of Neuroscience, Pontificia Universidad Catolica de Chile, Santiago, Chile.

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Classifications MeSH