Mitochondrial energetics is impaired in very long-chain acyl-CoA dehydrogenase deficiency and can be rescued by treatment with mitochondria-targeted electron scavengers.


Journal

Human molecular genetics
ISSN: 1460-2083
Titre abrégé: Hum Mol Genet
Pays: England
ID NLM: 9208958

Informations de publication

Date de publication:
15 03 2019
Historique:
received: 06 08 2018
revised: 12 11 2018
accepted: 13 11 2018
pubmed: 18 11 2018
medline: 10 3 2020
entrez: 17 11 2018
Statut: ppublish

Résumé

Very long-chain acyl-CoA dehydrogenase (VLCAD) deficiency is the most common defect of mitochondrial long-chain fatty acid β-oxidation. Patients present with heterogeneous clinical phenotypes affecting heart, liver and skeletal muscle predominantly. The full pathophysiology of the disease is unclear and patient response to current therapeutic regimens is incomplete. To identify additional cellular alterations and explore more effective therapies, mitochondrial bioenergetics and redox homeostasis were assessed in VLCAD-deficient fibroblasts, and several protective compounds were evaluated. The results revealed cellular and tissue changes, including decreased respiratory chain (RC) function, increased reactive oxygen species (ROS) production and altered mitochondrial function and signaling pathways in a variety of VLCAD-deficient fibroblasts. The mitochondrially enriched electron and free radical scavengers JP4-039 and XJB-5-131 improved RC function and decreased ROS production significantly, suggesting that they are viable candidate compounds to further develop to treat VLCAD-deficient patients.

Identifiants

pubmed: 30445591
pii: 5185121
doi: 10.1093/hmg/ddy403
pmc: PMC6400046
doi:

Substances chimiques

Antioxidants 0
Reactive Oxygen Species 0
Adenosine Triphosphate 8L70Q75FXE
Acyl-CoA Dehydrogenase, Long-Chain EC 1.3.8.8

Types de publication

Journal Article Research Support, N.I.H., Extramural

Langues

eng

Sous-ensembles de citation

IM

Pagination

928-941

Subventions

Organisme : NIDDK NIH HHS
ID : R01 DK078775
Pays : United States
Organisme : NIEHS NIH HHS
ID : R33 ES025606
Pays : United States

Informations de copyright

© The Author(s) 2018. Published by Oxford University Press.

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Auteurs

Bianca Seminotti (B)

Division Medical Genetics, Department of Pediatrics, University of Pittsburgh, Pittsburgh, PA, USA.
Programa de Pós-Graduação em Ciências Biológicas: Bioquímica, Departamento de Bioquímica, Instituto de Ciências Básicas da Saúde, Universidade Federal do Rio Grande do Sul, Porto Alegre, RS, Brazil.

Guilhian Leipnitz (G)

Division Medical Genetics, Department of Pediatrics, University of Pittsburgh, Pittsburgh, PA, USA.
Programa de Pós-Graduação em Ciências Biológicas: Bioquímica, Departamento de Bioquímica, Instituto de Ciências Básicas da Saúde, Universidade Federal do Rio Grande do Sul, Porto Alegre, RS, Brazil.

Anuradha Karunanidhi (A)

Division Medical Genetics, Department of Pediatrics, University of Pittsburgh, Pittsburgh, PA, USA.

Catherine Kochersperger (C)

Division Medical Genetics, Department of Pediatrics, University of Pittsburgh, Pittsburgh, PA, USA.

Vera Y Roginskaya (VY)

Department of Pharmacology and Chemical Biology, University of Pittsburgh, Pittsburgh, PA, USA.

Shrabani Basu (S)

Division Medical Genetics, Department of Pediatrics, University of Pittsburgh, Pittsburgh, PA, USA.

Yudong Wang (Y)

Division Medical Genetics, Department of Pediatrics, University of Pittsburgh, Pittsburgh, PA, USA.

Peter Wipf (P)

Department of Chemistry, University of Pittsburgh, Pittsburgh, PA, USA.

Bennett Van Houten (B)

Department of Pharmacology and Chemical Biology, University of Pittsburgh, Pittsburgh, PA, USA.

Al-Walid Mohsen (AW)

Division Medical Genetics, Department of Pediatrics, University of Pittsburgh, Pittsburgh, PA, USA.
Department of Human Genetics, Graduate School of Public Health, University of Pittsburgh, Pittsburgh, PA, USA.

Jerry Vockley (J)

Division Medical Genetics, Department of Pediatrics, University of Pittsburgh, Pittsburgh, PA, USA.
Department of Human Genetics, Graduate School of Public Health, University of Pittsburgh, Pittsburgh, PA, USA.

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