Platelet Inhibition With Cangrelor and Crushed Ticagrelor in Patients With ST-Segment-Elevation Myocardial Infarction Undergoing Primary Percutaneous Coronary Intervention.


Journal

Circulation
ISSN: 1524-4539
Titre abrégé: Circulation
Pays: United States
ID NLM: 0147763

Informations de publication

Date de publication:
02 04 2019
Historique:
pubmed: 12 1 2019
medline: 30 1 2020
entrez: 12 1 2019
Statut: ppublish

Résumé

The platelet inhibitory effects induced by oral P2Y This was a prospective, randomized, double-blind, placebo-controlled pharmacodynamic study conducted in patients undergoing primary percutaneous coronary intervention (n=50) who were randomized to treatment with either cangrelor or matching placebo (bolus followed by 2-hour infusion). All patients received ticagrelor 180-mg loading dose administered as crushed tablets at the time of cangrelor/placebo bolus administration. Pharmacodynamic analyses were performed at 8 time points. Pharmacodynamic effects were measured as P2Y Compared with placebo, cangrelor was associated with reduced P2Y In patients undergoing primary percutaneous coronary intervention, cangrelor is an effective strategy to bridge the gap in platelet inhibition associated with the use of oral P2Y URL: https://www.clinicaltrials.gov . Unique identifier: NCT03247738.

Sections du résumé

BACKGROUND
The platelet inhibitory effects induced by oral P2Y
METHODS
This was a prospective, randomized, double-blind, placebo-controlled pharmacodynamic study conducted in patients undergoing primary percutaneous coronary intervention (n=50) who were randomized to treatment with either cangrelor or matching placebo (bolus followed by 2-hour infusion). All patients received ticagrelor 180-mg loading dose administered as crushed tablets at the time of cangrelor/placebo bolus administration. Pharmacodynamic analyses were performed at 8 time points. Pharmacodynamic effects were measured as P2Y
RESULTS
Compared with placebo, cangrelor was associated with reduced P2Y
CONCLUSIONS
In patients undergoing primary percutaneous coronary intervention, cangrelor is an effective strategy to bridge the gap in platelet inhibition associated with the use of oral P2Y
CLINICAL TRIAL REGISTRATION
URL: https://www.clinicaltrials.gov . Unique identifier: NCT03247738.

Identifiants

pubmed: 30630341
doi: 10.1161/CIRCULATIONAHA.118.038317
doi:

Substances chimiques

Biomarkers 0
Cell Adhesion Molecules 0
Microfilament Proteins 0
P2RY12 protein, human 0
Phosphoproteins 0
Platelet Aggregation Inhibitors 0
Purinergic P2Y Receptor Antagonists 0
Receptors, Purinergic P2Y12 0
vasodilator-stimulated phosphoprotein 0
Adenosine Monophosphate 415SHH325A
cangrelor 6AQ1Y404U7
Ticagrelor GLH0314RVC

Banques de données

ClinicalTrials.gov
['NCT03247738']

Types de publication

Journal Article Randomized Controlled Trial Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

1661-1670

Commentaires et corrections

Type : CommentIn

Auteurs

Francesco Franchi (F)

Division of Cardiology, University of Florida College of Medicine-Jacksonville.

Fabiana Rollini (F)

Division of Cardiology, University of Florida College of Medicine-Jacksonville.

Andrea Rivas (A)

Division of Cardiology, University of Florida College of Medicine-Jacksonville.

Mustafa Wali (M)

Division of Cardiology, University of Florida College of Medicine-Jacksonville.

Maryuri Briceno (M)

Division of Cardiology, University of Florida College of Medicine-Jacksonville.

Malhar Agarwal (M)

Division of Cardiology, University of Florida College of Medicine-Jacksonville.

Zubair Shaikh (Z)

Division of Cardiology, University of Florida College of Medicine-Jacksonville.

Ahmed Nawaz (A)

Division of Cardiology, University of Florida College of Medicine-Jacksonville.

Gabriel Silva (G)

Division of Cardiology, University of Florida College of Medicine-Jacksonville.

Latonya Been (L)

Division of Cardiology, University of Florida College of Medicine-Jacksonville.

Ramez Smairat (R)

Division of Cardiology, University of Florida College of Medicine-Jacksonville.

Marc Kaufman (M)

Division of Cardiology, University of Florida College of Medicine-Jacksonville.

Andres M Pineda (AM)

Division of Cardiology, University of Florida College of Medicine-Jacksonville.

Siva Suryadevara (S)

Division of Cardiology, University of Florida College of Medicine-Jacksonville.

Daniel Soffer (D)

Division of Cardiology, University of Florida College of Medicine-Jacksonville.

Martin M Zenni (MM)

Division of Cardiology, University of Florida College of Medicine-Jacksonville.

Theodore A Bass (TA)

Division of Cardiology, University of Florida College of Medicine-Jacksonville.

Dominick J Angiolillo (DJ)

Division of Cardiology, University of Florida College of Medicine-Jacksonville.

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Classifications MeSH