Deaminative Reductive Cross-Electrophile Couplings of Alkylpyridinium Salts and Aryl Bromides.


Journal

Organic letters
ISSN: 1523-7052
Titre abrégé: Org Lett
Pays: United States
ID NLM: 100890393

Informations de publication

Date de publication:
19 04 2019
Historique:
pubmed: 28 3 2019
medline: 20 8 2019
entrez: 28 3 2019
Statut: ppublish

Résumé

A nickel-catalyzed reductive cross-coupling of alkylpyridinium salts and aryl bromides has been developed using Mn as the reductant. Both primary and secondary alkylpyridinium salts can be used, and high functional group and heterocycle tolerance is observed, including for protic groups. Mechanistic studies indicate the formation of an alkyl radical, and controlling its fate was key to the success of this reaction.

Identifiants

pubmed: 30917282
doi: 10.1021/acs.orglett.9b01014
pmc: PMC6517243
mid: NIHMS1020194
doi:

Substances chimiques

Amines 0
Boronic Acids 0
Free Radicals 0
Pyridines 0
Pyridinium Compounds 0
Magnesium Chloride 02F3473H9O
Manganese 42Z2K6ZL8P
nickel chloride 696BNE976J
Nickel 7OV03QG267
Bromine SBV4XY874G

Types de publication

Journal Article Research Support, N.I.H., Extramural Research Support, Non-U.S. Gov't

Langues

eng

Pagination

2941-2946

Subventions

Organisme : NIGMS NIH HHS
ID : P20 GM103541
Pays : United States
Organisme : NIGMS NIH HHS
ID : P20 GM104316
Pays : United States
Organisme : NIGMS NIH HHS
ID : R01 GM111820
Pays : United States
Organisme : NIH HHS
ID : S10 OD016267
Pays : United States

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Auteurs

Jennie Liao (J)

Department of Chemistry & Biochemistry , University of Delaware , Newark , Delaware 19716 , United States.

Corey H Basch (CH)

Department of Chemistry & Biochemistry , University of Delaware , Newark , Delaware 19716 , United States.

Megan E Hoerrner (ME)

Department of Chemistry & Biochemistry , University of Delaware , Newark , Delaware 19716 , United States.

Michael R Talley (MR)

Department of Chemistry & Biochemistry , University of Delaware , Newark , Delaware 19716 , United States.

Brian P Boscoe (BP)

Medicine Design, Pfizer Worldwide Research and Development , Groton , Connecticut 06340 , United States.

Joseph W Tucker (JW)

Medicine Design, Pfizer Worldwide Research and Development , Groton , Connecticut 06340 , United States.

Michelle R Garnsey (MR)

Medicine Design, Pfizer Worldwide Research and Development , Groton , Connecticut 06340 , United States.

Mary P Watson (MP)

Department of Chemistry & Biochemistry , University of Delaware , Newark , Delaware 19716 , United States.

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Classifications MeSH