Safety, Pharmacokinetics, and Food Effect of Tebipenem Pivoxil Hydrobromide after Single and Multiple Ascending Oral Doses in Healthy Adult Subjects.


Journal

Antimicrobial agents and chemotherapy
ISSN: 1098-6596
Titre abrégé: Antimicrob Agents Chemother
Pays: United States
ID NLM: 0315061

Informations de publication

Date de publication:
09 2019
Historique:
received: 22 03 2019
accepted: 16 05 2019
pubmed: 3 7 2019
medline: 18 7 2020
entrez: 3 7 2019
Statut: epublish

Résumé

Tebipenem pivoxil hydrobromide (TBPM-PI-HBr, formerly SPR994) is an orally available prodrug of tebipenem, a carbapenem with activity versus multidrug-resistant (MDR) Gram-negative pathogens, including quinolone-resistant and extended-spectrum-β-lactamase-producing

Identifiants

pubmed: 31262768
pii: AAC.00618-19
doi: 10.1128/AAC.00618-19
pmc: PMC6709501
pii:
doi:

Substances chimiques

Anti-Bacterial Agents 0
Carbapenems 0
Prodrugs 0
tebipenem Q2TWQ1I31U

Banques de données

ClinicalTrials.gov
['NCT03395249']

Types de publication

Journal Article Randomized Controlled Trial Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Informations de copyright

Copyright © 2019 Eckburg et al.

Références

J Infect Dis. 2017 Feb 15;215(suppl_1):S28-S36
pubmed: 28375512
Antimicrob Agents Chemother. 2019 Mar 27;63(4):
pubmed: 30718255
Drug Resist Updat. 2016 Nov;29:30-46
pubmed: 27912842
Antimicrob Agents Chemother. 2019 May 24;63(6):
pubmed: 30936096
Clin Infect Dis. 2018 Nov 28;67(12):1803-1814
pubmed: 30052813

Auteurs

Paul B Eckburg (PB)

Spero Therapeutics, Cambridge, Massachusetts, USA peckburg@sperotherapeutics.com.

Akash Jain (A)

Spero Therapeutics, Cambridge, Massachusetts, USA.

Susannah Walpole (S)

Spero Therapeutics, Cambridge, Massachusetts, USA.

Grayson Moore (G)

Spero Therapeutics, Cambridge, Massachusetts, USA.

Luke Utley (L)

Spero Therapeutics, Cambridge, Massachusetts, USA.

Erika Manyak (E)

Spero Therapeutics, Cambridge, Massachusetts, USA.

Aaron Dane (A)

DaneStat Consulting, Alderley Edge, United Kingdom.

David Melnick (D)

Spero Therapeutics, Cambridge, Massachusetts, USA.

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Classifications MeSH