Circulating dipeptidyl peptidase 3 is a myocardial depressant factor: dipeptidyl peptidase 3 inhibition rapidly and sustainably improves haemodynamics.


Journal

European journal of heart failure
ISSN: 1879-0844
Titre abrégé: Eur J Heart Fail
Pays: England
ID NLM: 100887595

Informations de publication

Date de publication:
02 2020
Historique:
received: 22 07 2019
revised: 01 08 2019
accepted: 05 08 2019
pubmed: 1 9 2019
medline: 19 5 2021
entrez: 1 9 2019
Statut: ppublish

Résumé

Acute heart failure is a high mortality disease and its pathophysiology is not completely understood. Dipeptidyl peptidase 3 (DPP3) is a cytosolic enzyme involved in angiotensin II and enkephalins cleavage. The aim of this study was to investigate the association of circulating DPP3 (cDPP3) levels and mortality in cardiogenic shock patients and to determine the effects of high cDPP3 on organ function in a heart failure (HF) model in mice. cDPP3 was measured in 174 patients in cardiogenic shock and high cDPP3 levels were associated with an increased short-term mortality risk (standardized hazard ratio: 1.4 (1.1-1.8)) and severe organ dysfunction. Additionally, a rapid decrease in cDPP3 in cardiogenic shock patients within 24 h of admission was associated with a favourable outcome. This study showed that injection of DPP3 induced myocardial depression (-10 ± 2% of shortening fraction) and impaired kidney haemodynamics (+0.30 ± 0.02 of renal resistive index) in healthy mice. cDPP3 inhibition by Procizumab, a specific antibody directed against cDPP3, promptly normalized cardiac function and kidney haemodynamics in an acute heart failure mouse model, with a marked reduction in oxidative stress and inflammatory signalling. Our study demonstrated cDPP3 is a newly discovered myocardial depressant factor, the levels of which at admission are associated with mortality in severe HF patients. Furthermore, inhibition of cDPP3 by Procizumab improved haemodynamics in a mouse model of HF. Our results suggest that DPP3 could be a new biomarker and biotarget for severe HF.

Identifiants

pubmed: 31472040
doi: 10.1002/ejhf.1601
doi:

Substances chimiques

Anti-Arrhythmia Agents 0
Antibodies, Monoclonal, Humanized 0
Biomarkers 0
procizumab 0
Dipeptidyl-Peptidases and Tripeptidyl-Peptidases EC 3.4.14.-
DPP3 protein, human EC 3.4.14.4

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

290-299

Subventions

Organisme : Aarne Koskelo Foundation
Pays : International
Organisme : Finnish Cardiac Foundation
Pays : International
Organisme : Investitionsbank des Landes Brandenburg (ILB)
Pays : International

Commentaires et corrections

Type : CommentIn

Informations de copyright

© 2019 The Authors. European Journal of Heart Failure © 2019 European Society of Cardiology.

Références

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Auteurs

Benjamin Deniau (B)

Inserm UMR-S 942, Cardiovascular Markers in Stress Conditions (MASCOT), University of Paris, Paris, France.

Linda Rehfeld (L)

4TEEN4 Pharmaceuticals GmbH, Hennigsdorf, Germany.

Karine Santos (K)

4TEEN4 Pharmaceuticals GmbH, Hennigsdorf, Germany.

Anke Dienelt (A)

4TEEN4 Pharmaceuticals GmbH, Hennigsdorf, Germany.

Feriel Azibani (F)

Inserm UMR-S 942, Cardiovascular Markers in Stress Conditions (MASCOT), University of Paris, Paris, France.

Malha Sadoune (M)

Inserm UMR-S 942, Cardiovascular Markers in Stress Conditions (MASCOT), University of Paris, Paris, France.

Paul R Kounde (PR)

Inserm UMR-S 942, Cardiovascular Markers in Stress Conditions (MASCOT), University of Paris, Paris, France.

Jane L Samuel (JL)

Inserm UMR-S 942, Cardiovascular Markers in Stress Conditions (MASCOT), University of Paris, Paris, France.

Heli Tolpannen (H)

Cardiology, University of Helsinki, Heart and Lung Center, Helsinki University Hospital, Helsinki, Finland.
Emergency Medicine, University of Helsinki, Helsinki University Hospital, Helsinki, Finland.

Johan Lassus (J)

Cardiology, University of Helsinki, Heart and Lung Center, Helsinki University Hospital, Helsinki, Finland.

Veli-Pekka Harjola (VP)

Emergency Medicine, University of Helsinki, Helsinki University Hospital, Helsinki, Finland.

Nicolas Vodovar (N)

Inserm UMR-S 942, Cardiovascular Markers in Stress Conditions (MASCOT), University of Paris, Paris, France.

Andreas Bergmann (A)

4TEEN4 Pharmaceuticals GmbH, Hennigsdorf, Germany.
Sphingotec GmbH, Hennigsdorf, Germany.

Oliver Hartmann (O)

4TEEN4 Pharmaceuticals GmbH, Hennigsdorf, Germany.
Sphingotec GmbH, Hennigsdorf, Germany.

Alexandre Mebazaa (A)

Inserm UMR-S 942, Cardiovascular Markers in Stress Conditions (MASCOT), University of Paris, Paris, France.
Department of Anaesthesiology, Burn and Critical Care, University Hospitals Saint-Louis-Lariboisière, AP-HP, Paris, France.

Alice Blet (A)

Inserm UMR-S 942, Cardiovascular Markers in Stress Conditions (MASCOT), University of Paris, Paris, France.
Department of Anaesthesiology, Burn and Critical Care, University Hospitals Saint-Louis-Lariboisière, AP-HP, Paris, France.

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Classifications MeSH