Histamine Receptors Regulate the Activity, Surface Expression, and Phosphorylation of Serotonin Transporters.
Histamine
clearance
depolarization
histamine H3 receptor
serotonin
serotonin transporter
Journal
ACS chemical neuroscience
ISSN: 1948-7193
Titre abrégé: ACS Chem Neurosci
Pays: United States
ID NLM: 101525337
Informations de publication
Date de publication:
05 02 2020
05 02 2020
Historique:
pubmed:
10
1
2020
medline:
4
3
2021
entrez:
10
1
2020
Statut:
ppublish
Résumé
Reuptake and clearance of released serotonin (5-HT) are critical in serotonergic neurotransmission. Serotonin transporter (SERT) is mainly responsible for clearing the extracellular 5-HT. Controlled trafficking, phosphorylation, and protein stability have been attributed to robust SERT activity. H
Identifiants
pubmed: 31916747
doi: 10.1021/acschemneuro.9b00664
pmc: PMC7004881
mid: NIHMS1068244
doi:
Substances chimiques
Receptors, Histamine
0
Serotonin Plasma Membrane Transport Proteins
0
Serotonin
333DO1RDJY
Types de publication
Journal Article
Research Support, N.I.H., Extramural
Langues
eng
Sous-ensembles de citation
IM
Pagination
466-476Subventions
Organisme : NIMH NIH HHS
ID : R01 MH062612
Pays : United States
Organisme : NIMH NIH HHS
ID : R01 MH112731
Pays : United States
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