Structure-Activity Relationship between Thiol Group-Trapping Ability of Morphinan Compounds with a Michael Acceptor and Anti-
1H-NMR experiments
BNTX
mechanism elucidation
morphinan
δ opioid receptor antagonist
Journal
Molecules (Basel, Switzerland)
ISSN: 1420-3049
Titre abrégé: Molecules
Pays: Switzerland
ID NLM: 100964009
Informations de publication
Date de publication:
02 Mar 2020
02 Mar 2020
Historique:
received:
24
01
2020
revised:
28
02
2020
accepted:
28
02
2020
entrez:
6
3
2020
pubmed:
7
3
2020
medline:
15
12
2020
Statut:
epublish
Résumé
7-Benzylidenenaltrexone (BNTX) and most of its derivatives showed in vitro antimalarial activities against chloroquine-resistant and -sensitive
Identifiants
pubmed: 32131542
pii: molecules25051112
doi: 10.3390/molecules25051112
pmc: PMC7179212
pii:
doi:
Substances chimiques
Antimalarials
0
Benzylidene Compounds
0
Morphinans
0
7-benzylidenenaltrexone
129468-28-6
Naltrexone
5S6W795CQM
Types de publication
Journal Article
Langues
eng
Sous-ensembles de citation
IM
Références
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