Inhibition of GPR91 Reduces Inflammatory Mediators Involved in Active Labor in Myometrium.


Journal

Mediators of inflammation
ISSN: 1466-1861
Titre abrégé: Mediators Inflamm
Pays: United States
ID NLM: 9209001

Informations de publication

Date de publication:
2020
Historique:
received: 01 12 2019
revised: 25 02 2020
accepted: 12 03 2020
entrez: 8 5 2020
pubmed: 8 5 2020
medline: 18 5 2021
Statut: epublish

Résumé

GPR91 mRNA expression was significantly higher in myometrium from women during term spontaneous labor compared to no labor. Likewise, in mice, GPR91 mRNA expression was significantly upregulated in myometrium during inflammation-induced preterm labor compared to preterm no labor. In myometrial cells, IL1B and TNF significantly increased GPR91 mRNA expression. Knockdown of GPR91 by siRNA in myometrial cells significantly suppressed the secretion and/or expression of IL1B- and TNF-induced proinflammatory cytokines (GM-CSF, IL1A, IL1B, and IL6) and chemokines (CXCL8 and CCL2), myometrial contractility (expression of the contraction-associated proteins PTGFR and CX43, secretion of the uterotonic PGF Our findings demonstrate that GPR91 is involved in the genesis of proinflammatory and prolabor mediators induced by IL1B or TNF and collectively suggest that GPR91 may contribute to augmentation of the labor processes.

Identifiants

pubmed: 32377163
doi: 10.1155/2020/6454282
pmc: PMC7180404
doi:

Substances chimiques

Inflammation Mediators 0
NF-kappa B 0
Receptors, G-Protein-Coupled 0
SUCNR1 protein, human 0

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

6454282

Informations de copyright

Copyright © 2020 Ratana Lim and Martha Lappas.

Déclaration de conflit d'intérêts

The authors have nothing to declare.

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Auteurs

Ratana Lim (R)

Obstetrics, Nutrition and Endocrinology Group, Department of Obstetrics and Gynaecology, University of Melbourne, Victoria, Australia.
Mercy Perinatal Research Centre, Mercy Hospital for Women, Heidelberg, Victoria, Australia.

Martha Lappas (M)

Obstetrics, Nutrition and Endocrinology Group, Department of Obstetrics and Gynaecology, University of Melbourne, Victoria, Australia.
Mercy Perinatal Research Centre, Mercy Hospital for Women, Heidelberg, Victoria, Australia.

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