In vivo evaluation of effects of histamine H
Animals
Central Nervous System Stimulants
/ administration & dosage
Dose-Response Relationship, Drug
Drug Evaluation, Preclinical
/ methods
Histamine H3 Antagonists
/ administration & dosage
Hyperkinesis
/ chemically induced
Injections, Intraperitoneal
Locomotion
/ drug effects
Male
Methamphetamine
/ administration & dosage
Mice
Mice, Inbred ICR
Morpholines
/ administration & dosage
Piperidines
/ administration & dosage
Conessine
Histamine H(3) receptor antagonist
Hyperlocomotion
JNJ-10181457
Methamphetamine
Pitolisant
Journal
Brain research
ISSN: 1872-6240
Titre abrégé: Brain Res
Pays: Netherlands
ID NLM: 0045503
Informations de publication
Date de publication:
01 08 2020
01 08 2020
Historique:
received:
14
03
2020
revised:
15
04
2020
accepted:
01
05
2020
pubmed:
11
5
2020
medline:
2
9
2021
entrez:
11
5
2020
Statut:
ppublish
Résumé
A single administration with METH (3 mg/kg) induced a hyperlocomotion in male ICR mice. Pretreatment of mice with pitolisant, a histamine H
Identifiants
pubmed: 32387137
pii: S0006-8993(20)30229-8
doi: 10.1016/j.brainres.2020.146873
pii:
doi:
Substances chimiques
4-(3-(4-piperidin-1-ylbut-1-ynyl)benzyl)morpholine
0
Central Nervous System Stimulants
0
Histamine H3 Antagonists
0
Morpholines
0
Piperidines
0
Methamphetamine
44RAL3456C
pitolisant
4BC83L4PIY
Types de publication
Journal Article
Research Support, Non-U.S. Gov't
Langues
eng
Sous-ensembles de citation
IM
Pagination
146873Informations de copyright
Copyright © 2020 Elsevier B.V. All rights reserved.
Déclaration de conflit d'intérêts
Declaration of Competing Interest The authors declare that they have no known competing financial interests or personal relationships that could have appeared to influence the work reported in this paper.