Inhibition of Acetylcholinesterases by Stereoisomeric Organophosphorus Compounds Containing Both Thioester and


Journal

Chemical research in toxicology
ISSN: 1520-5010
Titre abrégé: Chem Res Toxicol
Pays: United States
ID NLM: 8807448

Informations de publication

Date de publication:
21 09 2020
Historique:
pubmed: 25 8 2020
medline: 24 8 2021
entrez: 25 8 2020
Statut: ppublish

Résumé

Studies with acetylcholinesterase (AChE) inhibited by organophosphorus (OP) compounds with two chiral centers can serve as models or surrogates for understanding the rate, orientation, and postinhibitory mechanisms by the nerve agent soman that possesses dual phosphorus and carbon chiral centers. In the current approach, stereoisomers of

Identifiants

pubmed: 32833441
doi: 10.1021/acs.chemrestox.0c00236
doi:

Substances chimiques

Cholinesterase Inhibitors 0
Esters 0
Nitrophenols 0
Organophosphorus Compounds 0
Sulfhydryl Compounds 0
4-nitrophenyl acetate 830-03-5
Acetylcholinesterase EC 3.1.1.7

Types de publication

Journal Article Research Support, N.I.H., Extramural

Langues

eng

Sous-ensembles de citation

IM

Pagination

2455-2466

Subventions

Organisme : NINDS NIH HHS
ID : U01 NS092495
Pays : United States

Auteurs

Todd T Talley (TT)

Department of Biomedical and Pharmaceutical Sciences, The University of Montana, Missoula, Montana 59812, United States.

Chih-Kai Chao (CK)

Department of Biomedical and Pharmaceutical Sciences, The University of Montana, Missoula, Montana 59812, United States.

Clifford E Berkman (CE)

Department of Chemistry and Biochemistry, Washington State University, Pullman, Washington 99164, United States.

Rudy J Richardson (RJ)

Departments of Environmental Health Sciences and Neurology, University of Michigan, Ann Arbor, Michigan 48109, United States.
Center of Computational Medicine and Bioinformatics, University of Michigan, Ann Arbor, Michigan 48109, United States.

Charles M Thompson (CM)

Department of Biomedical and Pharmaceutical Sciences, The University of Montana, Missoula, Montana 59812, United States.

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Classifications MeSH