Compound heterozygosity for PTPN11 variants in a subject with Noonan syndrome provides insights into the mechanism of SHP2-related disorders.


Journal

Clinical genetics
ISSN: 1399-0004
Titre abrégé: Clin Genet
Pays: Denmark
ID NLM: 0253664

Informations de publication

Date de publication:
03 2021
Historique:
received: 28 09 2020
revised: 26 11 2020
accepted: 19 12 2020
pubmed: 24 12 2020
medline: 1 1 2022
entrez: 23 12 2020
Statut: ppublish

Résumé

The RASopathies are a family of clinically related disorders caused by mutations affecting genes participating in the RAS-MAPK signaling cascade. Among them, Noonan syndrome (NS) and Noonan syndrome with multiple lentigines (NSML) are allelic conditions principally associated with dominant mutations in PTPN11, which encodes the nonreceptor SH2 domain-containing protein tyrosine phosphatase SHP2. Individual PTPN11 mutations are specific to each syndrome and have opposite consequences on catalysis, but all favor SHP2's interaction with signaling partners. Here, we report on a subject with NS harboring biallelic variants in PTPN11. While the former (p.Leu261Phe) had previously been reported in NS, the latter (p.Thr357Met) is a novel change impairing catalysis. Members of the family carrying p.Thr357Met, however, did not show any obvious feature fitting NSML or within the RASopathy phenotypic spectrum. A major impact of this change on transcript processing and protein stability was excluded. These findings further support the view that NSML cannot be ascribed merely to impaired SHP2's catalytic activity and suggest that PTPN11 mutations causing this condition act through an alternative dominant mechanism.

Identifiants

pubmed: 33354767
doi: 10.1111/cge.13904
doi:

Substances chimiques

PTPN11 protein, human EC 3.1.3.48
Protein Tyrosine Phosphatase, Non-Receptor Type 11 EC 3.1.3.48

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

457-461

Informations de copyright

© 2020 John Wiley & Sons A/S. Published by John Wiley & Sons Ltd.

Références

Rauen KA. The RASopathies. Annu Rev Genomics Hum Genet. 2013;14:355-369.
Roberts AE, Allanson JE, Tartaglia M, Gelb BD. Noonan syndrome. Lancet. 2013;381:333-342.
Neel BG, Gu H, Pao L. The 'Shp'ing news: SH2 domain-containing tyrosine phosphatases in cell signaling. Trends Biochem Sci. 2003;28:284-293.
Sarkozy A, Digilio MC, Dallapiccola B. Leopard syndrome. Orphanet J Rare Dis. 2008;3:13.
Tartaglia M, Gelb BD, Zenker M. Noonan syndrome and clinically related disorders. Best Pract Res Clin Endocrinol Metab. 2011;25:161-179.
Hof P, Pluskey S, Dhe-Paganon S, Eck MJ, Shoelson SE. Crystal structure of the tyrosine phosphatase SHP-2. Cell. 1998;92:441-450.
Bocchinfuso G, Stella L, Martinelli S, et al. Structural and functional effects of disease-causing amino acid substitutions affecting residues Ala72 and Glu76 of the protein tyrosine phosphatase SHP-2. Proteins. 2007;66:963-974.
Keilhack H, David FS, McGregor M, Cantley LC, Neel BG. Diverse biochemical properties of Shp2 mutants. Implications for disease phenotypes. J Biol Chem. 2005;280:30984-30993.
Tartaglia M, Martinelli S, Stella L, et al. Diversity and functional consequences of germline and somatic PTPN11 mutations in human disease. Am J Hum Genet. 2006;78:279-290.
Fragale A, Tartaglia M, Wu J, Gelb BD. Noonan syndrome-associated SHP2/PTPN11 mutants cause EGF-dependent prolonged GAB1 binding and sustained ERK2/MAPK1 activation. Hum Mutat. 2004;23:267-277.
Araki T, Mohi MG, Ismat FA, et al. Mouse model of Noonan syndrome reveals cell type- and gene dosage-dependent effects of Ptpn11 mutation. Nat Med. 2004;10:849-857.
Hanna N, Montagner A, Lee WH, et al. Reduced phosphatase activity of SHP-2 in LEOPARD syndrome: consequences for PI3K binding on Gab1. FEBS Lett. 2006;580:2477-2482.
Martinelli S, Torreri P, Tinti M, et al. Diverse driving forces underlie the invariant occurrence of the T42A, E139D, I282V and T468M SHP2 amino acid substitutions causing Noonan and LEOPARD syndromes. Hum Mol Genet. 2008;17:2018-2029.
Edouard T, Combier JP, Nedelec A, et al. Functional effects of PTPN11 (SHP2) mutations causing LEOPARD syndrome on epidermal growth factor-induced phosphoinositide 3-kinase/AKT/glycogen synthase kinase 3beta signaling. Mol Cell Biol. 2010;30:2498-2507.
Yu ZH, Xu J, Walls CD, et al. Structural and mechanistic insights into LEOPARD syndrome-associated SHP2Mutations. J Biol Chem. 2013;288:10472-10482.
Yu ZH, Zhang RY, Walls CD, et al. Molecular basis of gain-of-function LEOPARD syndrome-associated SHP2 mutations. Biochemistry. 2014;53:4136-4151.
Pannone L, Bocchinfuso G, Flex E, et al. Structural, functional, and clinical characterization of a novel PTPN11 mutation cluster underlying Noonan syndrome. Hum Mutat. 2017;38:451-459.
Ezquieta B, Santome JL, Carcavilla A, et al. Alterations in RAS-MAPK genes in 200 Spanish patients with Noonan and other neuro-cardio-facio-cutaneous syndromes. Genotype and cardiopathy. Rev Esp Cardiol (Engl Ed). 2012;65:447-455.
Andersen JN, Mortensen OH, Peters GH, et al. Structural and evolutionary relationships among protein tyrosine phosphatase domains. Mol Cell Biol. 2001;21:7117-7136.
Zhu G, Xie J, Kong W, et al. Phase separation of disease-associated SHP2 mutants underlies MAPK Hyperactivation. Cell. 2020;183:490-502.
Bowen ME, Boyden ED, Holm IA, et al. Loss-of-function mutations in PTPN11 cause metachondromatosis, but not Ollier disease or Maffucci syndrome. PLoS Genet. 2011;7:e1002050.

Auteurs

Rebeca Lorca (R)

Unidad de Referencia de Cardiopatías Familiares-HUCA, Hospital Universitario Central de Asturias (HUCA) - Instituto de Investigación Sanitaria del Principado de Asturias (ISPA), Oviedo, Spain.

Luca Pannone (L)

Genetics and Rare Diseases Research Division, Ospedale Pediatrico Bambino Gesù, IRCCS, Rome, Italy.

Elías Cuesta-Llavona (E)

Unidad de Referencia de Cardiopatías Familiares-HUCA, Hospital Universitario Central de Asturias (HUCA) - Instituto de Investigación Sanitaria del Principado de Asturias (ISPA), Oviedo, Spain.
Grupo Eje Cardio-Renal, Instituto de Investigación Sanitaria del Principado de Asturias, Oviedo, Spain.

Gianfranco Bocchinfuso (G)

Dipartimento di Scienze e Tecnologie Chimiche, Università di Roma Tor Vergata, Rome, Italy.

Julian Rodríguez-Reguero (J)

Unidad de Referencia de Cardiopatías Familiares-HUCA, Hospital Universitario Central de Asturias (HUCA) - Instituto de Investigación Sanitaria del Principado de Asturias (ISPA), Oviedo, Spain.
Grupo Eje Cardio-Renal, Instituto de Investigación Sanitaria del Principado de Asturias, Oviedo, Spain.

Giovanna Carpentieri (G)

Genetics and Rare Diseases Research Division, Ospedale Pediatrico Bambino Gesù, IRCCS, Rome, Italy.

Inés Hernando (I)

Unidad de Referencia de Cardiopatías Familiares-HUCA, Hospital Universitario Central de Asturias (HUCA) - Instituto de Investigación Sanitaria del Principado de Asturias (ISPA), Oviedo, Spain.

Elisabetta Flex (E)

Department of Oncology and Molecular Medicine, Istituto Superiore di Sanità, Rome, Italy.

Marco Tartaglia (M)

Genetics and Rare Diseases Research Division, Ospedale Pediatrico Bambino Gesù, IRCCS, Rome, Italy.

Eliecer Coto (E)

Unidad de Referencia de Cardiopatías Familiares-HUCA, Hospital Universitario Central de Asturias (HUCA) - Instituto de Investigación Sanitaria del Principado de Asturias (ISPA), Oviedo, Spain.
Grupo Eje Cardio-Renal, Instituto de Investigación Sanitaria del Principado de Asturias, Oviedo, Spain.
Medicine Department, Universidad de Oviedo, Oviedo, Spain.
HUCA. Eje Cardio-Renal, Red de Investigación Renal (REDINREN), Madrid, Spain.

Juan Gómez (J)

Unidad de Referencia de Cardiopatías Familiares-HUCA, Hospital Universitario Central de Asturias (HUCA) - Instituto de Investigación Sanitaria del Principado de Asturias (ISPA), Oviedo, Spain.
Grupo Eje Cardio-Renal, Instituto de Investigación Sanitaria del Principado de Asturias, Oviedo, Spain.
HUCA. Eje Cardio-Renal, Red de Investigación Renal (REDINREN), Madrid, Spain.

Simone Martinelli (S)

Department of Oncology and Molecular Medicine, Istituto Superiore di Sanità, Rome, Italy.

Articles similaires

[Redispensing of expensive oral anticancer medicines: a practical application].

Lisanne N van Merendonk, Kübra Akgöl, Bastiaan Nuijen
1.00
Humans Antineoplastic Agents Administration, Oral Drug Costs Counterfeit Drugs

Smoking Cessation and Incident Cardiovascular Disease.

Jun Hwan Cho, Seung Yong Shin, Hoseob Kim et al.
1.00
Humans Male Smoking Cessation Cardiovascular Diseases Female
Humans United States Aged Cross-Sectional Studies Medicare Part C
1.00
Humans Yoga Low Back Pain Female Male

Classifications MeSH