Jorunnamycin A Suppresses Stem-Like Phenotypes and Sensitizes Cisplatin-Induced Apoptosis in Cancer Stem-Like Cell-Enriched Spheroids of Human Lung Cancer Cells.


Journal

Marine drugs
ISSN: 1660-3397
Titre abrégé: Mar Drugs
Pays: Switzerland
ID NLM: 101213729

Informations de publication

Date de publication:
03 May 2021
Historique:
received: 04 04 2021
revised: 29 04 2021
accepted: 30 04 2021
entrez: 2 6 2021
pubmed: 3 6 2021
medline: 17 11 2021
Statut: epublish

Résumé

It has been recognized that cancer stem-like cells (CSCs) in tumor tissue crucially contribute to therapeutic failure, resulting in a high mortality rate in lung cancer patients. Due to their stem-like features of self-renewal and tumor formation, CSCs can lead to drug resistance and tumor recurrence. Herein, the suppressive effect of jorunnamycin A, a bistetrahydroisoquinolinequinone isolated from Thai blue sponge

Identifiants

pubmed: 34063628
pii: md19050261
doi: 10.3390/md19050261
pmc: PMC8147647
pii:
doi:

Substances chimiques

BCL2 protein, human 0
Isoquinolines 0
NANOG protein, human 0
Nanog Homeobox Protein 0
Octamer Transcription Factor-3 0
POU5F1 protein, human 0
Proto-Oncogene Proteins c-bcl-2 0
Quinolones 0
SOX2 protein, human 0
SOXB1 Transcription Factors 0
TP53 protein, human 0
Transcription Factors 0
Tumor Suppressor Protein p53 0
jorunnamycin A 0
Cisplatin Q20Q21Q62J

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Subventions

Organisme : Chulalongkorn University
ID : 90th Anniversary of Chulalongkorn University
Organisme : Chulalongkorn University
ID : Ratchadaphiseksomphot Endowment Fund (grant no. CU_GR_62_20_33_01)
Organisme : National Research Council of Thailand (NRCT)
ID : Mid-Career Research Grant (RSA 6280009)

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Auteurs

Somruethai Sumkhemthong (S)

Department of Biochemistry and Microbiology, Faculty of Pharmaceutical Sciences, Chulalongkorn University, Bangkok 10330, Thailand.

Supakarn Chamni (S)

Department of Pharmacognosy and Pharmaceutical Botany, Faculty of Pharmaceutical Sciences, Chulalongkorn University, Bangkok 10330, Thailand.
Natural Products and Nanoparticles Research Unit (NP2), Chulalongkorn University, Bangkok 10330, Thailand.

Gea U Ecoy (GU)

Department of Biochemistry and Microbiology, Faculty of Pharmaceutical Sciences, Chulalongkorn University, Bangkok 10330, Thailand.
Department of Pharmacy, School of Health Care Professions, University of San Carlos, Cebu 6000, Philippines.

Pornchanok Taweecheep (P)

Department of Biochemistry and Microbiology, Faculty of Pharmaceutical Sciences, Chulalongkorn University, Bangkok 10330, Thailand.

Khanit Suwanborirux (K)

Department of Pharmacognosy and Pharmaceutical Botany, Faculty of Pharmaceutical Sciences, Chulalongkorn University, Bangkok 10330, Thailand.
Natural Products and Nanoparticles Research Unit (NP2), Chulalongkorn University, Bangkok 10330, Thailand.

Eakachai Prompetchara (E)

Department of Laboratory Medicine, Faculty of Medicine, Chulalongkorn University, Bangkok 10330, Thailand.
Center of Excellence in Vaccine Research and Development (Chula Vaccine Research Center-Chula VRC), Faculty of Medicine, Chulalongkorn University, Bangkok 10330, Thailand.

Pithi Chanvorachote (P)

Department of Pharmacology and Physiology, Faculty of Pharmaceutical Sciences, Chulalongkorn University, Bangkok 10330, Thailand.
Cell-Based Drug and Health Products Development Research Unit, Faculty of Pharmaceutical Sciences, Chulalongkorn University, Bangkok 10330, Thailand.

Chatchai Chaotham (C)

Department of Biochemistry and Microbiology, Faculty of Pharmaceutical Sciences, Chulalongkorn University, Bangkok 10330, Thailand.
Cell-Based Drug and Health Products Development Research Unit, Faculty of Pharmaceutical Sciences, Chulalongkorn University, Bangkok 10330, Thailand.

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