Siglec-6 is a novel target for CAR T-cell therapy in acute myeloid leukemia.


Journal

Blood
ISSN: 1528-0020
Titre abrégé: Blood
Pays: United States
ID NLM: 7603509

Informations de publication

Date de publication:
11 11 2021
Historique:
received: 17 09 2020
accepted: 26 06 2021
pubmed: 22 7 2021
medline: 22 12 2021
entrez: 21 7 2021
Statut: ppublish

Résumé

Acute myeloid leukemia (AML) is an attractive entity for the development of chimeric antigen receptor (CAR) T-cell immunotherapy because AML blasts are susceptible to T-cell-mediated elimination. Here, we introduce sialic acid-binding immunoglobulin-like lectin 6 (Siglec-6) as a novel target for CAR T cells in AML. We designed a Siglec-6-specific CAR with a targeting domain derived from the human monoclonal antibody JML-1. We found that Siglec-6 is commonly expressed on AML cell lines and primary AML blasts, including the subpopulation of AML stem cells. Treatment with Siglec-6 CAR T cells confers specific antileukemia reactivity that correlates with Siglec-6 expression in preclinical models, including induction of complete remission in a xenograft AML model in immunodeficient mice (NSG/U937). In addition, we confirmed Siglec-6 expression on transformed B cells in chronic lymphocytic leukemia (CLL), and specific anti-CLL reactivity of Siglec-6 CAR T cells in vitro. Of particular interest, we found that Siglec-6 is not detectable on normal hematopoietic stem and progenitor cells (HSPCs) and that treatment with Siglec-6 CAR T cells does not affect their viability and lineage differentiation in colony-formation assays. These data suggest that Siglec-6 CAR T-cell therapy may be used to effectively treat AML without the need for subsequent allogeneic hematopoietic stem cell transplantation. In mature normal hematopoietic cells, we detected Siglec-6 in a proportion of memory (and naïve) B cells and basophilic granulocytes, suggesting the potential for limited on-target/off-tumor reactivity. The lack of expression of Siglec-6 on normal HSPCs is a key to differentiating it from other Siglec family members (eg, Siglec-3 [CD33]) and other CAR target antigens (eg, CD123) that are under investigation in AML, and it warrants the clinical investigation of Siglec-6 CAR T-cell therapy.

Identifiants

pubmed: 34289026
pii: S0006-4971(21)01374-4
doi: 10.1182/blood.2020009192
pmc: PMC9642786
doi:

Substances chimiques

Antigens, CD 0
Antigens, Differentiation, Myelomonocytic 0
Lectins 0
SIGLEC6 protein, human 0

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

1830-1842

Commentaires et corrections

Type : CommentIn

Informations de copyright

© 2021 by The American Society of Hematology.

Références

Blood Cancer J. 2016 Jul 01;6(7):e441
pubmed: 27367478
Blood Cancer J. 2014 Jun 13;4:e218
pubmed: 24927407
Nat Med. 2018 Jan;24(1):20-28
pubmed: 29155426
J Immunol. 2015 Feb 1;194(3):911-20
pubmed: 25520398
Front Immunol. 2018 Sep 20;9:2138
pubmed: 30294327
J Immunol. 1995 May 1;154(9):4466-75
pubmed: 7722303
N Engl J Med. 2019 May 2;380(18):1726-1737
pubmed: 31042825
Blood. 2021 Jul 29;138(4):318-330
pubmed: 34323938
Nat Commun. 2019 Jul 17;10(1):3137
pubmed: 31316055
Leukemia. 2015 Aug;29(8):1637-47
pubmed: 25721896
Cancer Discov. 2015 Dec;5(12):1282-95
pubmed: 26516065
N Engl J Med. 2018 Feb 1;378(5):439-448
pubmed: 29385370
Blood. 2009 Jan 15;113(3):635-45
pubmed: 18974375
Exp Hematol. 2006 Jun;34(6):728-35
pubmed: 16728277
Cell. 2018 May 31;173(6):1439-1453.e19
pubmed: 29856956
Blood. 2010 Nov 25;116(22):4532-41
pubmed: 20702778
Immunology. 2001 Jun;103(2):137-45
pubmed: 11412300
Leukemia. 2019 Jan;33(1):64-74
pubmed: 29946192
Allergy. 2006 Jun;61(6):769-76
pubmed: 16677248
N Engl J Med. 2014 Oct 16;371(16):1507-17
pubmed: 25317870
Blood. 2017 Mar 23;129(12):1577-1585
pubmed: 28159741
Blood. 2020 Jan 9;135(2):85-96
pubmed: 31765470
Nat Med. 2018 Oct;24(10):1504-1506
pubmed: 30275569
Mol Ther. 2017 Sep 6;25(9):2189-2201
pubmed: 28676342
Blood. 2014 Apr 10;123(15):2343-54
pubmed: 24596416
Nat Commun. 2016 Jul 27;7:12320
pubmed: 27460500
Blood. 2016 Sep 29;128(13):1688-700
pubmed: 27412889
J Biol Chem. 1999 Aug 6;274(32):22729-38
pubmed: 10428856
Immunity. 2016 Feb 16;44(2):380-90
pubmed: 26885860
J Clin Invest. 2016 Jun 1;126(6):2123-38
pubmed: 27111235
Leukemia. 2018 May;32(5):1168-1179
pubmed: 29472720
Blood. 2020 May 7;135(19):1650-1660
pubmed: 32076701
Leukemia. 2016 Jun;30(6):1355-64
pubmed: 26898190
Glycobiology. 2007 Sep;17(9):922-31
pubmed: 17580316
Mol Ther. 2019 Jan 2;27(1):272-280
pubmed: 30391141
Leukemia. 2021 Sep;35(9):2581-2591
pubmed: 33633313
J Clin Pathol. 1998 May;51(5):364-9
pubmed: 9708202
Cancer Immunol Res. 2018 Sep;6(9):1008-1013
pubmed: 29980538
Oncoimmunology. 2012 Sep 1;1(6):863-873
pubmed: 23162754
N Engl J Med. 2018 Feb 1;378(5):449-459
pubmed: 29385376
Mol Ther. 2017 Sep 6;25(9):2202-2213
pubmed: 28676343
Blood. 2009 Nov 12;114(20):4494-502
pubmed: 19667400

Auteurs

Hardikkumar Jetani (H)

Medizinische Klinik und Poliklinik II, Universitätsklinikum Würzburg, Würzburg, Germany.

Almudena Navarro-Bailón (A)

Medizinische Klinik und Poliklinik II, Universitätsklinikum Würzburg, Würzburg, Germany.
Servicio de Hematología, Hospital Universitario de Salamanca-Instituto de Investigación Biomédica de Salamanca, Centro de Investigación Biomédica en Red de Cáncer (CB16/12/00233), Centro de Investigación del Cáncer-Instituto de Biología Molecular y Celular del Cáncer, Universidad de Salamanca-Consejo Superior de Investigaciones Científicas, Salamanca, Spain.

Marius Maucher (M)

Medizinische Klinik und Poliklinik II, Universitätsklinikum Würzburg, Würzburg, Germany.

Silke Frenz (S)

Medizinische Klinik und Poliklinik II, Universitätsklinikum Würzburg, Würzburg, Germany.

Christina Verbruggen (C)

Lehrstuhl für Biotechnologie und Biophysik, Biozentrum, Universität Würzburg, Würzburg, Germany.

Ana Yeguas (A)

Servicio de Hematología, Hospital Universitario de Salamanca-Instituto de Investigación Biomédica de Salamanca, Centro de Investigación Biomédica en Red de Cáncer (CB16/12/00233), Centro de Investigación del Cáncer-Instituto de Biología Molecular y Celular del Cáncer, Universidad de Salamanca-Consejo Superior de Investigaciones Científicas, Salamanca, Spain.

María Belén Vidriales (MB)

Servicio de Hematología, Hospital Universitario de Salamanca-Instituto de Investigación Biomédica de Salamanca, Centro de Investigación Biomédica en Red de Cáncer (CB16/12/00233), Centro de Investigación del Cáncer-Instituto de Biología Molecular y Celular del Cáncer, Universidad de Salamanca-Consejo Superior de Investigaciones Científicas, Salamanca, Spain.

Marcos González (M)

Servicio de Hematología, Hospital Universitario de Salamanca-Instituto de Investigación Biomédica de Salamanca, Centro de Investigación Biomédica en Red de Cáncer (CB16/12/00233), Centro de Investigación del Cáncer-Instituto de Biología Molecular y Celular del Cáncer, Universidad de Salamanca-Consejo Superior de Investigaciones Científicas, Salamanca, Spain.

Judit Rial Saborido (J)

Medizinische Klinik 5, Hämatologie und Onkologie, Universitätsklinikum Erlangen-Nürnberg, Erlangen, Germany.

Sabrina Kraus (S)

Medizinische Klinik und Poliklinik II, Universitätsklinikum Würzburg, Würzburg, Germany.

Katrin Mestermann (K)

Medizinische Klinik und Poliklinik II, Universitätsklinikum Würzburg, Würzburg, Germany.

Simone Thomas (S)

Klinik und Poliklinik für Innere Medizin III, Universitätsklinikum Regensburg, Regensburg, Germany.
Regensburger Centrum für Interventionelle Immunologie, Regensburg, Germany.

Halvard Bonig (H)

Institut für Transfusionsmedizin und Immunhämatologie, Goethe Universität Frankfurt, Frankfurt am Main, Germany; and.
Deutsches Rote Kreuz Blutspendedienst BaWüHe, Frankfurt, Germany.

Maik Luu (M)

Medizinische Klinik und Poliklinik II, Universitätsklinikum Würzburg, Würzburg, Germany.

Razieh Monjezi (R)

Medizinische Klinik und Poliklinik II, Universitätsklinikum Würzburg, Würzburg, Germany.

Dimitrios Mougiakakos (D)

Medizinische Klinik 5, Hämatologie und Onkologie, Universitätsklinikum Erlangen-Nürnberg, Erlangen, Germany.

Markus Sauer (M)

Lehrstuhl für Biotechnologie und Biophysik, Biozentrum, Universität Würzburg, Würzburg, Germany.

Hermann Einsele (H)

Medizinische Klinik und Poliklinik II, Universitätsklinikum Würzburg, Würzburg, Germany.

Michael Hudecek (M)

Medizinische Klinik und Poliklinik II, Universitätsklinikum Würzburg, Würzburg, Germany.

Articles similaires

[Redispensing of expensive oral anticancer medicines: a practical application].

Lisanne N van Merendonk, Kübra Akgöl, Bastiaan Nuijen
1.00
Humans Antineoplastic Agents Administration, Oral Drug Costs Counterfeit Drugs

Smoking Cessation and Incident Cardiovascular Disease.

Jun Hwan Cho, Seung Yong Shin, Hoseob Kim et al.
1.00
Humans Male Smoking Cessation Cardiovascular Diseases Female
Humans United States Aged Cross-Sectional Studies Medicare Part C
1.00
Humans Yoga Low Back Pain Female Male

Classifications MeSH