Enantioselective organocatalytic syntheses of α-selenated α- and β-amino acid derivatives.


Journal

Organic & biomolecular chemistry
ISSN: 1477-0539
Titre abrégé: Org Biomol Chem
Pays: England
ID NLM: 101154995

Informations de publication

Date de publication:
26 01 2022
Historique:
pubmed: 12 1 2022
medline: 9 3 2022
entrez: 11 1 2022
Statut: epublish

Résumé

Selenium-containing amino acids are valuable targets but methods for the stereoselective α-selenation of simple amino acid precursors are rare. We herein report the enantioselective electrophilic α-selenation of azlactones (masked α-amino acid derivatives) and isoxazolidin-5-ones (masked β-amino acids) using Cinchona alkaloids as easily accessible organocatalysts. A variety of differently substituted derivatives was accessed with reasonable levels of enantioselectivities and further studies concerning the stability and suitability of these compounds for further manipulations have been carried out as well.

Identifiants

pubmed: 35015015
doi: 10.1039/d1ob02235k
pmc: PMC8790592
doi:

Substances chimiques

Alkaloids 0
Amino Acids 0

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

824-830

Subventions

Organisme : Austrian Science Fund FWF
ID : P 30237
Pays : Austria
Organisme : Austrian Science Fund FWF
ID : P 31784
Pays : Austria

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Auteurs

Victoria Haider (V)

Institute of Organic Chemistry, Johannes Kepler University Linz, Altenbergerstrasse 69, 4040 Linz, Austria. mario.waser@jku.at.

Paul Zebrowski (P)

Institute of Organic Chemistry, Johannes Kepler University Linz, Altenbergerstrasse 69, 4040 Linz, Austria. mario.waser@jku.at.

Jessica Michalke (J)

Institute of Catalysis, Johannes Kepler University Linz, Altenbergerstrasse 69, 4040 Linz, Austria.

Uwe Monkowius (U)

School of Education, Chemistry, Johannes Kepler University Linz, Altenbergerstrasse 69, 4040 Linz, Austria.

Mario Waser (M)

Institute of Organic Chemistry, Johannes Kepler University Linz, Altenbergerstrasse 69, 4040 Linz, Austria. mario.waser@jku.at.

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Classifications MeSH