Biological investigation of
Escherichia coli
Thiosemicarbazones
antimicrobial agents
carbonic anhydrases
dermatophytes
Journal
Journal of enzyme inhibition and medicinal chemistry
ISSN: 1475-6374
Titre abrégé: J Enzyme Inhib Med Chem
Pays: England
ID NLM: 101150203
Informations de publication
Date de publication:
Dec 2022
Dec 2022
Historique:
entrez:
24
3
2022
pubmed:
25
3
2022
medline:
29
3
2022
Statut:
ppublish
Résumé
The enormous burden of the COVID-19 pandemic in economic and healthcare terms has cast a shadow on the serious threat of antimicrobial resistance, increasing the inappropriate use of antibiotics and shifting the focus of drug discovery programmes from antibacterial and antifungal fields. Thus, there is a pressing need for new antimicrobials involving innovative modes of action (MoAs) to avoid cross-resistance rise. Thiosemicarbazones (TSCs) stand out due to their easy preparation and polypharmacological application, also in infectious diseases. Recently, we reported a small library of TSCs (
Identifiants
pubmed: 35322729
doi: 10.1080/14756366.2022.2055009
pmc: PMC8956313
doi:
Substances chimiques
Anti-Infective Agents
0
Carbonic Anhydrase Inhibitors
0
Thiosemicarbazones
0
Carbonic Anhydrases
EC 4.2.1.1
Types de publication
Journal Article
Langues
eng
Sous-ensembles de citation
IM
Pagination
986-993Références
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