Design, synthesis and biological evaluation of novel
Alzheimer’s disease
cholinesterase inhibitory activity
hepatotoxicity
molecular docking
neurotoxicity
phosphorus tacrine analogs
tacrine
Journal
Journal of enzyme inhibition and medicinal chemistry
ISSN: 1475-6374
Titre abrégé: J Enzyme Inhib Med Chem
Pays: England
ID NLM: 101150203
Informations de publication
Date de publication:
Dec 2022
Dec 2022
Historique:
entrez:
1
4
2022
pubmed:
2
4
2022
medline:
5
4
2022
Statut:
ppublish
Résumé
In this work, we designed, synthesised and biologically investigated a novel series of 14
Identifiants
pubmed: 35361039
doi: 10.1080/14756366.2022.2045591
pmc: PMC8979514
doi:
Substances chimiques
Cholinesterase Inhibitors
0
Tacrine
4VX7YNB537
Acetylcholinesterase
EC 3.1.1.7
Types de publication
Journal Article
Langues
eng
Sous-ensembles de citation
IM
Pagination
1012-1022Références
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