Mimetics of ADP-Ribosylated Histidine through Copper(I)-Catalyzed Click Chemistry.


Journal

Organic letters
ISSN: 1523-7052
Titre abrégé: Org Lett
Pays: United States
ID NLM: 100890393

Informations de publication

Date de publication:
03 06 2022
Historique:
pubmed: 20 5 2022
medline: 7 6 2022
entrez: 19 5 2022
Statut: ppublish

Résumé

A convergent synthesis provided nearly perfect τ-ADP-ribosylated histidine isosteres (His*-τ-ADPr) via a copper(I)-catalyzed cycloaddition between an azido-ADP-ribosyl analogue and an oligopeptide carrying a propargyl glycine. Both α- and β-configured azido-ADP-ribosyl analogues have been synthesized. The former required participation of the C-2 ester functionality during glycosylation, while the latter was obtained in high stereoselectivity from an imidate donor with a nonparticipating

Identifiants

pubmed: 35587229
doi: 10.1021/acs.orglett.2c01300
pmc: PMC9171823
doi:

Substances chimiques

Histidine 4QD397987E
Adenosine Diphosphate 61D2G4IYVH
Copper 789U1901C5

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

3776-3780

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Auteurs

Hugo Minnee (H)

Bio-Organic Synthesis, Leiden Institute of Chemistry, Leiden University, P.O. Box 9502, 2300 RA Leiden, The Netherlands.

Johannes G M Rack (JGM)

Sir William Dunn School of Pathology, University of Oxford, South Parks Road, Oxford OX1 3RE, United Kingdom.

Gijsbert A van der Marel (GA)

Bio-Organic Synthesis, Leiden Institute of Chemistry, Leiden University, P.O. Box 9502, 2300 RA Leiden, The Netherlands.

Herman S Overkleeft (HS)

Bio-Organic Synthesis, Leiden Institute of Chemistry, Leiden University, P.O. Box 9502, 2300 RA Leiden, The Netherlands.

Jeroen D C Codée (JDC)

Bio-Organic Synthesis, Leiden Institute of Chemistry, Leiden University, P.O. Box 9502, 2300 RA Leiden, The Netherlands.

Ivan Ahel (I)

Sir William Dunn School of Pathology, University of Oxford, South Parks Road, Oxford OX1 3RE, United Kingdom.

Dmitri V Filippov (DV)

Bio-Organic Synthesis, Leiden Institute of Chemistry, Leiden University, P.O. Box 9502, 2300 RA Leiden, The Netherlands.

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Classifications MeSH