Fluorescent A


Journal

Purinergic signalling
ISSN: 1573-9546
Titre abrégé: Purinergic Signal
Pays: Netherlands
ID NLM: 101250499

Informations de publication

Date de publication:
09 2023
Historique:
received: 25 03 2022
accepted: 24 05 2022
medline: 23 10 2023
pubmed: 11 6 2022
entrez: 10 6 2022
Statut: ppublish

Résumé

Adenosine receptor (AR) ligands are being developed for metabolic, cardiovascular, neurological, and inflammatory diseases and cancer. The ease of drug discovery is contingent on the availability of pharmacological tools. Fluorescent antagonist ligands for the human A

Identifiants

pubmed: 35687212
doi: 10.1007/s11302-022-09873-3
pii: 10.1007/s11302-022-09873-3
pmc: PMC10539269
doi:

Substances chimiques

Purinergic P1 Receptor Antagonists 0
Fluorescent Dyes 0
Amines 0
Receptor, Adenosine A3 0
Receptor, Adenosine A2A 0
Adenosine A2 Receptor Antagonists 0

Types de publication

Journal Article Research Support, N.I.H., Intramural

Langues

eng

Sous-ensembles de citation

IM

Pagination

565-578

Subventions

Organisme : Intramural NIH HHS
ID : ZIA DK031117
Pays : United States
Organisme : NIDDK NIH HHS
ID : ZIADK031117
Pays : United States

Informations de copyright

© 2022. This is a U.S. government work and not under copyright protection in the U.S.; foreign copyright protection may apply.

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Auteurs

Kiran S Toti (KS)

Molecular Recognition Section, Laboratory of Bioorganic Chemistry, National Institute of Diabetes and Digestive and Kidney Diseases, National Institutes of Health, NIH, NIDDK, LBC, Bldg. 8A, Rm. B1A-19, Bethesda, MD, 20892-0810, USA.
Current Address: Chemistry Department, Emory University, 1093 Rollins Research Center, Atlanta, GA, 30322, USA.

Ryan G Campbell (RG)

Molecular Recognition Section, Laboratory of Bioorganic Chemistry, National Institute of Diabetes and Digestive and Kidney Diseases, National Institutes of Health, NIH, NIDDK, LBC, Bldg. 8A, Rm. B1A-19, Bethesda, MD, 20892-0810, USA.

Hobin Lee (H)

Molecular Recognition Section, Laboratory of Bioorganic Chemistry, National Institute of Diabetes and Digestive and Kidney Diseases, National Institutes of Health, NIH, NIDDK, LBC, Bldg. 8A, Rm. B1A-19, Bethesda, MD, 20892-0810, USA.

Veronica Salmaso (V)

Molecular Recognition Section, Laboratory of Bioorganic Chemistry, National Institute of Diabetes and Digestive and Kidney Diseases, National Institutes of Health, NIH, NIDDK, LBC, Bldg. 8A, Rm. B1A-19, Bethesda, MD, 20892-0810, USA.

R Rama Suresh (RR)

Molecular Recognition Section, Laboratory of Bioorganic Chemistry, National Institute of Diabetes and Digestive and Kidney Diseases, National Institutes of Health, NIH, NIDDK, LBC, Bldg. 8A, Rm. B1A-19, Bethesda, MD, 20892-0810, USA.

Zhan-Guo Gao (ZG)

Molecular Recognition Section, Laboratory of Bioorganic Chemistry, National Institute of Diabetes and Digestive and Kidney Diseases, National Institutes of Health, NIH, NIDDK, LBC, Bldg. 8A, Rm. B1A-19, Bethesda, MD, 20892-0810, USA.

Kenneth A Jacobson (KA)

Molecular Recognition Section, Laboratory of Bioorganic Chemistry, National Institute of Diabetes and Digestive and Kidney Diseases, National Institutes of Health, NIH, NIDDK, LBC, Bldg. 8A, Rm. B1A-19, Bethesda, MD, 20892-0810, USA. kennethj@niddk.nih.gov.

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Classifications MeSH