Direct Synthesis of 3-Aryl Substituted Isocoumarins and Phthalides through Palladium Acetate Catalyzed C(sp

C−H activation benzylidenephthalide ionic liquid isocoumarin palladium catalysis

Journal

Chemistry (Weinheim an der Bergstrasse, Germany)
ISSN: 1521-3765
Titre abrégé: Chemistry
Pays: Germany
ID NLM: 9513783

Informations de publication

Date de publication:
21 Nov 2022
Historique:
received: 28 07 2022
pubmed: 24 8 2022
medline: 24 11 2022
entrez: 23 8 2022
Statut: ppublish

Résumé

A novel Pd-catalysed oxidative coupling between benzoic acids and vinylarenes or acrylates to furnish isocoumarins and phthalides is reported. The reaction proceeds smoothly in molten tetrabutylammonium acetate via a selective C-H bond activation, with very low percentage of ligand-free palladium acetate as the catalyst, under atmospheric pressure of oxygen. Sub-stoichiometric amount of copper acetate is also required as a reoxidant for the palladium.

Identifiants

pubmed: 35997238
doi: 10.1002/chem.202202350
pmc: PMC9826210
doi:

Substances chimiques

Palladium 5TWQ1V240M
Isocoumarins 0
phthalide 8VV922U86J
Ionic Liquids 0
Acetates 0

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

e202202350

Subventions

Organisme : Ministero dell'Istruzione, dell'Università e della Ricerca
ID : ECOTEC _ARS 01_00951

Informations de copyright

© 2022 The Authors. Chemistry - A European Journal published by Wiley-VCH GmbH.

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Auteurs

Andrea Aloia (A)

Chemistry Department, Università degli Studi di Bari Aldo Moro, Via Orabona 4, 70126, Bari, Italy.

Michele Casiello (M)

Chemistry Department, Università degli Studi di Bari Aldo Moro, Via Orabona 4, 70126, Bari, Italy.

Lucia D'Accolti (L)

Chemistry Department, Università degli Studi di Bari Aldo Moro, Via Orabona 4, 70126, Bari, Italy.
CNR - Istituto di Chimica dei Composti Organometallici (ICCOM) Bari Section, Consiglio Nazionale delle Ricerche, Via Orabona 4, 70126, Bari, Italy.

Caterina Fusco (C)

CNR - Istituto di Chimica dei Composti Organometallici (ICCOM) Bari Section, Consiglio Nazionale delle Ricerche, Via Orabona 4, 70126, Bari, Italy.

Angelo Nacci (A)

Chemistry Department, Università degli Studi di Bari Aldo Moro, Via Orabona 4, 70126, Bari, Italy.
CNR - Istituto di Chimica dei Composti Organometallici (ICCOM) Bari Section, Consiglio Nazionale delle Ricerche, Via Orabona 4, 70126, Bari, Italy.

Antonio Monopoli (A)

Chemistry Department, Università degli Studi di Bari Aldo Moro, Via Orabona 4, 70126, Bari, Italy.
CNR - Istituto di Chimica dei Composti Organometallici (ICCOM) Bari Section, Consiglio Nazionale delle Ricerche, Via Orabona 4, 70126, Bari, Italy.

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Classifications MeSH