Dynamin-independent Ca

Ca(V)1.2 channels Dynasore Dyngo-4a K(Ca)1.1 channels Mitochondrial fission Molecular dynamic simulations

Journal

European journal of pharmacology
ISSN: 1879-0712
Titre abrégé: Eur J Pharmacol
Pays: Netherlands
ID NLM: 1254354

Informations de publication

Date de publication:
15 Jul 2023
Historique:
received: 02 01 2023
revised: 03 05 2023
accepted: 10 05 2023
medline: 5 6 2023
pubmed: 14 5 2023
entrez: 13 5 2023
Statut: ppublish

Résumé

A role for mitochondrial fission in vascular contraction has been proposed based on the vasorelaxant activity of the dynamin (and mitochondrial fission) inhibitors mdivi-1 and dynasore. However, mdivi-1 is capable to inhibit Ba

Identifiants

pubmed: 37179045
pii: S0014-2999(23)00297-2
doi: 10.1016/j.ejphar.2023.175786
pii:
doi:

Substances chimiques

dyngo-4a 0
N'-(3,4-dihydroxybenzylidene)-3-hydroxy-2-naphthahydrazide 0
3-(2,4-dichloro-5-methoxyphenyl)-2-sulfanyl-4(3H)-quinazolinone 0
Dynamins EC 3.6.5.5
Niacinamide 25X51I8RD4
Caffeine 3G6A5W338E
Phenylephrine 1WS297W6MV

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

175786

Informations de copyright

Copyright © 2023 Elsevier B.V. All rights reserved.

Déclaration de conflit d'intérêts

Declaration of competing interest The authors declare that they have no known competing financial interests or personal relationships that could have appeared to influence the work reported in this paper.

Auteurs

Amer Ahmed (A)

Dipartimento di Scienze della Vita, Università di Siena, via A. Moro 2, 53100, Siena, Italy.

Alfonso Trezza (A)

Dipartimento di Biotecnologie, Chimica e Farmacia, Università di Siena, via A. Moro 2, 53100, Siena, Italy.

Mariangela Gentile (M)

Dipartimento di Scienze della Vita, Università di Siena, via A. Moro 2, 53100, Siena, Italy.

Eugenio Paccagnini (E)

Dipartimento di Scienze della Vita, Università di Siena, via A. Moro 2, 53100, Siena, Italy.

Alice Panti (A)

Dipartimento di Scienze della Vita, Università di Siena, via A. Moro 2, 53100, Siena, Italy.

Pietro Lupetti (P)

Dipartimento di Scienze della Vita, Università di Siena, via A. Moro 2, 53100, Siena, Italy.

Ottavia Spiga (O)

Dipartimento di Biotecnologie, Chimica e Farmacia, Università di Siena, via A. Moro 2, 53100, Siena, Italy.

Sergio Bova (S)

Department of Pharmaceutical and Pharmacological Sciences, University of Padova, Padova, Italy.

Fabio Fusi (F)

Dipartimento di Biotecnologie, Chimica e Farmacia, Università di Siena, via A. Moro 2, 53100, Siena, Italy. Electronic address: fabio.fusi@unisi.it.

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Classifications MeSH