Divergent Pharmacology and Biased Signaling of the Four Melanocortin-4 Receptor Isoforms in Rainbow Trout (
MC4R
allosteric ligand
biased signaling
constitutive activity
paralogs
rainbow trout
Journal
Biomolecules
ISSN: 2218-273X
Titre abrégé: Biomolecules
Pays: Switzerland
ID NLM: 101596414
Informations de publication
Date de publication:
16 08 2023
16 08 2023
Historique:
received:
03
07
2023
revised:
13
08
2023
accepted:
14
08
2023
medline:
28
8
2023
pubmed:
26
8
2023
entrez:
26
8
2023
Statut:
epublish
Résumé
The melanocortin-4 receptor (MC4R) is essential for the modulation of energy balance and reproduction in both fish and mammals. Rainbow trout (
Identifiants
pubmed: 37627313
pii: biom13081248
doi: 10.3390/biom13081248
pmc: PMC10452266
pii:
doi:
Substances chimiques
Receptor, Melanocortin, Type 4
0
Types de publication
Journal Article
Research Support, Non-U.S. Gov't
Langues
eng
Sous-ensembles de citation
IM
Références
Prog Mol Biol Transl Sci. 2022;189(1):215-257
pubmed: 35595350
Prog Mol Biol Transl Sci. 2009;88:173-204
pubmed: 20374728
Pharmacol Rev. 2019 Apr;71(2):267-315
pubmed: 30914442
Proc Natl Acad Sci U S A. 1969 Sep;64(1):367-73
pubmed: 4189501
J Mol Endocrinol. 2012 Oct 30;49(3):237-48
pubmed: 23014839
Gen Comp Endocrinol. 2016 May 1;230-231:143-52
pubmed: 27080551
Front Endocrinol (Lausanne). 2019 Oct 18;10:705
pubmed: 31681175
Biochim Biophys Acta. 2007 Oct;1772(10):1167-74
pubmed: 17964765
Proc Natl Acad Sci U S A. 2010 Nov 23;107(47):20164-71
pubmed: 20980662
Curr Biol. 2010 Oct 12;20(19):1729-34
pubmed: 20869245
Gen Comp Endocrinol. 2014 Dec 1;209:3-10
pubmed: 24768673
Gen Comp Endocrinol. 2009 Jan 15;160(2):134-8
pubmed: 19027741
Pharmacol Ther. 2008 Nov;120(2):129-48
pubmed: 18768149
Nat Rev Drug Discov. 2013 Mar;12(3):205-16
pubmed: 23411724
Mol Endocrinol. 1995 Jun;9(6):725-33
pubmed: 8592518
J Comp Physiol B. 2017 May;187(4):603-612
pubmed: 28197776
Nat Commun. 2014 Apr 22;5:3657
pubmed: 24755649
J Mol Endocrinol. 2012 Oct 30;49(3):221-35
pubmed: 23014838
Cell. 2005 Nov 4;123(3):493-505
pubmed: 16269339
Biochim Biophys Acta. 2016 Sep;1862(9):1485-94
pubmed: 27208795
Fish Physiol Biochem. 2023 Feb;49(1):61-74
pubmed: 36525144
Bioorg Med Chem Lett. 2007 Aug 15;17(16):4464-70
pubmed: 17574418
Gen Comp Endocrinol. 2019 Dec 1;284:113234
pubmed: 31398355
J Clin Endocrinol Metab. 2005 Oct;90(10):5632-8
pubmed: 16030156
Cell Metab. 2012 Feb 8;15(2):256-64
pubmed: 22245570
Peptides. 2006 Nov;27(11):2846-57
pubmed: 16806584
Adv Pharmacol. 2014;70:135-54
pubmed: 24931195
Eur J Biochem. 2004 Nov;271(21):4320-31
pubmed: 15511238
Comp Biochem Physiol B Biochem Mol Biol. 2002 Dec;133(4):609-46
pubmed: 12470823
Domest Anim Endocrinol. 2017 Apr;59:140-151
pubmed: 28152402
Endocr Connect. 2021 Nov 15;10(11):1489-1501
pubmed: 34678761
Annu Rev Pharmacol Toxicol. 2012;52:179-97
pubmed: 21942629
N Engl J Med. 2003 Mar 20;348(12):1085-95
pubmed: 12646665
Mol Cell Endocrinol. 2005 Jul 15;239(1-2):1-14
pubmed: 15975705
Mol Biol Evol. 2004 Mar;21(3):563-79
pubmed: 14694081
Pharmacol Ther. 2022 Jun;234:108044
pubmed: 34822948
Prog Mol Biol Transl Sci. 2013;114:147-91
pubmed: 23317785
Nat Rev Drug Discov. 2010 May;9(5):373-86
pubmed: 20431569
Gen Comp Endocrinol. 2008 Jan 15;155(2):280-7
pubmed: 17575981
Annu Rev Pharmacol Toxicol. 2007;47:53-87
pubmed: 17029567
Nature. 2016 Apr 18;533(7602):200-5
pubmed: 27088604
Cell. 1997 Jan 10;88(1):131-41
pubmed: 9019399
Mol Cell Endocrinol. 2020 Sep 15;515:110929
pubmed: 32615281
Gen Comp Endocrinol. 2006 Sep 1;148(2):150-62
pubmed: 16620815
Biochim Biophys Acta Mol Basis Dis. 2017 Oct;1863(10 Pt A):2486-2495
pubmed: 28433713
Mol Cell Biol. 1987 Aug;7(8):2745-52
pubmed: 3670292
Endocrinology. 2000 Sep;141(9):3514-7
pubmed: 10965926
Biomolecules. 2022 Feb 02;12(2):
pubmed: 35204745
Regul Pept. 2004 Aug 15;120(1-3):113-8
pubmed: 15177928
Nat Rev Drug Discov. 2018 Apr;17(4):243-260
pubmed: 29302067
Regul Pept. 2003 Sep 15;115(2):101-13
pubmed: 12972325
Endocr Rev. 2010 Aug;31(4):506-43
pubmed: 20190196
Front Neuroanat. 2020 Aug 21;14:48
pubmed: 32973463
Gen Comp Endocrinol. 2019 Jun 1;277:90-103
pubmed: 30905760
J Clin Invest. 2004 Oct;114(8):1158-64
pubmed: 15489963
Biomolecules. 2021 Mar 23;11(3):
pubmed: 33807040
Gene. 2020 May 30;741:144541
pubmed: 32165303
J Neurochem. 2002 Jul;82(1):6-18
pubmed: 12091460
Naunyn Schmiedebergs Arch Pharmacol. 2002 Nov;366(5):381-416
pubmed: 12382069
Gene. 2018 Dec 15;678:79-89
pubmed: 30075196
Endocrinology. 2003 Oct;144(10):4544-51
pubmed: 12959994
Mol Endocrinol. 2001 Jan;15(1):164-71
pubmed: 11145747
Endocrinology. 2005 Sep;146(9):3739-47
pubmed: 15961554
Brain Res. 2003 Oct 3;986(1-2):1-11
pubmed: 12965224
Endocrinology. 2003 Jun;144(6):2336-49
pubmed: 12746294
Biochem Pharmacol. 2008 Aug 15;76(4):520-30
pubmed: 18614155
J Biol Chem. 2002 Feb 8;277(6):3958-64
pubmed: 11723133
Gen Comp Endocrinol. 2006 Aug;148(1):85-94
pubmed: 16289182
Science. 2013 Jul 19;341(6143):278-81
pubmed: 23869017
Proc Natl Acad Sci U S A. 2015 Aug 4;112(31):9668-73
pubmed: 26170297
Nat Chem Biol. 2012 Aug;8(8):725-30
pubmed: 22729149
Front Endocrinol (Lausanne). 2020 Aug 14;11:538
pubmed: 32922362
Peptides. 2005 Oct;26(10):1952-64
pubmed: 15979204
Biochim Biophys Acta Mol Basis Dis. 2021 Jan 1;1867(1):165973
pubmed: 32949766
J Med Chem. 2004 Mar 25;47(7):1602-4
pubmed: 15027849
Methods Enzymol. 2010;484:267-79
pubmed: 21036237
Gen Comp Endocrinol. 2019 Oct 1;282:113219
pubmed: 31299224
Biochim Biophys Acta. 2013 Dec;1832(12):1939-48
pubmed: 23791567
Endocrinology. 2003 Oct;144(10):4552-61
pubmed: 12960082
J Pharmacol Exp Ther. 2003 Feb;304(2):818-26
pubmed: 12538838
Int J Biol Sci. 2014 Oct 09;10(10):1128-37
pubmed: 25332687