C(21)-Di- and monofluorinated scaffold for thevinol/orvinol-based opioid receptor ligands.

Receptors, Opioid Morphinans / chemistry Oxidation-Reduction Ligands Protein Binding Receptors, Opioid, mu

Journal

Organic & biomolecular chemistry
ISSN: 1477-0539
Titre abrégé: Org Biomol Chem
Pays: England
ID NLM: 101154995

Informations de publication

Date de publication:
22 11 2023
Historique:
medline: 27 11 2023
pubmed: 10 11 2023
entrez: 10 11 2023
Statut: epublish

Résumé

Defluorination of the readily available 21,21,21-trifluorothevinone (7) with Mg + Me

Identifiants

DOI: 10.1039/d3ob01577g PMID: 37947030
pubmed: 37947030
doi: 10.1039/d3ob01577g
doi:

Substances chimiques

Receptors, Opioid 0
Morphinans 0
Ligands 0
Receptors, Opioid, mu 0

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

9091-9100

Auteurs

Maria V Zelentsova (MV)

A.N.Nesmeyanov Institute of Organoelement Compounds, Russian Academy of Sciences, ul. Vavilova, 28, bld. 1, Moscow, 119334, Russia. skm@ineos.ac.ru.
ORCID: 0000-0002-6335-0855

Irina V Sandulenko (IV)

A.N.Nesmeyanov Institute of Organoelement Compounds, Russian Academy of Sciences, ul. Vavilova, 28, bld. 1, Moscow, 119334, Russia. skm@ineos.ac.ru.

Asmik A Ambartsumyan (AA)

A.N.Nesmeyanov Institute of Organoelement Compounds, Russian Academy of Sciences, ul. Vavilova, 28, bld. 1, Moscow, 119334, Russia. skm@ineos.ac.ru.
ORCID: 0000-0001-5492-9630

Anastasia A Danshina (AA)

A.N.Nesmeyanov Institute of Organoelement Compounds, Russian Academy of Sciences, ul. Vavilova, 28, bld. 1, Moscow, 119334, Russia. skm@ineos.ac.ru.
Moscow Institute of Physics and Technology (National Research University), Institutskiy per., 9, Dolgoprudny, Moscow Region, 141700, Russia.

Sergey K Moiseev (SK)

A.N.Nesmeyanov Institute of Organoelement Compounds, Russian Academy of Sciences, ul. Vavilova, 28, bld. 1, Moscow, 119334, Russia. skm@ineos.ac.ru.
ORCID: 0000-0002-9104-8725

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Classifications MeSH

questionsmedicales.fr › Acides aminés, peptides et protéines › Protéines › Protéines membranaires › Récepteurs de surface cellulaire › Récepteurs peptidiques › Récepteur aux neuropeptides › Récepteurs aux opioïdes › C(21)-Di- and monofluorinated scaffold for...
questionsmedicales.fr › Composés polycycliques › Hydrocarbures aromatiques polycycliques › Phénanthrènes › Morphinanes › C(21)-Di- and monofluorinated scaffold for...
questionsmedicales.fr › Métabolisme › Métabolisme énergétique › Oxydoréduction › C(21)-Di- and monofluorinated scaffold for...
questionsmedicales.fr › Actions chimiques et utilisations › Utilisations spécialisées de produits chimiques › Produits chimiques de laboratoire › Ligands › C(21)-Di- and monofluorinated scaffold for...
questionsmedicales.fr › Métabolisme › Liaison aux protéines › C(21)-Di- and monofluorinated scaffold for...
questionsmedicales.fr › Acides aminés, peptides et protéines › Protéines › Protéines membranaires › Récepteurs de surface cellulaire › Récepteurs peptidiques › Récepteur aux neuropeptides › Récepteurs aux opioïdes › Récepteur mu › C(21)-Di- and monofluorinated scaffold for...