Dimerization mechanism of an inverted-topology ion channel in membranes.

Fluc computational modeling dimerization ion channel single-molecule microscopy

Journal

Proceedings of the National Academy of Sciences of the United States of America
ISSN: 1091-6490
Titre abrégé: Proc Natl Acad Sci U S A
Pays: United States
ID NLM: 7505876

Informations de publication

Date de publication:
21 Nov 2023
Historique:
pmc-release: 13 05 2024
medline: 15 11 2023
pubmed: 13 11 2023
entrez: 13 11 2023
Statut: ppublish

Résumé

Many ion channels are multisubunit complexes where oligomerization is an obligatory requirement for function as the binding axis forms the charged permeation pathway. However, the mechanisms of in-membrane assembly of thermodynamically stable channels are largely unknown. Here, we demonstrate a key advance by reporting the dimerization equilibrium reaction of an inverted-topology, homodimeric fluoride channel Fluc in lipid bilayers. While the wild-type channel is a long-lived dimer, we leverage a known mutation, N43S, that weakens Na

Identifiants

pubmed: 37956279
doi: 10.1073/pnas.2308454120
pmc: PMC10666096
doi:

Substances chimiques

Lipid Bilayers 0
Fluorides Q80VPU408O
Ion Channels 0

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

e2308454120

Subventions

Organisme : NIGMS NIH HHS
ID : R35 GM128768
Pays : United States
Organisme : NIGMS NIH HHS
ID : R01 GM120260
Pays : United States

Commentaires et corrections

Type : UpdateOf

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Auteurs

Melanie Ernst (M)

Department of Biochemistry and Molecular Biophysics, Washington University School of Medicine, St. Louis, MO 63110.

Esam A Orabi (EA)

Theoretical Molecular Biophysics Section, National Heart, Lung, and Blood Institute, NIH, Bethesda, MD 20894.

Randy B Stockbridge (RB)

Department of Molecular, Cellular, and Developmental Biology, University of Michigan, Ann Arbor, MI 48109.

José D Faraldo-Gómez (JD)

Theoretical Molecular Biophysics Section, National Heart, Lung, and Blood Institute, NIH, Bethesda, MD 20894.

Janice L Robertson (JL)

Department of Biochemistry and Molecular Biophysics, Washington University School of Medicine, St. Louis, MO 63110.

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