Titre : Antienzymes

Antienzymes : Questions médicales fréquentes

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"D27.505.519.389.745.800.900" } } } ] }, { "@type": "MedicalWebPage", "name": "Inhibiteurs de protéines kinases", "alternateName": "Protein Kinase Inhibitors", "url": "https://questionsmedicales.fr/mesh/D047428", "about": { "@type": "MedicalCondition", "name": "Inhibiteurs de protéines kinases", "code": { "@type": "MedicalCode", "code": "D047428", "codingSystem": "MeSH" }, "identifier": { "@type": "PropertyValue", "propertyID": "MeSH Tree", "value": "D27.505.519.389.755" } }, "hasPart": [ { "@type": "MedicalWebPage", "name": "Inhibiteurs des Janus kinases", "alternateName": "Janus Kinase Inhibitors", "url": "https://questionsmedicales.fr/mesh/D000075242", "about": { "@type": "MedicalCondition", "name": "Inhibiteurs des Janus kinases", "code": { "@type": "MedicalCode", "code": "D000075242", "codingSystem": "MeSH" }, "identifier": { "@type": "PropertyValue", "propertyID": "MeSH Tree", "value": "D27.505.519.389.755.500" } } }, { "@type": "MedicalWebPage", "name": "Inhibiteurs de protéine-tyrosine kinase", "alternateName": "Tyrosine Protein Kinase Inhibitors", "url": "https://questionsmedicales.fr/mesh/D000092004", "about": { "@type": "MedicalCondition", "name": "Inhibiteurs de protéine-tyrosine kinase", "code": { "@type": "MedicalCode", "code": "D000092004", "codingSystem": "MeSH" }, "identifier": { "@type": "PropertyValue", "propertyID": "MeSH Tree", "value": "D27.505.519.389.755.875" } } } ] }, { "@type": "MedicalWebPage", "name": "Inhibiteurs de la synthèse protéique", "alternateName": "Protein Synthesis Inhibitors", "url": "https://questionsmedicales.fr/mesh/D011500", "about": { "@type": "MedicalCondition", "name": "Inhibiteurs de la synthèse protéique", "code": { "@type": "MedicalCode", "code": "D011500", "codingSystem": "MeSH" }, "identifier": { "@type": "PropertyValue", "propertyID": "MeSH Tree", "value": "D27.505.519.389.760" } } }, { "@type": "MedicalWebPage", "name": "Inhibiteurs de la pompe à protons", "alternateName": "Proton Pump Inhibitors", 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"https://questionsmedicales.fr/author/Xiaoxi%20Liu", "affiliation": { "@type": "Organization", "name": "Department of Cancer Biology and the Linde Program in Cancer Chemical Biology, Dana-Farber Cancer Institute, Boston, MA, USA." } }, { "@type": "Person", "name": "Robert S Magin", "url": "https://questionsmedicales.fr/author/Robert%20S%20Magin", "affiliation": { "@type": "Organization", "name": "Department of Cancer Biology and the Linde Program in Cancer Chemical Biology, Dana-Farber Cancer Institute, Boston, MA, USA." } }, { "@type": "Person", "name": "Nathan J Schauer", "url": "https://questionsmedicales.fr/author/Nathan%20J%20Schauer", "affiliation": { "@type": "Organization", "name": "Department of Cancer Biology and the Linde Program in Cancer Chemical Biology, Dana-Farber Cancer Institute, Boston, MA, USA." } }, { "@type": "Person", "name": "Sara J Buhrlage", "url": "https://questionsmedicales.fr/author/Sara%20J%20Buhrlage", "affiliation": { "@type": "Organization", "name": "Department of Cancer Biology and the Linde Program in Cancer Chemical Biology, Dana-Farber Cancer Institute, Boston, MA, USA. saraj_buhrlage@dfci.harvard.edu." } }, { "@type": "Person", "name": "R Gentry Wilkerson", "url": "https://questionsmedicales.fr/author/R%20Gentry%20Wilkerson", "affiliation": { "@type": "Organization", "name": "Department of Emergency Medicine, University of Maryland School of Medicine, 110 South Paca Street, 6th Floor, Suite 200, Baltimore, MD 21201, USA. Electronic address: gwilkerson@som.umaryland.edu." } } ], "citation": [ { "@type": "ScholarlyArticle", "name": "Recent development of multi-targeted inhibitors of human topoisomerase II enzyme as potent cancer therapeutics.", "datePublished": "2022-12-07", "url": "https://questionsmedicales.fr/article/36495993", "identifier": { "@type": "PropertyValue", "propertyID": "DOI", "value": "10.1016/j.ijbiomac.2022.12.013" } }, { "@type": "ScholarlyArticle", "name": "Steady-state kinetic analysis of reversible enzyme inhibitors: A case study on calf intestine alkaline phosphatase.", "datePublished": "2023-07-26", "url": "https://questionsmedicales.fr/article/37858536", "identifier": { "@type": "PropertyValue", "propertyID": "DOI", "value": "10.1016/bs.mie.2023.06.015" } }, { "@type": "ScholarlyArticle", "name": "Specific glycine-dependent enzyme motion determines the potency of conformation selective inhibitors of threonyl-tRNA synthetase.", "datePublished": "2024-07-16", "url": 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"MedicalWebPage", "name": "Diagnostic", "headline": "Diagnostic sur Antienzymes", "description": "Comment diagnostiquer une inhibition enzymatique ?\nQuels symptômes indiquent une inhibition enzymatique ?\nQuels tests sont utilisés pour détecter les antienzymes ?\nPeut-on utiliser l'imagerie pour diagnostiquer ?\nQuels marqueurs biochimiques sont associés aux antienzymes ?", "url": "https://questionsmedicales.fr/mesh/D004791?page=3#section-diagnostic" }, { "@type": "MedicalWebPage", "name": "Symptômes", "headline": "Symptômes sur Antienzymes", "description": "Quels sont les symptômes d'une inhibition enzymatique ?\nL'inhibition enzymatique peut-elle causer des douleurs ?\nY a-t-il des symptômes spécifiques selon l'enzyme inhibée ?\nLes symptômes sont-ils toujours présents ?\nComment les symptômes évoluent-ils avec le temps ?", "url": "https://questionsmedicales.fr/mesh/D004791?page=3#section-symptômes" }, { "@type": "MedicalWebPage", "name": "Prévention", "headline": "Prévention sur Antienzymes", "description": "Comment prévenir l'inhibition enzymatique ?\nLes vaccinations peuvent-elles prévenir des inhibitions enzymatiques ?\nY a-t-il des habitudes de vie à adopter ?\nLes contrôles médicaux réguliers sont-ils importants ?\nL'éducation sur les médicaments est-elle nécessaire ?", "url": "https://questionsmedicales.fr/mesh/D004791?page=3#section-prévention" }, { "@type": "MedicalWebPage", "name": "Traitements", "headline": "Traitements sur Antienzymes", "description": "Quels traitements existent pour l'inhibition enzymatique ?\nLes antienzymes sont-ils utilisés en chimiothérapie ?\nComment les inhibiteurs enzymatiques sont-ils administrés ?\nY a-t-il des effets secondaires aux antienzymes ?\nLes traitements sont-ils personnalisés ?", "url": "https://questionsmedicales.fr/mesh/D004791?page=3#section-traitements" }, { "@type": "MedicalWebPage", "name": "Complications", "headline": "Complications sur Antienzymes", "description": "Quelles complications peuvent survenir avec l'inhibition enzymatique ?\nL'inhibition enzymatique peut-elle entraîner des maladies chroniques ?\nY a-t-il des risques de surdosage avec les antienzymes ?\nComment gérer les complications liées aux antienzymes ?\nLes complications sont-elles réversibles ?", "url": "https://questionsmedicales.fr/mesh/D004791?page=3#section-complications" }, { "@type": "MedicalWebPage", "name": "Facteurs de risque", "headline": "Facteurs de risque sur Antienzymes", "description": "Quels sont les facteurs de risque d'inhibition enzymatique ?\nL'âge influence-t-il le risque d'inhibition enzymatique ?\nLes maladies auto-immunes sont-elles un facteur de risque ?\nLe mode de vie affecte-t-il le risque ?\nLes médicaments peuvent-ils être des facteurs de risque ?", "url": "https://questionsmedicales.fr/mesh/D004791?page=3#section-facteurs de risque" } ] }, { "@type": "FAQPage", "mainEntity": [ { "@type": "Question", "name": "Comment diagnostiquer une inhibition enzymatique ?", "position": 1, "acceptedAnswer": { "@type": "Answer", "text": "Des tests sanguins et des analyses biochimiques évaluent l'activité enzymatique." } }, { "@type": "Question", "name": "Quels symptômes indiquent une inhibition enzymatique ?", "position": 2, "acceptedAnswer": { "@type": "Answer", "text": "Des symptômes comme la fatigue, la douleur abdominale ou des troubles digestifs peuvent apparaître." } }, { "@type": "Question", "name": "Quels tests sont utilisés pour détecter les antienzymes ?", "position": 3, "acceptedAnswer": { "@type": "Answer", "text": "Les tests d'activité enzymatique et les dosages spécifiques d'anticorps sont courants." } }, { "@type": "Question", "name": "Peut-on utiliser l'imagerie pour diagnostiquer ?", "position": 4, "acceptedAnswer": { "@type": "Answer", "text": "L'imagerie peut aider à évaluer les organes affectés, mais n'est pas spécifique aux antienzymes." } }, { "@type": "Question", "name": "Quels marqueurs biochimiques sont associés aux antienzymes ?", "position": 5, "acceptedAnswer": { "@type": "Answer", "text": "Les niveaux d'enzymes spécifiques dans le sang peuvent indiquer une inhibition enzymatique." } }, { "@type": "Question", "name": "Quels sont les symptômes d'une inhibition enzymatique ?", "position": 6, "acceptedAnswer": { "@type": "Answer", "text": "Les symptômes incluent douleurs abdominales, nausées, et troubles métaboliques." } }, { "@type": "Question", "name": "L'inhibition enzymatique peut-elle causer des douleurs ?", "position": 7, "acceptedAnswer": { "@type": "Answer", "text": "Oui, elle peut entraîner des douleurs dues à des troubles digestifs ou métaboliques." } }, { "@type": "Question", "name": "Y a-t-il des symptômes spécifiques selon l'enzyme inhibée ?", "position": 8, "acceptedAnswer": { "@type": "Answer", "text": "Oui, les symptômes varient selon l'enzyme affectée, comme la lactase ou la lipase." } }, { "@type": "Question", "name": "Les symptômes sont-ils toujours présents ?", "position": 9, "acceptedAnswer": { "@type": "Answer", "text": "Non, certains patients peuvent être asymptomatiques malgré une inhibition enzymatique." } }, { "@type": "Question", "name": "Comment les symptômes évoluent-ils avec le temps ?", "position": 10, "acceptedAnswer": { "@type": "Answer", "text": "Les symptômes peuvent s'aggraver si l'inhibition persiste sans traitement approprié." } }, { "@type": "Question", "name": "Comment prévenir l'inhibition enzymatique ?", "position": 11, "acceptedAnswer": { "@type": "Answer", "text": "Une alimentation équilibrée et l'évitement de substances toxiques peuvent aider." } }, { "@type": "Question", "name": "Les vaccinations peuvent-elles prévenir des inhibitions enzymatiques ?", "position": 12, "acceptedAnswer": { "@type": "Answer", "text": "Certaines vaccinations peuvent prévenir des infections qui causent des inhibitions enzymatiques." } }, { "@type": "Question", "name": "Y a-t-il des habitudes de vie à adopter ?", "position": 13, "acceptedAnswer": { "@type": "Answer", "text": "Oui, éviter l'alcool et le tabac peut réduire le risque d'inhibition enzymatique." } }, { "@type": "Question", "name": "Les contrôles médicaux réguliers sont-ils importants ?", "position": 14, "acceptedAnswer": { "@type": "Answer", "text": "Oui, des contrôles réguliers permettent de détecter précocement des problèmes enzymatiques." } }, { "@type": "Question", "name": "L'éducation sur les médicaments est-elle nécessaire ?", "position": 15, "acceptedAnswer": { "@type": "Answer", "text": "Oui, comprendre les effets des médicaments aide à prévenir les inhibitions enzymatiques." } }, { "@type": "Question", "name": "Quels traitements existent pour l'inhibition enzymatique ?", "position": 16, "acceptedAnswer": { "@type": "Answer", "text": "Les traitements incluent des médicaments spécifiques et des modifications diététiques." } }, { "@type": "Question", "name": "Les antienzymes sont-ils utilisés en chimiothérapie ?", "position": 17, "acceptedAnswer": { "@type": "Answer", "text": "Oui, certains antienzymes sont utilisés pour cibler des enzymes dans les cellules cancéreuses." } }, { "@type": "Question", "name": "Comment les inhibiteurs enzymatiques sont-ils administrés ?", "position": 18, "acceptedAnswer": { "@type": "Answer", "text": "Ils peuvent être administrés par voie orale, intraveineuse ou topique selon le cas." } }, { "@type": "Question", "name": "Y a-t-il des effets secondaires aux antienzymes ?", "position": 19, "acceptedAnswer": { "@type": "Answer", "text": "Oui, des effets secondaires comme des nausées, des éruptions cutanées ou des douleurs peuvent survenir." } }, { "@type": "Question", "name": "Les traitements sont-ils personnalisés ?", "position": 20, "acceptedAnswer": { "@type": "Answer", "text": "Oui, le traitement est souvent adapté en fonction de la cause et de la gravité de l'inhibition." } }, { "@type": "Question", "name": "Quelles complications peuvent survenir avec l'inhibition enzymatique ?", "position": 21, "acceptedAnswer": { "@type": "Answer", "text": "Des complications comme des troubles métaboliques ou des maladies organiques peuvent survenir." } }, { "@type": "Question", "name": "L'inhibition enzymatique peut-elle entraîner des maladies chroniques ?", "position": 22, "acceptedAnswer": { "@type": "Answer", "text": "Oui, une inhibition prolongée peut contribuer à des maladies chroniques comme le diabète." } }, { "@type": "Question", "name": "Y a-t-il des risques de surdosage avec les antienzymes ?", "position": 23, "acceptedAnswer": { "@type": "Answer", "text": "Oui, un surdosage peut entraîner des effets indésirables graves et des complications." } }, { "@type": "Question", "name": "Comment gérer les complications liées aux antienzymes ?", "position": 24, "acceptedAnswer": { "@type": "Answer", "text": "La gestion implique un suivi médical régulier et des ajustements de traitement." } }, { "@type": "Question", "name": "Les complications sont-elles réversibles ?", "position": 25, "acceptedAnswer": { "@type": "Answer", "text": "Certaines complications peuvent être réversibles avec un traitement approprié et rapide." } }, { "@type": "Question", "name": "Quels sont les facteurs de risque d'inhibition enzymatique ?", "position": 26, "acceptedAnswer": { "@type": "Answer", "text": "Les facteurs incluent des antécédents familiaux, des maladies héréditaires et des habitudes alimentaires." } }, { "@type": "Question", "name": "L'âge influence-t-il le risque d'inhibition enzymatique ?", "position": 27, "acceptedAnswer": { "@type": "Answer", "text": "Oui, le risque augmente souvent avec l'âge en raison de la dégradation enzymatique naturelle." } }, { "@type": "Question", "name": "Les maladies auto-immunes sont-elles un facteur de risque ?", "position": 28, "acceptedAnswer": { "@type": "Answer", "text": "Oui, certaines maladies auto-immunes peuvent augmenter le risque d'inhibition enzymatique." } }, { "@type": "Question", "name": "Le mode de vie affecte-t-il le risque ?", "position": 29, "acceptedAnswer": { "@type": "Answer", "text": "Oui, un mode de vie sédentaire et une mauvaise alimentation augmentent le risque." } }, { "@type": "Question", "name": "Les médicaments peuvent-ils être des facteurs de risque ?", "position": 30, "acceptedAnswer": { "@type": "Answer", "text": "Oui, certains médicaments peuvent interférer avec l'activité enzymatique et augmenter le risque." } } ] } ] }

Sous-catégories

48 au total
└─

Inhibiteurs des protéines activatrices de la 5-lipoxygénase

5-Lipoxygenase-Activating Protein Inhibitors D058946 - D27.505.519.389.086
└─

Inhibiteurs de l'acétaldéhyde déshydrogénase

Acetaldehyde Dehydrogenase Inhibitors D065086 - D27.505.519.389.089
└─

Inhibiteurs de l'adénosine désaminase

Adenosine Deaminase Inhibitors D058892 - D27.505.519.389.092
└─

Inhibiteurs des adénylate cyclases

Adenylyl Cyclase Inhibitors D000067956 - D27.505.519.389.108
└─

Inhibiteurs de la calcineurine

Calcineurin Inhibitors D065095 - D27.505.519.389.174
└─

Inhibiteurs de l'anhydrase carbonique

Carbonic Anhydrase Inhibitors D002257 - D27.505.519.389.200
└─

Inhibiteurs et modulateurs de la gamma-secrétase

Gamma Secretase Inhibitors and Modulators D000091062 - D27.505.519.389.315
└─

Inhibiteurs des enzymes du cytochrome P-450

Cytochrome P-450 Enzyme Inhibitors D065607 - D27.505.519.389.335
└─

Antifoliques

Folic Acid Antagonists D005493 - D27.505.519.389.350
└─

Inhibiteurs de désacétylase d'histone

Histone Deacetylase Inhibitors D056572 - D27.505.519.389.360
└─

Inhibiteurs de l'intégrase

Integrase Inhibitors D019429 - D27.505.519.389.375
└─

Inhibiteurs de la lipoxygénase

Lipoxygenase Inhibitors D016859 - D27.505.519.389.480
└─

Inhibiteurs de la monoamine oxydase

Monoamine Oxidase Inhibitors D008996 - D27.505.519.389.616
└─

Inhibiteurs de la synthèse d'acide nucléique

Nucleic Acid Synthesis Inhibitors D019384 - D27.505.519.389.675
└─

Inhibiteurs de l'ornithine décarboxylase

Ornithine Decarboxylase Inhibitors D065108 - D27.505.519.389.705
└─

Inhibiteurs de la phosphodiestérase

Phosphodiesterase Inhibitors D010726 - D27.505.519.389.735
└─

Inhibiteurs des phosphoinositide-3 kinases

Phosphoinositide-3 Kinase Inhibitors D000081082 - D27.505.519.389.736
└─

Inhibiteurs de la phospholipase A2

Phospholipase A2 Inhibitors D064801 - D27.505.519.389.737
└─

Inhibiteurs de prolyle hydroxylases

Prolyl-Hydroxylase Inhibitors D064800 - D27.505.519.389.740
└─

Inhibiteurs de protéases

Protease Inhibitors D011480 - D27.505.519.389.745
└─

Inhibiteurs de protéines kinases

Protein Kinase Inhibitors D047428 - D27.505.519.389.755
└─

Inhibiteurs de la synthèse protéique

Protein Synthesis Inhibitors D011500 - D27.505.519.389.760
└─

Inhibiteurs de la pompe à protons

Proton Pump Inhibitors D054328 - D27.505.519.389.848
└─

Agents découplants

Uncoupling Agents D014475 - D27.505.519.389.936
└─└─

Inhibiteurs du cytochrome P-450 CYP1A2

Cytochrome P-450 CYP1A2 Inhibitors D065609 - D27.505.519.389.335.120
└─└─

Inhibiteurs du cytochrome P-450 CYP2B6

Cytochrome P-450 CYP2B6 Inhibitors D065686 - D27.505.519.389.335.260
└─└─

Inhibiteurs du cytochrome P-450 CYP2C8

Cytochrome P-450 CYP2C8 Inhibitors D065687 - D27.505.519.389.335.308
└─└─

Inhibiteurs du cytochrome P-450 CYP2C19

Cytochrome P-450 CYP2C19 Inhibitors D065689 - D27.505.519.389.335.319
└─└─

Inhibiteurs du cytochrome P-450 CYP2C9

Cytochrome P-450 CYP2C9 Inhibitors D065688 - D27.505.519.389.335.329
└─└─

Inhibiteurs du cytochrome P-450 CYP2D6

Cytochrome P-450 CYP2D6 Inhibitors D065690 - D27.505.519.389.335.368
└─└─

Inhibiteurs du cytochrome P-450 CYP2E1

Cytochrome P-450 CYP2E1 Inhibitors D065691 - D27.505.519.389.335.421
└─└─

Inhibiteurs du cytochrome P-450 CYP3A

Cytochrome P-450 CYP3A Inhibitors D065692 - D27.505.519.389.335.503
└─└─

Inhibiteurs de la phosphodiestérase-3

Phosphodiesterase 3 Inhibitors D058987 - D27.505.519.389.735.249
└─└─

Inhibiteurs de la phosphodiestérase-4

Phosphodiesterase 4 Inhibitors D058988 - D27.505.519.389.735.374
└─└─

Inhibiteurs de la phosphodiestérase-5

Phosphodiesterase 5 Inhibitors D058986 - D27.505.519.389.735.500
└─└─

Inhibiteurs de l'enzyme de conversion de l'angiotensine

Angiotensin-Converting Enzyme Inhibitors D000806 - D27.505.519.389.745.085
└─└─

Inhibiteurs de la cystéine protéinase

Cysteine Proteinase Inhibitors D015853 - D27.505.519.389.745.325
└─└─

Inhibiteurs de métalloprotéinases matricielles

Matrix Metalloproteinase Inhibitors D061965 - D27.505.519.389.745.610
└─└─

Inhibiteurs du protéasome

Proteasome Inhibitors D061988 - D27.505.519.389.745.705
└─└─

Inhibiteurs de la rénine

Renin Inhibitors D000092502 - D27.505.519.389.745.753
└─└─

Inhibiteurs de la sérine protéinase

Serine Proteinase Inhibitors D015842 - D27.505.519.389.745.800
└─└─

Inhibiteurs des Janus kinases

Janus Kinase Inhibitors D000075242 - D27.505.519.389.755.500
└─└─

Inhibiteurs de protéine-tyrosine kinase

Tyrosine Protein Kinase Inhibitors D000092004 - D27.505.519.389.755.875
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Inhibiteurs des vasopeptidases

Vasopeptidase Inhibitors D000075563 - D27.505.519.389.745.085.500
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Inhibiteurs des caspases

Caspase Inhibitors D061945 - D27.505.519.389.745.325.500
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Inhibiteurs de serine peptidase de type Kazal

Serine Peptidase Inhibitors, Kazal Type D000074162 - D27.505.519.389.745.800.562
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Serpines

Serpins D015843 - D27.505.519.389.745.800.675
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Inhibiteurs trypsiques

Trypsin Inhibitors D014361 - D27.505.519.389.745.800.900

Sources (10000 au total)

Synthesis, crystal structure, spectroscopic and computational investigations of the newly synthesized Schiff bases scaffold as enzyme inhibitor.

The current project was planned to access the enzyme inhibition potential of the synthesize imines; (E)-2-(2-hydroxy-4,5-dimethoxybenzylideneamino)benzonitrile 1 and (E)-2-(((3-hydroxy-4-methylphenyl)...

Development of human lactate dehydrogenase a inhibitors: high-throughput screening, molecular dynamics simulation and enzyme activity assay.

Lactate dehydrogenase A (LDHA) is highly expressed in many tumor cells and promotes the conversion of pyruvate to lactic acid in the glucose pathway, providing energy and synthetic precursors for rapi...

The screening of lipase inhibitors based on the metal-organic framework Zeolitic Imidazolate Framework-8-immobilized enzyme microreactor.

An online capillary electrophoresis method based-lipase immobilized enzyme microreactor was developed for lipase kinetic study and inhibitor screening from compounds from natural products. Zeolitic Im...

Chemical similarities and differences among inhibitors of nitric oxide synthase, arginase and dimethylarginine dimethylaminohydrolase-1: Implications for the design of novel enzyme inhibitors modulating the nitric oxide pathway.

Nitric oxide (NO) is a signalling molecule that controls a multitude of regulatory functions including neurotransmission, vascular tone, immune response, and angiogenesis. Regulating NO concentrations...