Tricyclic Imidazolidin-4-ones by Witkop Oxidation of Tetrahydro-β-carbolines.


Journal

The Journal of organic chemistry
ISSN: 1520-6904
Titre abrégé: J Org Chem
Pays: United States
ID NLM: 2985193R

Informations de publication

Date de publication:
21 02 2020
Historique:
pubmed: 7 1 2020
medline: 24 6 2021
entrez: 7 1 2020
Statut: ppublish

Résumé

1-Substituted and 1,1-disubstituted tetrahydro-β-carbolines undergo sodium periodate oxidative ring expansion in the presence of formaldehyde and other aldehydes to form 5,6-dihydro-7

Identifiants

pubmed: 31904963
doi: 10.1021/acs.joc.9b03402
pmc: PMC7092372
mid: NIHMS1565307
doi:

Substances chimiques

Aldehydes 0
Carbolines 0
tryptoline 65027TMI0H

Types de publication

Journal Article Research Support, N.I.H., Extramural

Langues

eng

Sous-ensembles de citation

IM

Pagination

2846-2853

Subventions

Organisme : NIAID NIH HHS
ID : R01 AI116723
Pays : United States

Références

Org Lett. 2004 Aug 5;6(16):2641-4
pubmed: 15281733
Org Lett. 2018 Apr 20;20(8):2333-2337
pubmed: 29582653
Org Lett. 2019 Mar 15;21(6):1559-1563
pubmed: 30844292
Bioorg Med Chem. 2003 Nov 17;11(23):5149-53
pubmed: 14604678
Chemistry. 2017 Jul 3;23(37):8780-8799
pubmed: 28295709
Nat Chem Biol. 2013 Jan;9(1):21-9
pubmed: 23160003
Eur J Med Chem. 2001 Mar;36(3):265-86
pubmed: 11337105
J Med Chem. 2016 Jul 14;59(13):6121-35
pubmed: 27280693

Auteurs

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Classifications MeSH