An Anti-CD22-


Journal

Molecular cancer therapeutics
ISSN: 1538-8514
Titre abrégé: Mol Cancer Ther
Pays: United States
ID NLM: 101132535

Informations de publication

Date de publication:
02 2021
Historique:
received: 21 01 2020
revised: 07 07 2020
accepted: 09 11 2020
pubmed: 5 12 2020
medline: 21 10 2021
entrez: 4 12 2020
Statut: ppublish

Résumé

We are interested in developing a second generation of antibody-drug conjugates (ADCs) for the treatment of non-Hodgkin lymphoma (NHL) that could provide a longer duration of response and be more effective in indolent NHL than the microtubule-inhibiting ADCs pinatuzumab vedotin [anti-CD22-vc-monomethyl auristatin E (MMAE)] and polatuzumab vedotin (anti-CD79b-vc-MMAE). Pinatuzumab vedotin (anti-CD22-vc-MMAE) and polatuzumab vedotin (anti-CD79b-vc-MMAE) are ADCs that contain the microtubule inhibitor MMAE. Clinical trial data suggest that these ADCs have promising efficacy for the treatment of NHL; however, some patients do not respond or become resistant to the ADCs. We tested an anti-CD22 ADC with a

Identifiants

pubmed: 33273056
pii: 1535-7163.MCT-20-0046
doi: 10.1158/1535-7163.MCT-20-0046
doi:

Substances chimiques

Aminobenzoates 0
CD22 protein, human 0
Immunoconjugates 0
Oligopeptides 0
Sialic Acid Binding Ig-like Lectin 2 0
auristatin 0

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

340-346

Informations de copyright

©2020 American Association for Cancer Research.

Références

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Chen R, Hou J, Newman E, Kim Y, Donohue C, Liu X, et al. CD30 downregulation, MMAE resistance, and MDR1 upregulation are all associated with resistance to Brentuximab Vedotin. Mol Cancer Ther. 2015;14:1376–84.
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Giddens AC, Lee HH, Lu G-L, Miller CK, Guo J, Lewis Phillips GD, et al. Analogues of DNA minor groove cross-linking agents incorporating aminoCBI, an amino derivative of the duocarmycins: synthesis, cytotoxicity, and potential as payloads for antibody-drug conjugates. Bioorg Med Chem. 2016;24:6075–81.
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Auteurs

Shang-Fan Yu (SF)

Research and Early Development, Genentech Inc., South San Francisco, California.

Donna W Lee (DW)

Research and Early Development, Genentech Inc., South San Francisco, California.

Bing Zheng (B)

Research and Early Development, Genentech Inc., South San Francisco, California.

Geoffrey Del Rosario (G)

Research and Early Development, Genentech Inc., South San Francisco, California.

Douglas Leipold (D)

Research and Early Development, Genentech Inc., South San Francisco, California.

Helen Booler (H)

Research and Early Development, Genentech Inc., South San Francisco, California.

Fiona Zhong (F)

Research and Early Development, Genentech Inc., South San Francisco, California.

Montserrat Carrasco-Triguero (M)

Research and Early Development, Genentech Inc., South San Francisco, California.

Kyu Hong (K)

Research and Early Development, Genentech Inc., South San Francisco, California.

Peter Yan (P)

Research and Early Development, Genentech Inc., South San Francisco, California.

Rebecca K Rowntree (RK)

Research and Early Development, Genentech Inc., South San Francisco, California.

Melissa M Schutten (MM)

Research and Early Development, Genentech Inc., South San Francisco, California.

Thomas Pillow (T)

Research and Early Development, Genentech Inc., South San Francisco, California.

Jack D Sadowsky (JD)

Research and Early Development, Genentech Inc., South San Francisco, California.

Peter S Dragovich (PS)

Research and Early Development, Genentech Inc., South San Francisco, California.

Andrew G Polson (AG)

Research and Early Development, Genentech Inc., South San Francisco, California. polson@gene.com.

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Classifications MeSH