Design and In Vitro Evaluation of Splice-Switching Oligonucleotides Bearing Locked Nucleic Acids, Amido-Bridged Nucleic Acids, and Guanidine-Bridged Nucleic Acids.

amido-bridged nucleic acids (AmNAs) bridged nucleic acids (BNAs) chemical modification dystrophin exon skipping guanidine-bridged nucleic acids (GuNAs) locked nucleic acids (LNAs) splice-switching oligonucleotide

Journal

International journal of molecular sciences
ISSN: 1422-0067
Titre abrégé: Int J Mol Sci
Pays: Switzerland
ID NLM: 101092791

Informations de publication

Date de publication:
29 Mar 2021
Historique:
received: 15 02 2021
revised: 20 03 2021
accepted: 26 03 2021
entrez: 3 4 2021
pubmed: 4 4 2021
medline: 2 6 2021
Statut: epublish

Résumé

Our group previously developed a series of bridged nucleic acids (BNAs), including locked nucleic acids (LNAs), amido-bridged nucleic acids (AmNAs), and guanidine-bridged nucleic acids (GuNAs), to impart specific characteristics to oligonucleotides such as high-affinity binding and enhanced enzymatic resistance. In this study, we designed a series of LNA-, AmNA-, and GuNA-modified splice-switching oligonucleotides (SSOs) with different lengths and content modifications. We measured the melting temperature (

Identifiants

pubmed: 33805378
pii: ijms22073526
doi: 10.3390/ijms22073526
pmc: PMC8037388
pii:
doi:

Substances chimiques

DMD protein, human 0
Dystrophin 0
Nucleic Acids 0
Oligonucleotides 0
locked nucleic acid 0
Guanidine JU58VJ6Y3B

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Subventions

Organisme : Japan Society for the Promotion of Science
ID : 15J05689
Organisme : Japan Agency for Medical Research and Development
ID : JP20am0101084
Organisme : Japan Agency for Medical Research and Development
ID : JP18am0301004
Organisme : Japan Agency for Medical Research and Development
ID : JP20am0401003

Références

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Auteurs

Takenori Shimo (T)

Graduate School of Pharmaceutical Sciences, Osaka University, 1-6 Yamadaoka, Suita, Osaka 565-0871, Japan.

Yusuke Nakatsuji (Y)

Graduate School of Pharmaceutical Sciences, Osaka University, 1-6 Yamadaoka, Suita, Osaka 565-0871, Japan.

Keisuke Tachibana (K)

Graduate School of Pharmaceutical Sciences, Osaka University, 1-6 Yamadaoka, Suita, Osaka 565-0871, Japan.

Satoshi Obika (S)

Graduate School of Pharmaceutical Sciences, Osaka University, 1-6 Yamadaoka, Suita, Osaka 565-0871, Japan.

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Classifications MeSH