Multi-material 3D printing of programmable and stretchable oromucosal patches for delivery of saquinavir.

3D printing Buccal delivery Direct ink writing Microenvironmental pH Oromucosal patch Saquinavir

Journal

International journal of pharmaceutics
ISSN: 1873-3476
Titre abrégé: Int J Pharm
Pays: Netherlands
ID NLM: 7804127

Informations de publication

Date de publication:
15 Dec 2021
Historique:
received: 21 09 2021
revised: 19 10 2021
accepted: 23 10 2021
pubmed: 9 11 2021
medline: 15 12 2021
entrez: 8 11 2021
Statut: ppublish

Résumé

Oromucosal patches for drug delivery allow fast onset of action and ability to circumvent hepatic first pass metabolism of drugs. While conventional fabrication methods such as solvent casting or hot melt extrusion are ideal for scalable production of low-cost delivery patches, these methods chiefly allow for simple, homogenous patch designs. As alternative, a multi-material direct-ink-write 3D printing for rapid fabrication of complex oromucosal patches with unique design features was demonstrated in the present study. Specifically, three print-materials: an acidic saquinavir-loaded hydroxypropyl methylcellulose ink, an alkaline effervescent sodium carbonate-loaded ink, and a methyl cellulose backing material were combined in various designs. The CO

Identifiants

pubmed: 34748810
pii: S0378-5173(21)01042-5
doi: 10.1016/j.ijpharm.2021.121236
pii:
doi:

Substances chimiques

Hypromellose Derivatives 3NXW29V3WO
Saquinavir L3JE09KZ2F

Types de publication

Journal Article

Langues

eng

Sous-ensembles de citation

IM

Pagination

121236

Informations de copyright

Copyright © 2021 The Author(s). Published by Elsevier B.V. All rights reserved.

Auteurs

Shaolong He (S)

Department of Pharmacy, Faculty of Health and Medical Sciences, University of Copenhagen, Universitetsparken 2, DK-2100 Copenhagen, Denmark.

Carmen Radeke (C)

Department of Health Technology, Technical University of Denmark, Building 423, 2800 Kgs. Lyngby, Denmark.

Jette Jacobsen (J)

Department of Pharmacy, Faculty of Health and Medical Sciences, University of Copenhagen, Universitetsparken 2, DK-2100 Copenhagen, Denmark.

Johan Ulrik Lind (JU)

Department of Health Technology, Technical University of Denmark, Building 423, 2800 Kgs. Lyngby, Denmark. Electronic address: joli@dtu.dk.

Huiling Mu (H)

Department of Pharmacy, Faculty of Health and Medical Sciences, University of Copenhagen, Universitetsparken 2, DK-2100 Copenhagen, Denmark. Electronic address: huiling.mu@sund.ku.dk.

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Classifications MeSH