Aiming to improve binding of porphyrin diphenyl guanidinium conjugates to guanine-quadruplexes: When size matters.


Journal

Bioorganic & medicinal chemistry letters
ISSN: 1464-3405
Titre abrégé: Bioorg Med Chem Lett
Pays: England
ID NLM: 9107377

Informations de publication

Date de publication:
01 11 2022
Historique:
received: 31 05 2022
revised: 12 08 2022
accepted: 22 08 2022
pubmed: 29 8 2022
medline: 4 10 2022
entrez: 28 8 2022
Statut: ppublish

Résumé

Aiming to improve the binding to Guanine quadruplexes of different topologies, docking studies of porphyrin diphenyl guanidine conjugates previously prepared with an O or a S bridge between the diphenyl moiety and a newly design derivative with an SO

Identifiants

pubmed: 36031019
pii: S0960-894X(22)00430-9
doi: 10.1016/j.bmcl.2022.128954
pii:
doi:

Substances chimiques

Biphenyl Compounds 0
Porphyrins 0
diphenyl 2L9GJK6MGN
DNA 9007-49-2
Guanidine JU58VJ6Y3B

Types de publication

Journal Article Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

128954

Informations de copyright

Copyright © 2022 The Authors. Published by Elsevier Ltd.. All rights reserved.

Déclaration de conflit d'intérêts

Declaration of Competing Interest The authors declare that they have no known competing financial interests or personal relationships that could have appeared to influence the work reported in this paper.

Auteurs

Nikolina Stipaničev (N)

School of Chemistry, Trinity College Dublin, 152-160 Pearse Street, Dublin 2, Ireland.

Konstantin Raabe (K)

School of Chemistry, Trinity College Dublin, 152-160 Pearse Street, Dublin 2, Ireland.

Isabel Rozas (I)

School of Chemistry, Trinity College Dublin, 152-160 Pearse Street, Dublin 2, Ireland. Electronic address: rozasi@tcd.ie.

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Classifications MeSH