Promising Perspectives of the Antiproliferative GPER Inverse Agonist ERα17p in Breast Cancer.
GPER
apoptosis
peptide
triple-negative breast cancer
Journal
Cells
ISSN: 2073-4409
Titre abrégé: Cells
Pays: Switzerland
ID NLM: 101600052
Informations de publication
Date de publication:
18 02 2023
18 02 2023
Historique:
received:
02
12
2022
revised:
07
02
2023
accepted:
14
02
2023
entrez:
25
2
2023
pubmed:
26
2
2023
medline:
3
3
2023
Statut:
epublish
Résumé
The estrogen receptor α (ERα) corresponds to a large platform in charge of the recruitment of a panel of molecules, including steroids and related heterocyclic derivatives, oligonucleotides, peptides and proteins. Its 295-311 region is particularly targeted by post-translational modifications, suggesting that it could be crucial for the control of transcription. In addition to anionic phospholipids, the ERα 295-311 fragment interacts with Ca
Identifiants
pubmed: 36831322
pii: cells12040653
doi: 10.3390/cells12040653
pmc: PMC9954065
pii:
doi:
Substances chimiques
Estrogen Receptor alpha
0
Estrogens
0
Receptors, G-Protein-Coupled
0
Peptides
0
Types de publication
Journal Article
Research Support, Non-U.S. Gov't
Langues
eng
Sous-ensembles de citation
IM
Références
Biochem Biophys Res Commun. 2012 Mar 9;419(2):356-61
pubmed: 22342729
Methods Mol Biol. 2016;1366:241-259
pubmed: 26585140
Chem Sci. 2019 Oct 3;10(45):10595-10600
pubmed: 32110345
Bioorg Med Chem Lett. 2018 Feb 15;28(4):658-663
pubmed: 29395974
Cells. 2019 Mar 07;8(3):
pubmed: 30866584
Essays Biochem. 2021 Dec 17;65(6):867-875
pubmed: 34028522
Anticancer Agents Med Chem. 2019;19(6):760-771
pubmed: 30451119
Biochem J. 2015 Nov 15;472(1):97-109
pubmed: 26371374
Front Endocrinol (Lausanne). 2020 Nov 23;11:591217
pubmed: 33329395
Biochemistry. 2016 Sep 27;55(38):5366-76
pubmed: 27641460
Sci Rep. 2023 Jan 24;13(1):1326
pubmed: 36693877
Mol Oncol. 2013 Jun;7(3):595-610
pubmed: 23474223
Steroids. 2012 Aug;77(10):979-87
pubmed: 22426414
Mol Endocrinol. 2000 Oct;14(10):1649-60
pubmed: 11043579
Nucl Recept Signal. 2008 Apr 18;6:e007
pubmed: 18432312
EMBO J. 1992 Oct;11(10):3681-94
pubmed: 1327748
J Steroid Biochem Mol Biol. 2018 Feb;176:49-56
pubmed: 28249728
Essays Biochem. 2021 Dec 17;65(6):857-866
pubmed: 34061186
Chirality. 2013 Oct;25(10):628-42
pubmed: 23925889
J Exp Clin Cancer Res. 2019 Aug 1;38(1):335
pubmed: 31370872
Front Endocrinol (Lausanne). 2022 Jun 30;13:943343
pubmed: 35846328
Endocrinology. 2003 Jun;144(6):2425-36
pubmed: 12746304
Int J Mol Sci. 2019 Jan 14;20(2):
pubmed: 30646517
Biochemistry. 1995 Oct 3;34(39):12605-15
pubmed: 7548010
J Steroid Biochem Mol Biol. 2019 May;189:176-186
pubmed: 30851383
Int J Mol Sci. 2018 Jun 27;19(7):
pubmed: 29954076
Front Endocrinol (Lausanne). 2020 Mar 31;11:148
pubmed: 32296387
Front Endocrinol (Lausanne). 2022 Sep 06;13:954629
pubmed: 36147566
Clin Cancer Res. 2006 Nov 1;12(21):6359-66
pubmed: 17085646
Cells. 2019 Jun 14;8(6):
pubmed: 31207943
Future Med Chem. 2015;7(4):437-48
pubmed: 25875871
Molecules. 2018 Apr 12;23(4):
pubmed: 29649162
Nucleic Acids Res. 2022 Jan 7;50(D1):D439-D444
pubmed: 34791371
Cancers (Basel). 2022 May 21;14(10):
pubmed: 35626139
Ann Pharm Fr. 2019 Nov;77(6):488-495
pubmed: 31563266
Cells. 2020 Mar 04;9(3):
pubmed: 32143514
Anticancer Agents Med Chem. 2018;18(11):1629-1638
pubmed: 29745344
Mol Endocrinol. 2005 Nov;19(11):2671-84
pubmed: 15961505
J Pept Sci. 2015 Feb;21(2):95-104
pubmed: 25530026
EMBO J. 2009 Mar 4;28(5):523-32
pubmed: 19153601
Front Endocrinol (Lausanne). 2020 Aug 04;11:517
pubmed: 32849301
J Steroid Biochem Mol Biol. 2007 Apr;104(1-2):1-10
pubmed: 17258904
J Steroid Biochem Mol Biol. 2008 Mar;109(1-2):138-49
pubmed: 18262408
Oncogene. 2010 Apr 22;29(16):2404-14
pubmed: 20101208
Methods Mol Biol. 2022;2418:345-362
pubmed: 35119674
Mol Oncol. 2011 Feb;5(1):36-47
pubmed: 21163714
Front Genet. 2018 Dec 12;9:641
pubmed: 30619466
Mol Cell Endocrinol. 2007 Mar 30;268(1-2):37-49
pubmed: 17316976
Nat Rev Drug Discov. 2020 Jun;19(6):389-413
pubmed: 32494050
J Cell Biochem. 2011 Dec;112(12):3786-96
pubmed: 21826705
Mol Endocrinol. 1997 Jun;11(6):747-54
pubmed: 9171238
Mol Cell Endocrinol. 2013 Aug 25;376(1-2):23-32
pubmed: 23748028
Mol Cancer Res. 2014 Nov;12(11):1644-1654
pubmed: 25030371
Breast Cancer Res Treat. 2010 Aug;123(1):51-8
pubmed: 19902352
Bioessays. 2022 Dec;44(12):e2200148
pubmed: 36192154
Breast Cancer Res Treat. 2019 Feb;174(1):121-127
pubmed: 30478785
Biomolecules. 2020 Mar 26;10(4):
pubmed: 32224970
Front Endocrinol (Lausanne). 2021 Mar 17;12:578250
pubmed: 33815268
Mol Cell Endocrinol. 2009 Sep 24;308(1-2):32-8
pubmed: 19464786
Cells. 2020 Feb 15;9(2):
pubmed: 32075246
Endocrinology. 2007 Jul;148(7):3236-45
pubmed: 17379646
Front Endocrinol (Lausanne). 2014 May 06;5:66
pubmed: 24834064
Amino Acids. 2017 Apr;49(4):705-713
pubmed: 28185014
Int J Endocrinol. 2022 May 9;2022:7690166
pubmed: 35586275
Int J Mol Sci. 2018 Dec 02;19(12):
pubmed: 30513833