Radiochemistry for positron emission tomography.


Journal

Nature communications
ISSN: 2041-1723
Titre abrégé: Nat Commun
Pays: England
ID NLM: 101528555

Informations de publication

Date de publication:
05 06 2023
Historique:
received: 29 03 2022
accepted: 30 01 2023
medline: 7 6 2023
pubmed: 6 6 2023
entrez: 5 6 2023
Statut: epublish

Résumé

Positron emission tomography (PET) constitutes a functional imaging technique that is harnessed to probe biological processes in vivo. PET imaging has been used to diagnose and monitor the progression of diseases, as well as to facilitate drug development efforts at both preclinical and clinical stages. The wide applications and rapid development of PET have ultimately led to an increasing demand for new methods in radiochemistry, with the aim to expand the scope of synthons amenable for radiolabeling. In this work, we provide an overview of commonly used chemical transformations for the syntheses of PET tracers in all aspects of radiochemistry, thereby highlighting recent breakthrough discoveries and contemporary challenges in the field. We discuss the use of biologicals for PET imaging and highlight general examples of successful probe discoveries for molecular imaging with PET - with a particular focus on translational and scalable radiochemistry concepts that have been entered to clinical use.

Identifiants

pubmed: 37277339
doi: 10.1038/s41467-023-36377-4
pii: 10.1038/s41467-023-36377-4
pmc: PMC10241151
doi:

Substances chimiques

Radiopharmaceuticals 0

Types de publication

Journal Article Review Research Support, N.I.H., Extramural Research Support, Non-U.S. Gov't

Langues

eng

Sous-ensembles de citation

IM

Pagination

3257

Subventions

Organisme : NINDS NIH HHS
ID : R61 NS130128
Pays : United States
Organisme : NIA NIH HHS
ID : RF1 AG073428
Pays : United States
Organisme : NIA NIH HHS
ID : R01 AG079956
Pays : United States
Organisme : NIA NIH HHS
ID : R21 AG080262
Pays : United States
Organisme : NIA NIH HHS
ID : R01 AG070060
Pays : United States
Organisme : NIA NIH HHS
ID : R21 AG078058
Pays : United States

Informations de copyright

© 2023. The Author(s).

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Auteurs

Jian Rong (J)

Department of Radiology and Imaging Sciences, Emory University, 1364 Clifton Rd, Atlanta, GA, 30322, USA.
Division of Nuclear Medicine and Molecular Imaging, Massachusetts General Hospital & Department of Radiology, Harvard Medical School, Boston, MA, 02114, USA.

Ahmed Haider (A)

Department of Radiology and Imaging Sciences, Emory University, 1364 Clifton Rd, Atlanta, GA, 30322, USA.
Division of Nuclear Medicine and Molecular Imaging, Massachusetts General Hospital & Department of Radiology, Harvard Medical School, Boston, MA, 02114, USA.

Troels E Jeppesen (TE)

Division of Nuclear Medicine and Molecular Imaging, Massachusetts General Hospital & Department of Radiology, Harvard Medical School, Boston, MA, 02114, USA.

Lee Josephson (L)

Division of Nuclear Medicine and Molecular Imaging, Massachusetts General Hospital & Department of Radiology, Harvard Medical School, Boston, MA, 02114, USA.

Steven H Liang (SH)

Department of Radiology and Imaging Sciences, Emory University, 1364 Clifton Rd, Atlanta, GA, 30322, USA. steven.liang@emory.edu.
Division of Nuclear Medicine and Molecular Imaging, Massachusetts General Hospital & Department of Radiology, Harvard Medical School, Boston, MA, 02114, USA. steven.liang@emory.edu.

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