Titre : Mécanismes moléculaires de l'action pharmacologique

Mécanismes moléculaires de l'action pharmacologique : Questions médicales fréquentes

Termes MeSH sélectionnés :

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"L'imagerie par résonance magnétique et la tomographie permettent d'observer les effets des médicaments." } }, { "@type": "Question", "name": "Comment les biomarqueurs sont-ils utilisés dans le diagnostic ?", "position": 4, "acceptedAnswer": { "@type": "Answer", "text": "Les biomarqueurs aident à évaluer l'efficacité et la sécurité des médicaments en fonction de leur mécanisme." } }, { "@type": "Question", "name": "Quel rôle joue la pharmacogénomique dans le diagnostic ?", "position": 5, "acceptedAnswer": { "@type": "Answer", "text": "Elle permet d'adapter les traitements en fonction des variations génétiques influençant les mécanismes d'action." } }, { "@type": "Question", "name": "Quels symptômes indiquent un effet pharmacologique ?", "position": 6, "acceptedAnswer": { "@type": "Answer", "text": "Les symptômes peuvent inclure des changements physiologiques, des effets secondaires ou des améliorations cliniques." } }, { "@type": "Question", "name": "Comment les effets indésirables sont-ils liés aux mécanismes d'action ?", "position": 7, "acceptedAnswer": { "@type": "Answer", "text": "Les effets indésirables résultent souvent d'interactions non spécifiques avec des cibles moléculaires." } }, { "@type": "Question", "name": "Quels symptômes sont associés aux médicaments ciblant les récepteurs ?", "position": 8, "acceptedAnswer": { "@type": "Answer", "text": "Les symptômes peuvent inclure des modifications de la perception, de l'humeur ou de la douleur." } }, { "@type": "Question", "name": "Comment les symptômes varient-ils selon les mécanismes d'action ?", "position": 9, "acceptedAnswer": { "@type": "Answer", "text": "Les symptômes varient en fonction des cibles moléculaires et des voies de signalisation affectées." } }, { "@type": "Question", "name": "Quels symptômes peuvent indiquer une surdose ?", "position": 10, "acceptedAnswer": { "@type": "Answer", "text": "Des symptômes tels que des nausées, des vertiges ou des troubles de la conscience peuvent indiquer une surdose." } }, { "@type": "Question", "name": "Comment prévenir les effets indésirables des médicaments ?", "position": 11, "acceptedAnswer": { "@type": "Answer", "text": "Une évaluation des mécanismes d'action et des interactions médicamenteuses peut aider à prévenir les effets indésirables." } }, { "@type": "Question", "name": "Quel rôle joue l'éducation des patients dans la prévention ?", "position": 12, "acceptedAnswer": { "@type": "Answer", "text": "L'éducation des patients sur les mécanismes d'action des médicaments peut améliorer l'adhésion et réduire les risques." } }, { "@type": "Question", "name": "Comment les études cliniques aident-elles à prévenir les complications ?", "position": 13, "acceptedAnswer": { "@type": "Answer", "text": "Les études cliniques identifient les mécanismes d'action et les effets indésirables potentiels, permettant une meilleure prévention." } }, { "@type": "Question", "name": "Quels facteurs influencent la prévention des effets indésirables ?", "position": 14, "acceptedAnswer": { "@type": "Answer", "text": "Les facteurs incluent la génétique, l'âge, les comorbidités et les interactions médicamenteuses." } }, { "@type": "Question", "name": "Comment les recommandations de traitement aident-elles à prévenir les risques ?", "position": 15, "acceptedAnswer": { "@type": "Answer", "text": "Les recommandations basées sur les mécanismes d'action aident à choisir des traitements plus sûrs et efficaces." } }, { "@type": "Question", "name": "Comment les médicaments ciblent-ils des mécanismes spécifiques ?", "position": 16, "acceptedAnswer": { "@type": "Answer", "text": "Les médicaments sont conçus pour interagir avec des cibles moléculaires spécifiques, comme des enzymes ou des récepteurs." } }, { "@type": "Question", "name": "Quels traitements utilisent des mécanismes d'action innovants ?", "position": 17, "acceptedAnswer": { "@type": "Answer", "text": "Les thérapies géniques et les médicaments biologiques exploitent des mécanismes d'action novateurs." } }, { "@type": "Question", "name": "Comment les traitements sont-ils personnalisés ?", "position": 18, "acceptedAnswer": { "@type": "Answer", "text": "Les traitements sont adaptés en fonction des caractéristiques moléculaires des patients et des médicaments." } }, { "@type": "Question", "name": "Quel est l'impact des mécanismes d'action sur l'efficacité des traitements ?", "position": 19, "acceptedAnswer": { "@type": "Answer", "text": "Une compréhension approfondie des mécanismes d'action permet d'optimiser l'efficacité et de réduire les effets secondaires." } }, { "@type": "Question", "name": "Comment les combinaisons de médicaments exploitent les mécanismes d'action ?", "position": 20, "acceptedAnswer": { "@type": "Answer", "text": "Les combinaisons de médicaments peuvent cibler plusieurs mécanismes pour améliorer l'efficacité thérapeutique." } }, { "@type": "Question", "name": "Quelles complications peuvent survenir avec des médicaments ?", "position": 21, "acceptedAnswer": { "@type": "Answer", "text": "Les complications peuvent inclure des réactions allergiques, des effets toxiques ou des interactions médicamenteuses." } }, { "@type": "Question", "name": "Comment les mécanismes d'action influencent-ils les complications ?", "position": 22, "acceptedAnswer": { "@type": "Answer", "text": "Les mécanismes d'action peuvent déterminer la sévérité et la nature des complications observées." } }, { "@type": "Question", "name": "Quels sont les signes de complications graves ?", "position": 23, "acceptedAnswer": { "@type": "Answer", "text": "Des signes tels que des difficultés respiratoires, des éruptions cutanées ou des douleurs thoraciques peuvent indiquer des complications graves." } }, { "@type": "Question", "name": "Comment gérer les complications liées aux médicaments ?", "position": 24, "acceptedAnswer": { "@type": "Answer", "text": "La gestion des complications implique l'arrêt du médicament, le traitement des symptômes et la surveillance étroite." } }, { "@type": "Question", "name": "Quel rôle joue la pharmacovigilance dans la détection des complications ?", "position": 25, "acceptedAnswer": { "@type": "Answer", "text": "La pharmacovigilance surveille les effets indésirables et les complications pour améliorer la sécurité des médicaments." } }, { "@type": "Question", "name": "Quels facteurs de risque influencent l'efficacité des médicaments ?", "position": 26, "acceptedAnswer": { "@type": "Answer", "text": "Les facteurs incluent l'âge, le sexe, la génétique et les comorbidités qui peuvent affecter l'efficacité." } }, { "@type": "Question", "name": "Comment les interactions médicamenteuses sont-elles un facteur de risque ?", "position": 27, "acceptedAnswer": { "@type": "Answer", "text": "Les interactions médicamenteuses peuvent altérer les mécanismes d'action et augmenter le risque d'effets indésirables." } }, { "@type": "Question", "name": "Quel impact a l'alimentation sur les mécanismes d'action ?", "position": 28, "acceptedAnswer": { "@type": "Answer", "text": "L'alimentation peut influencer l'absorption et le métabolisme des médicaments, affectant leur efficacité." } }, { "@type": "Question", "name": "Comment le mode de vie affecte-t-il les traitements ?", "position": 29, "acceptedAnswer": { "@type": "Answer", "text": "Le mode de vie, y compris l'exercice et le tabagisme, peut modifier la réponse aux médicaments et leurs mécanismes d'action." } }, { "@type": "Question", "name": "Quels facteurs environnementaux influencent les effets des médicaments ?", "position": 30, "acceptedAnswer": { "@type": "Answer", "text": "Les facteurs environnementaux, comme la pollution, peuvent interagir avec les mécanismes d'action des médicaments." } } ] } ] }

Sous-catégories

86 au total
└─

Antagonistes des récepteurs aux angiotensines

Angiotensin Receptor Antagonists D057911 - D27.505.519.162
└─

Agents antiglycation

Antiglycation Agents D000093744 - D27.505.519.182
└─

Antagonistes des récepteurs de la bradykinine

Bradykinin Receptor Antagonists D065168 - D27.505.519.265
└─

Agents de déplétion en cystine

Cystine Depleting Agents D065104 - D27.505.519.334
└─

Inducteurs des enzymes du cytochrome P-450

Cytochrome P-450 Enzyme Inducers D065693 - D27.505.519.349
└─

Antagonistes des récepteurs de l'endothéline

Endothelin Receptor Antagonists D065128 - D27.505.519.364
└─

Activateurs d'enzymes

Enzyme Activators D020536 - D27.505.519.374
└─

Antienzymes

Enzyme Inhibitors D004791 - D27.505.519.389
└─

Réactivateurs d'enzymes

Enzyme Reactivators D004793 - D27.505.519.405
└─

Modulateurs de la fibrinolyse

Fibrin Modulating Agents D050299 - D27.505.519.421
└─

Modulateurs du transport transmembranaire

Membrane Transport Modulators D049990 - D27.505.519.562
└─

Modulateurs de la mitose

Mitosis Modulators D050258 - D27.505.519.593
└─

Peptidomimétiques

Peptidomimetics D057786 - D27.505.519.828
└─└─

Antagonistes du récepteur de type 1 de l'angiotensine-II

Angiotensin II Type 1 Receptor Blockers D047228 - D27.505.519.162.500
└─└─

Antagonistes du récepteur de type 2 de l'angiotensine-II

Angiotensin II Type 2 Receptor Blockers D057912 - D27.505.519.162.750
└─└─

Piégeurs de radicaux libres

Free Radical Scavengers D016166 - D27.505.519.217.500
└─└─

Antagonistes du récepteur B1 de la bradykinine

Bradykinin B1 Receptor Antagonists D065169 - D27.505.519.265.249
└─└─

Inducteurs du cytochrome P-450 CYP1A2

Cytochrome P-450 CYP1A2 Inducers D065694 - D27.505.519.349.120
└─└─

Inducteurs du cytochrome P-450 CYP2B6

Cytochrome P-450 CYP2B6 Inducers D065695 - D27.505.519.349.260
└─└─

Inducteurs du cytochrome P-450 CYP2C8

Cytochrome P-450 CYP2C8 Inducers D065696 - D27.505.519.349.308
└─└─

Inducteurs du cytochrome P-450 CYP2C9

Cytochrome P-450 CYP2C9 Inducers D065698 - D27.505.519.349.320
└─└─

Inducteurs du cytochrome P-450 CYP2C19

Cytochrome P-450 CYP2C19 Inducers D065697 - D27.505.519.349.350
└─└─

Inducteurs du cytochrome P-450 CYP2D6

Cytochrome P-450 CYP2D6 Inducers D065699 - D27.505.519.349.500
└─└─

Inducteurs du cytochrome P-450 CYP2E1

Cytochrome P-450 CYP2E1 Inducers D065700 - D27.505.519.349.600
└─└─

Inducteurs du cytochrome P-450 CYP3A

Cytochrome P-450 CYP3A Inducers D065701 - D27.505.519.349.700
└─└─

Antagonistes du récepteur de type A de l'endothéline

Endothelin A Receptor Antagonists D065130 - D27.505.519.364.500
└─└─

Antagonistes du récepteur de type B de l'endothéline

Endothelin B Receptor Antagonists D065131 - D27.505.519.364.750
└─└─

Activateurs de la Carbamoyl phosphate synthetase I

Carbamoyl Phosphate Synthetase I Activators D065097 - D27.505.519.374.099
└─└─

Activateurs de la GTPase

GTP Phosphohydrolase Activators D020549 - D27.505.519.374.200
└─└─

Inhibiteurs des protéines activatrices de la 5-lipoxygénase

5-Lipoxygenase-Activating Protein Inhibitors D058946 - D27.505.519.389.086
└─└─

Inhibiteurs de l'acétaldéhyde déshydrogénase

Acetaldehyde Dehydrogenase Inhibitors D065086 - D27.505.519.389.089
└─└─

Inhibiteurs de l'adénosine désaminase

Adenosine Deaminase Inhibitors D058892 - D27.505.519.389.092
└─└─

Inhibiteurs des adénylate cyclases

Adenylyl Cyclase Inhibitors D000067956 - D27.505.519.389.108
└─└─

Inhibiteurs de la calcineurine

Calcineurin Inhibitors D065095 - D27.505.519.389.174
└─└─

Inhibiteurs de l'anhydrase carbonique

Carbonic Anhydrase Inhibitors D002257 - D27.505.519.389.200
└─└─

Inhibiteurs et modulateurs de la gamma-secrétase

Gamma Secretase Inhibitors and Modulators D000091062 - D27.505.519.389.315
└─└─

Inhibiteurs des enzymes du cytochrome P-450

Cytochrome P-450 Enzyme Inhibitors D065607 - D27.505.519.389.335
└─└─

Antifoliques

Folic Acid Antagonists D005493 - D27.505.519.389.350
└─└─

Inhibiteurs de désacétylase d'histone

Histone Deacetylase Inhibitors D056572 - D27.505.519.389.360
└─└─

Inhibiteurs de l'intégrase

Integrase Inhibitors D019429 - D27.505.519.389.375
└─└─

Inhibiteurs de la lipoxygénase

Lipoxygenase Inhibitors D016859 - D27.505.519.389.480
└─└─

Inhibiteurs de la monoamine oxydase

Monoamine Oxidase Inhibitors D008996 - D27.505.519.389.616
└─└─

Inhibiteurs de la synthèse d'acide nucléique

Nucleic Acid Synthesis Inhibitors D019384 - D27.505.519.389.675
└─└─

Inhibiteurs de l'ornithine décarboxylase

Ornithine Decarboxylase Inhibitors D065108 - D27.505.519.389.705
└─└─

Inhibiteurs de la phosphodiestérase

Phosphodiesterase Inhibitors D010726 - D27.505.519.389.735
└─└─

Inhibiteurs des phosphoinositide-3 kinases

Phosphoinositide-3 Kinase Inhibitors D000081082 - D27.505.519.389.736
└─└─

Inhibiteurs de la phospholipase A2

Phospholipase A2 Inhibitors D064801 - D27.505.519.389.737
└─└─

Inhibiteurs de prolyle hydroxylases

Prolyl-Hydroxylase Inhibitors D064800 - D27.505.519.389.740
└─└─

Inhibiteurs de protéases

Protease Inhibitors D011480 - D27.505.519.389.745
└─└─

Inhibiteurs de protéines kinases

Protein Kinase Inhibitors D047428 - D27.505.519.389.755
└─└─

Inhibiteurs de la synthèse protéique

Protein Synthesis Inhibitors D011500 - D27.505.519.389.760
└─└─

Inhibiteurs de la pompe à protons

Proton Pump Inhibitors D054328 - D27.505.519.389.848
└─└─

Agents découplants

Uncoupling Agents D014475 - D27.505.519.389.936
└─└─

Agonistes de canaux chlorure

Chloride Channel Agonists D065101 - D27.505.519.562.311
└─└─

Agonistes de canaux sodiques

Sodium Channel Agonists D062687 - D27.505.519.562.625
└─└─

Mitogènes

Mitogens D008934 - D27.505.519.593.624
└─└─

Gazotransmetteurs

Gasotransmitters D064426 - D27.505.519.625.270
└─└─└─

Inhibiteurs de la synthèse d'acides gras

Fatty Acid Synthesis Inhibitors D054872 - D27.505.519.186.071.401
└─└─└─

Inhibiteurs du cytochrome P-450 CYP1A2

Cytochrome P-450 CYP1A2 Inhibitors D065609 - D27.505.519.389.335.120
└─└─└─

Inhibiteurs du cytochrome P-450 CYP2B6

Cytochrome P-450 CYP2B6 Inhibitors D065686 - D27.505.519.389.335.260
└─└─└─

Inhibiteurs du cytochrome P-450 CYP2C8

Cytochrome P-450 CYP2C8 Inhibitors D065687 - D27.505.519.389.335.308
└─└─└─

Inhibiteurs du cytochrome P-450 CYP2C19

Cytochrome P-450 CYP2C19 Inhibitors D065689 - D27.505.519.389.335.319
└─└─└─

Inhibiteurs du cytochrome P-450 CYP2C9

Cytochrome P-450 CYP2C9 Inhibitors D065688 - D27.505.519.389.335.329
└─└─└─

Inhibiteurs du cytochrome P-450 CYP2D6

Cytochrome P-450 CYP2D6 Inhibitors D065690 - D27.505.519.389.335.368
└─└─└─

Inhibiteurs du cytochrome P-450 CYP2E1

Cytochrome P-450 CYP2E1 Inhibitors D065691 - D27.505.519.389.335.421
└─└─└─

Inhibiteurs du cytochrome P-450 CYP3A

Cytochrome P-450 CYP3A Inhibitors D065692 - D27.505.519.389.335.503
└─└─└─

Inhibiteurs de la phosphodiestérase-3

Phosphodiesterase 3 Inhibitors D058987 - D27.505.519.389.735.249
└─└─└─

Inhibiteurs de la phosphodiestérase-4

Phosphodiesterase 4 Inhibitors D058988 - D27.505.519.389.735.374
└─└─└─

Inhibiteurs de la phosphodiestérase-5

Phosphodiesterase 5 Inhibitors D058986 - D27.505.519.389.735.500
└─└─└─

Inhibiteurs de l'enzyme de conversion de l'angiotensine

Angiotensin-Converting Enzyme Inhibitors D000806 - D27.505.519.389.745.085
└─└─└─

Inhibiteurs de la cystéine protéinase

Cysteine Proteinase Inhibitors D015853 - D27.505.519.389.745.325
└─└─└─

Inhibiteurs de métalloprotéinases matricielles

Matrix Metalloproteinase Inhibitors D061965 - D27.505.519.389.745.610
└─└─└─

Inhibiteurs du protéasome

Proteasome Inhibitors D061988 - D27.505.519.389.745.705
└─└─└─

Inhibiteurs de la rénine

Renin Inhibitors D000092502 - D27.505.519.389.745.753
└─└─└─

Inhibiteurs de la sérine protéinase

Serine Proteinase Inhibitors D015842 - D27.505.519.389.745.800
└─└─└─

Inhibiteurs des Janus kinases

Janus Kinase Inhibitors D000075242 - D27.505.519.389.755.500
└─└─└─

Inhibiteurs de protéine-tyrosine kinase

Tyrosine Protein Kinase Inhibitors D000092004 - D27.505.519.389.755.875
└─└─└─

Agonistes de canaux sodiques épithéliaux

Epithelial Sodium Channel Agonists D062708 - D27.505.519.562.625.249
└─└─└─

Agonistes de canaux sodiques voltage-dépendants

Voltage-Gated Sodium Channel Agonists D061585 - D27.505.519.562.625.500
└─└─└─

Inhibiteurs de canaux ioniques sensibles à l'acidité

Acid Sensing Ion Channel Blockers D062646 - D27.505.519.562.750.100
└─└─└─

Modulateurs de la polymérisation de la tubuline

Tubulin Modulators D050257 - D27.505.519.593.249.500
└─└─└─└─

Inhibiteurs des vasopeptidases

Vasopeptidase Inhibitors D000075563 - D27.505.519.389.745.085.500
└─└─└─└─

Inhibiteurs des caspases

Caspase Inhibitors D061945 - D27.505.519.389.745.325.500
└─└─└─└─

Inhibiteurs de serine peptidase de type Kazal

Serine Peptidase Inhibitors, Kazal Type D000074162 - D27.505.519.389.745.800.562
└─└─└─└─

Serpines

Serpins D015843 - D27.505.519.389.745.800.675
└─└─└─└─

Inhibiteurs trypsiques

Trypsin Inhibitors D014361 - D27.505.519.389.745.800.900

Sources (4688 au total)

Effect of thickness on color and translucency of a multi-color polymer-infiltrated ceramic-network material.

To evaluate the effect of thickness on color and translucency of a multi-color polymer-infiltrated ceramic-network (PICN) material.... Specimens of 0.5, 1.0, 1.5 mm thicknesses were obtained by sectioning VITA ENAMIC® multiColor (E-MC) High Translucent CAD-CAM blocks (1M1-HT, 1M2-HT, 2M2-HT, 3M2-HT, and 4M2-HT). Spectral reflectance ... In general, ΔE... The gradient in color and translucency of E-MC PICN material was influenced by the thickness of the CAD-CAM block. In addition, color and TP transition values between the layers depends on the thickne... The effect of thickness must be taken into account by dental technicians and dentists when CAD-CAM multicolor PICN materials are used....

Linked color imaging provides enhanced visibility with a high color difference in upper gastrointestinal neoplasms.

The aim of this post-hoc analysis in a randomized, controlled, multicenter trial was to evaluate the visibility of upper gastrointestinal (UGI) neoplasms detected using linked color imaging (LCI) comp... The visibility of the detected UGI neoplasm images obtained using both WLI and LCI was subjectively reviewed, and the median color difference (ΔE) between each lesion and the surrounding mucosa accord... A total of 120 neoplasms, including 10, 32, and 78 neoplasms in the pharynx, esophagus, and stomach, respectively, were analyzed in this study. LCI enhanced the visibility 80.9% and 93.6% of neoplasms... Color differences were independently associated with missing gastric neoplasms under WLI, suggesting that LCI has an obvious advantage over WLI in enhancing neoplastic visibility....

Linked color imaging improves visibility of colorectal serrated lesion by high color contrast to surrounding mucosa.

This study aimed to objectively evaluate the efficacy of linked color imaging (LCI) in diagnosing colorectal serrated lesions by utilizing visibility scores and color differences.... We examined 89 serrated lesions, including 36 hyperplastic polyps (HPs), 47 sessile serrated lesions (SSLs), and six traditional serrated adenomas (TSAs). Visibility changes were scored by six endosco... The visibility scores of both HPs and SSLs in LCI were significantly higher than that in WLI (HPs, 3.67/2.89, P < 0.001; SSLs, 3.07/2.36, P < 0.001). Furthermore, SSLs showed a significantly higher L*... Linked color imaging showed higher color contrast between serrated lesions and the surrounding mucosae compared with WLI, indicating improved visibility of colorectal serrated lesion using LCI....

Color change of tooth-colored restorative materials bonded to silver diamine fluoride-treated dentine: a systematic review.

The desirable properties of silver diamine fluoride (SDF) make it an effective agent for managing dental caries and tooth hypersensitivity. There are several clinical instances that SDF application mi... Comprehensive search of PubMed, Embase, Scopus and ISI Web of Science databases (until August 2023) as well as reference lists of retrieved studies was performed. In vitro studies reported color or co... Eleven studies/reports with a total of 394 tooth-colored restorations placed following a) no SDF (control) or b) SDF with/without potassium iodide (KI)/glutathione dentine pre-treatments were included... The limited evidence suggested comparable color changes of RBC restorations with and without 38% SDF + KI pre-treatment up to 60 days. The included studies lacked uniformity in methodology and reporte... The protocol of this systematic review was registered in PROSPERO database under number CRD42023485083....

In vitro surface and color changes of tooth-colored restorative materials after sport and energy drink cyclic immersions.

There has not been any research conducted on surface properties and color changes from sport and energy drinks on bulk-fill resin composite, nanohybrid resin composite and glass ionomer restorative ma... One hundred and forty-seven specimens of each tooth-colored restorative material were prepared in a polytetrafluoroethylene mold (10 mm. in diameter and 2 mm. in thickness). Before immersion, baseline... After immersion, the glass ionomer restorative material had statistically less hardness, more roughness and more color changes than the others (P < 0.05). Energy drink groups statistically caused more... Sport and energy drinks affected hardness, roughness, and color changes in all the tooth-colored restorative materials evaluated....

Effect of hydrogen peroxide versus charcoal-based whitening mouthwashes on color, surface roughness, and color stability of enamel.

Patients tend to favor the whitening mouthwashes as they are easily applied and affordable. This study aimed to evaluate the effect of hydrogen peroxide versus charcoal-based whitening mouthwashes on ... A total of 21 permanent central incisor teeth extracted for periodontal reasons were used in the present study. Teeth roots were sectioned and crowns were mounted in self-cured acrylic resin blocks. T... Color change results revealed that both whitening mouthwashes were able to restore color comparable to the control group with no significant difference between them. Regarding surface roughness, the c... Hydrogen peroxide and charcoal-based whitening mouthwashes improve the color of enamel with no adverse effect on the surface roughness. Both whitening mouthwashes were beneficial to maintain the color...