questionsmedicales.fr
Acides aminés, peptides et protéines
Protéines
Hémoprotéines
Cytochromes
Cytochrome P-450 enzyme system
Famille-2 de cytochromes P450
Limonène hydroxylases
Cytochrome P-450 CYP2C9
Cytochrome P-450 CYP2C9 : Questions médicales fréquentes
Termes MeSH sélectionnés :
Diagnostic
5
Tests génétiques
Polymorphisme génétique
Effets indésirables
Réponse au traitement
Interactions médicamenteuses
Profil métabolique
Métabolisme hépatique
Analyses sanguines
Symptômes
5
Nausées
Réactions allergiques
Surdose
Douleurs abdominales
Effets secondaires
Efficacité des médicaments
Carence enzymatique
Effets indésirables
Toxicité médicamenteuse
Éruptions cutanées
Prévention
5
Prévention
Suivi régulier
Anticoagulants
Saignement
Interactions médicamenteuses
Information médicale
Tests préventifs
Complications
Sensibilisation
Tests génétiques
Traitements
5
Ajustement de dose
Tests génétiques
Gestion des interactions
Surveillance thérapeutique
Traitements alternatifs
Médicaments
Surdose
Soins symptomatiques
Complications
5
Complications
Réactions allergiques
Surdose
Dommages organiques
Gestion des complications
Surveillance étroite
Déficience enzymatique
Maladies chroniques
Interactions médicamenteuses
Hospitalisations
Facteurs de risque
5
Facteurs de risque
Génétique
Alimentation
Inhibition enzymatique
Antifongiques
Inhibition enzymatique
Maladies hépatiques
Métabolisme des médicaments
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"name": "Quels conseils pour les patients sous anticoagulants ?",
"position": 12,
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"position": 14,
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"@type": "Question",
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"name": "Comment ajuster les doses pour CYP2C9 ?",
"position": 16,
"acceptedAnswer": {
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{
"@type": "Question",
"name": "Quels médicaments sont métabolisés par CYP2C9 ?",
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"acceptedAnswer": {
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}
},
{
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"name": "Quels traitements alternatifs pour les déficients ?",
"position": 19,
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"name": "Comment traiter une surdose liée à CYP2C9 ?",
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"acceptedAnswer": {
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"position": 23,
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"@type": "Question",
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"position": 24,
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}
},
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"position": 25,
"acceptedAnswer": {
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}
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{
"@type": "Question",
"name": "Quels facteurs influencent CYP2C9 ?",
"position": 26,
"acceptedAnswer": {
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}
},
{
"@type": "Question",
"name": "Comment l'âge affecte CYP2C9 ?",
"position": 27,
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},
{
"@type": "Question",
"name": "Quel rôle de l'alimentation sur CYP2C9 ?",
"position": 28,
"acceptedAnswer": {
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"text": "Certaines substances alimentaires peuvent inhiber ou induire l'activité de CYP2C9."
}
},
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"name": "Quels médicaments augmentent le risque ?",
"position": 29,
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"name": "Comment les maladies hépatiques affectent CYP2C9 ?",
"position": 30,
"acceptedAnswer": {
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"text": "Les maladies hépatiques peuvent réduire l'activité de CYP2C9, affectant le métabolisme des médicaments."
}
}
]
}
]
}
Expert en Médecine, Optimisation des Parcours de Soins et Révision Médicale
Validation scientifique effectuée le 29/03/2025
Contenu vérifié selon les dernières recommandations médicales
3 publications dans cette catégorie
Affiliations :
Department of Pharmacology, Faculty of Pharmacy, University of Pécs, Rókus u. 2, Pécs H-7624, Hungary; Lab-on-a-Chip Research Group, János Szentágothai Research Centre, University of Pécs, Ifjúság útja 20, Pécs H-7624, Hungary. Electronic address: poor.miklos@pte.hu.
Publications dans "Cytochrome P-450 CYP2C9" :
In vitro interaction of potential antiviral TMPRSS2 inhibitors with human serum albumin and cytochrome P 450 isoenzymes.
Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie
2021-12-13
Interaction of myricetin, ampelopsin (dihydromyricetin), and their sulfate metabolites with serum albumin, cytochrome P450 (CYP2C9, 2C19, and 3A4) enzymes, and organic anion-transporting polypeptides (OATP1B1 and OATP2B1).
Pharmacology research & perspectives
Interaction of luteolin, naringenin, and their sulfate and glucuronide conjugates with human serum albumin, cytochrome P450 (CYP2C9, CYP2C19, and CYP3A4) enzymes and organic anion transporting polypeptide (OATP1B1 and OATP2B1) transporters.
Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie
2022-12-05
3 publications dans cette catégorie
Affiliations :
The Key laboratory of Geriatrics, Beijing Institute of Geriatrics, Beijing Hospital, National Center of Gerontology, National Health Commission, Institute of Geriatric Medicine, Chinese Academy of Medical Sciences, Beijing, P. R. China.
Publications dans "Cytochrome P-450 CYP2C9" :
2 publications dans cette catégorie
Affiliations :
Department of Pharmacology, Faculty of Pharmacy, University of Pécs, Rókus u. 2, Pécs H-7624, Hungary; Lab-on-a-Chip Research Group, János Szentágothai Research Centre, University of Pécs, Ifjúság útja 20, Pécs H-7624, Hungary.
Publications dans "Cytochrome P-450 CYP2C9" :
2 publications dans cette catégorie
Affiliations :
Department of Pharmacology, Faculty of Pharmacy, University of Pécs, Rókus u. 2, Pécs H-7624, Hungary; Lab-on-a-Chip Research Group, János Szentágothai Research Centre, University of Pécs, Ifjúság útja 20, Pécs H-7624, Hungary.
Publications dans "Cytochrome P-450 CYP2C9" :
2 publications dans cette catégorie
Affiliations :
The Key laboratory of Geriatrics, Beijing Institute of Geriatrics, Beijing Hospital, National Center of Gerontology, National Health Commission, Institute of Geriatric Medicine, Chinese Academy of Medical Sciences, Beijing, P. R. China.
Publications dans "Cytochrome P-450 CYP2C9" :
2 publications dans cette catégorie
Affiliations :
Cardiovascular Department, Beijing Hospital, National Center of Gerontology, Institute of Geriatric Medicine, Chinese Academy of Medical Sciences, Beijing, P. R. China.
Publications dans "Cytochrome P-450 CYP2C9" :
2 publications dans cette catégorie
Affiliations :
Laboratory of Clinical Pharmacy, The Sixth Affiliated Hospital of Wenzhou Medical University, The People's Hospital of Lishui, Lishui, P.R. China.
Publications dans "Cytochrome P-450 CYP2C9" :
2 publications dans cette catégorie
Affiliations :
Laboratory of Clinical Pharmacy, The Sixth Affiliated Hospital of Wenzhou Medical University, The People's Hospital of Lishui, Lishui, P.R. China.
Publications dans "Cytochrome P-450 CYP2C9" :
2 publications dans cette catégorie
Affiliations :
Laboratory of Clinical Pharmacy, The Sixth Affiliated Hospital of Wenzhou Medical University, The People's Hospital of Lishui, Lishui, P.R. China.
Publications dans "Cytochrome P-450 CYP2C9" :
2 publications dans cette catégorie
Affiliations :
Cardiovascular Department, Beijing Hospital, National Center of Gerontology, Institute of Geriatric Medicine, Chinese Academy of Medical Sciences, Beijing, P. R. China.
Publications dans "Cytochrome P-450 CYP2C9" :
2 publications dans cette catégorie
Affiliations :
Cardiovascular Department, Beijing Hospital, National Center of Gerontology, Institute of Geriatric Medicine, Chinese Academy of Medical Sciences, Beijing, P. R. China.
Publications dans "Cytochrome P-450 CYP2C9" :
2 publications dans cette catégorie
Affiliations :
The Key laboratory of Geriatrics, Beijing Institute of Geriatrics, Beijing Hospital, National Center of Gerontology, National Health Commission, Institute of Geriatric Medicine, Chinese Academy of Medical Sciences, Beijing, P. R. China.
Publications dans "Cytochrome P-450 CYP2C9" :
2 publications dans cette catégorie
Affiliations :
Department of Pharmacotherapy and Translational Research, Center for Pharmacogenomics and Precision Medicine, University of Florida, Gainesville, Florida, USA.
Publications dans "Cytochrome P-450 CYP2C9" :
2 publications dans cette catégorie
Affiliations :
Federal University of Sao Joao del-Rei, Av. Sebastiao Goncalves Coelho, 400, Campus Centro-Oeste, Chanadour, Divinopolis-MG, CEP: 35501-296, Brazil.
Federal University of Minas Gerais, Av. Presidente Antonio Carlos, 667, Campus Pampulha, Belo Horizonte-MG, CEP: 31270-901, Brazil.
Publications dans "Cytochrome P-450 CYP2C9" :
2 publications dans cette catégorie
Affiliations :
Federal University of Sao Joao del-Rei, Av. Sebastiao Goncalves Coelho, 400, Campus Centro-Oeste, Chanadour, Divinopolis-MG, CEP: 35501-296, Brazil.
Publications dans "Cytochrome P-450 CYP2C9" :
2 publications dans cette catégorie
Affiliations :
Federal University of Sao Joao del-Rei, Av. Sebastiao Goncalves Coelho, 400, Campus Centro-Oeste, Chanadour, Divinopolis-MG, CEP: 35501-296, Brazil.
Publications dans "Cytochrome P-450 CYP2C9" :
2 publications dans cette catégorie
Affiliations :
Federal University of Sao Joao del-Rei, Av. Sebastiao Goncalves Coelho, 400, Campus Centro-Oeste, Chanadour, Divinopolis-MG, CEP: 35501-296, Brazil.
Publications dans "Cytochrome P-450 CYP2C9" :
2 publications dans cette catégorie
Affiliations :
Drug Resistance Research Group, Institute of Molecular Life Sciences, Research Centre for Natural Sciences, HUN-REN, Budapest, Hungary.
Doctoral School of Biology, Institute of Biology, Eötvös Loránd University, Budapest, Hungary.
Publications dans "Cytochrome P-450 CYP2C9" :
2 publications dans cette catégorie
Affiliations :
Institute of Microbiology of the Czech Academy of Sciences, Prague, Czech Republic.
Publications dans "Cytochrome P-450 CYP2C9" :
2 publications dans cette catégorie
Affiliations :
Drug Resistance Research Group, Institute of Molecular Life Sciences, Research Centre for Natural Sciences, HUN-REN, Budapest, Hungary.
Publications dans "Cytochrome P-450 CYP2C9" :
Casein kinase CK2 is a highly conserved serine/threonine protein kinase and exists in all eukaryotes. It has been demonstrated to be widely involved in the biological processes of plants. The CK2 holo...
Casein kinase 2 (CK2) is a ubiquitous, highly pleiotropic serine-threonine kinase. CK2 has been identified as a potential drug target for the treatment of cancer and related disorders. Several adenosi...
Chronic myelogenous leukemia (CML) is a myeloproliferative disease characterized by the BCR-ABL oncogene. Despite the high performance of treatment with tyrosine kinase inhibitors (TKI), about 30% of ...
DDX RNA helicases promote RNA processing, but DDX3X also activates casein kinase 1 (CK1ε). We show that other DDX proteins also stimulate the protein kinase activity of CK1ε and that this extends to c...
BCL-2 family proteins are frequently aberrantly expressed in mantle cell lymphoma (MCL). Recently, the BCL-2-specific inhibitor venetoclax has been approved by the US Food and Drug Administration for ...
Tumor cell extravasation across endothelial barrier has been recognized as a pivotal event in orchestrating metastasis formation. This event is initiated by the interactions of extravasating tumor cel...
Resistance to therapy commonly develops in patients with high-grade serous ovarian carcinoma (HGSC) and triple-negative breast cancer (TNBC), urging the search for improved therapeutic combinations an...
Accumulating evidence shows that high expression of casein kinase 2 (CK2) and phosphorylated acetyl CoA carboxylase (pACC) in patients with squamous cell carcinoma of the head and neck (SCCHN) correla...
Three aggressive SCCHN cell lines (OSC-19, FaDu and HN31) were cultured to investigate the anticancer mechanism of the CK2 inhibitor, CX-4945. Cell cycle analysis, Annexin V/PI staining, and cleavage ...
Cellular metabolism was impeded by CX-4945 in aggressive SCCHN cells by Seahorse XF24 Extracellular Flux Analyzer and mass spectrometry, and consequently time- and dose-dependent lipid droplet accumul...
The findings demonstrate that CK2 inhibition impairs normal cellular energy metabolism and may be an attractive therapy for treating aggressive SCCHN....
Triple-negative breast cancer (TNBC) is an aggressive malignancy that requires effective targeted drug therapy. In this study, we employed in silico methods to evaluate the efficacy of seven approved ...
Cisplatin is a platinum agent used in the treatment of non-small cell lung cancer (NSCLC). Much remains unknown regarding the basic operative mechanisms underlying cisplatin resistance in NSCLC. In th...